New arylpiperazine derivatives with high affinity for α1A, D2 and 5-HT2A receptors

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 2, 2003, Pages 175-178

  Gonzalez Gomez J C ^a   Santana, L ^a   Uriarte, E ^a   Brea, J ^a   Villazon M ^a   Loza, M I ^a   De Luca, M ^a,b   Rivas, M E ^a   Montenegro, G Y ^a   Fontenla, J A ^a  

^a UNIVERSITY OF SANTIAGO DE COMPOSTELA   (Spain)

^b UNIVERSITY OF CAGLIARI   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

ALPHA 1A ADRENERGIC RECEPTOR; COUMARIN; DOPAMINE 2 RECEPTOR; HALOPERIDOL; PIPERAZINE DERIVATIVE; SEROTONIN 2A RECEPTOR; ADRENERGIC RECEPTOR ALPHA(1A); ALPHA 1 ADRENERGIC RECEPTOR; COUMARIN DERIVATIVE; DOPAMINE RECEPTOR BLOCKING AGENT; DYES, REAGENTS, INDICATORS, MARKERS AND BUFFERS; SEROTONIN RECEPTOR;

ARTICLE; BINDING AFFINITY; DRUG SYNTHESIS; ALGORITHM; ANIMAL; CHEMISTRY; DRUG EFFECT; IN VITRO STUDY; MALE; RAT; SPRAGUE DAWLEY RAT; STRUCTURE ACTIVITY RELATION; SYNTHESIS; THORACIC AORTA; VASCULAR SMOOTH MUSCLE;

ALGORITHMS; ANIMALS; AORTA, THORACIC; COUMARINS; DOPAMINE ANTAGONISTS; HALOPERIDOL; INDICATORS AND REAGENTS; MALE; MUSCLE, SMOOTH, VASCULAR; PIPERAZINES; RATS; RATS, SPRAGUE-DAWLEY; RECEPTOR, SEROTONIN, 5-HT2A; RECEPTORS, ADRENERGIC, ALPHA-1; RECEPTORS, DOPAMINE D2; RECEPTORS, SEROTONIN; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 17944395201     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(02)00933-2     Document Type: Article

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