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Bioorganic and Medicinal Chemistry

Volumn 20, Issue 17, 2012, Pages 5094-5102

A novel thiazolidine compound induces caspase-9 dependent apoptosis in cancer cells

(5) Onen Bayram, F Esra b Durmaz, Irem a Scherman, Daniel c Herscovici, Jean c Cetin Atalay, Rengul a

a BILKENT UNIVERSITY (Turkey)

b YEDITEPE UNIVERSITY (Turkey)

c Centre National de la Recherche Scientifique (France)

Author keywords

Apoptosis; Cancer; Caspase 9; Cytotoxic; Terminal alkyne; Thiazolidine

Indexed keywords

2 PHENYL 3 PROPIONYL THIAZOLIDINE 4 CARBOXYLIC ACID ETHYL ESTER; 2 PHENYL 4 THIAZOLIDINECARBOXYLIC ACID; 2 PHENYLTHIAZOLIDINE 4 CARBOXYLIC ACID ETHYL ESTER; ALC 67; ANTINEOPLASTIC AGENT; CAMPTOTHECIN; CASPASE 9; DEATH RECEPTOR; FLUOROURACIL; THIAZOLIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; APOPTOSIS; ARTICLE; BREAST CANCER; CANCER CELL CULTURE; CELL CYCLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG CYTOTOXICITY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; DRUG TRANSFORMATION; ENDOMETRIUM CANCER; ENZYME ACTIVATION; ENZYME ACTIVITY; ENZYME INDUCTION; G1 PHASE CELL CYCLE CHECKPOINT; HUMAN; HUMAN CELL; IC 50; IN VITRO STUDY; LIVER CANCER; MOLECULAR LIBRARY; STRUCTURE ACTIVITY RELATION;

ANTINEOPLASTIC AGENTS; APOPTOSIS; CASPASE 9; CELL LINE, TUMOR; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG SCREENING ASSAYS, ANTITUMOR; HUMANS; NEOPLASMS; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLIDINES;

EID: 84864976797 PISSN: 09680896 EISSN: 14643391 Source Type: Journal
DOI: 10.1016/j.bmc.2012.07.016 Document Type: Article

Times cited : (43)

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