Studies on chemical-structure modification and structure-activity relationship of gambogic acid derivatives at carbon(34)

Chemistry and Biodiversity

Volumn 9, Issue 10, 2012, Pages 2295-2308

  Zhang, Xiao Jin ^a   Li, Xiang ^a   Yang, Ying Rui ^a   Sun, Hao Peng ^a   Gao, Yuan ^a   Zhang, Lei ^a   Wang, Jin Xin ^a   Guo, Qing Long ^a   You, Qi Dong ^a  

^a CHINA PHARMACEUTICAL UNIVERSITY   (China)

Author keywords

Antitumor activity; Gambogic acid derivatives; Structure activity relationship (SAR)

Indexed keywords

ALIPHATIC AMINE; AMINE; ANTINEOPLASTIC AGENT; CARBON; GAMBOGIC ACID; GAMBOGIC ACID DERIVATIVE; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; ARTICLE; BREAST CARCINOMA; CANCER CELL CULTURE; CELL STRAIN A 549; CELL STRAIN BGC 823; CELL STRAIN HEPG2; CELL STRAIN MB 231; CELL STRAIN U 251; CHEMICAL MODIFICATION; CONTROLLED STUDY; CYTOTOXICITY; DRUG POTENCY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; GLIOMA; HUMAN; HUMAN CELL; HYDROPHILICITY; IC 50; LIVER CELL CARCINOMA; LUNG CANCER; MITOSIS INHIBITION; STOMACH CARCINOMA; STRUCTURE ACTIVITY RELATION;

ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CELL PROLIFERATION; DRUG SCREENING ASSAYS, ANTITUMOR; HEP G2 CELLS; HUMANS; STRUCTURE-ACTIVITY RELATIONSHIP; XANTHONES;

EID: 84867801406     PISSN: 16121872     EISSN: 16121880     Source Type: Journal    
DOI: 10.1002/cbdv.201200081     Document Type: Article

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