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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 3, 2013, Pages 839-843

Selective inhibitors and tailored activity probes for lipoprotein- associated phospholipase A2

(15) Nagano, Joseph M G a Hsu, Ku Lung a Whitby, Landon R a Niphakis, Micah J a Speers, Anna E a Brown, Steven J a Spicer, Timothy b Fernandez Vega, Virneliz b Ferguson, Jill a Hodder, Peter b Srinivasan, Prabhavathi c Gonzalez, Tara D c Rosen, Hugh a Bahnson, Brian J c Cravatt, Benjamin F a

a SCRIPPS RESEARCH INSTITUTE (United States)

b SCRIPPS RESEARCH INSTITUTE (United States)

c UNIVERSITY OF DELAWARE (United States)

Author keywords

Inhibitor; Phospholipase; Proteomics; Screening

Indexed keywords

DARAPLADIB; PHOSPHOLIPASE A2;

ANIMAL CELL; ARTICLE; BRAIN MEMBRANE; CONCENTRATION (PARAMETERS); HUMAN; HUMAN CELL; IC 50; MOLECULAR PROBE; MOLECULAR WEIGHT; NONHUMAN; PHASE 3 CLINICAL TRIAL (TOPIC); PROSTATE CANCER;

1-ALKYL-2-ACETYLGLYCEROPHOSPHOCHOLINE ESTERASE; ANIMALS; BENZALDEHYDES; CARBAMATES; CELL LINE, TUMOR; ENZYME INHIBITORS; HUMANS; MICE; MOLECULAR STRUCTURE; OXIMES; PIPERAZINES; QUINOLINES;

EID: 84872302269 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.11.061 Document Type: Article

Times cited : (27)

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