Long-lasting inhibitory effect of apple and orange juices, but not grapefruit juice, on OATP2B1-mediated drug absorption

Drug Metabolism and Disposition

Volumn 41, Issue 3, 2013, Pages 615-621

  Shirasaka, Yoshiyuki ^a   Shichiri, Megumi ^a   Murata, Yukiko ^a   Mori, Takanori ^a   Nakanishi, Takeo ^a   Tamai, Ikumi ^a  

^a KANAZAWA UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

ESTRONE SULFATE; FEXOFENADINE; ORGANIC ANION TRANSPORTER 2; ORGANIC ANION TRANSPORTING PROTEIN 2B1; UNCLASSIFIED DRUG;

ANIMAL CELL; APPLE JUICE; ARTICLE; COMPETITIVE INHIBITION; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG ABSORPTION; DRUG TRANSPORT; DRUG UPTAKE; FOOD DRUG INTERACTION; GRAPEFRUIT JUICE; IC 50; IN VITRO STUDY; NONHUMAN; OOCYTE; ORANGE JUICE; PRIORITY JOURNAL; XENOPUS;

ABSORPTION; ANIMALS; BEVERAGES; BINDING SITES; BINDING, COMPETITIVE; BIOLOGICAL TRANSPORT; CITRUS PARADISI; CITRUS SINENSIS; ESTRONE; FOOD-DRUG INTERACTIONS; FRUIT; KINETICS; MALUS; OOCYTES; ORGANIC ANION TRANSPORTERS; TERFENADINE; XENOPUS LAEVIS;

EID: 84874071287     PISSN: 00909556     EISSN: 1521009X     Source Type: Journal    
DOI: 10.1124/dmd.112.049635     Document Type: Article

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