Thieno[3,2-b]thiophene-2-carboxylic acid derivatives as GPR35 agonists

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 12, 2012, Pages 4148-4152

  Deng, Huayun ^a   Hu, Jieyu ^a   Hu, Haibei ^a   He, Mingqian ^a   Fang, Ye ^a  

^a Corning Inc ^*  (United States)

Author keywords

Agonists; GPR35; Thieno 3,2 b thiophene 2 carboxylic acid

Indexed keywords

BETA ARRESTIN; CARBOXYLIC ACID DERIVATIVE;

ARTICLE; BIOLOGY; DRUG EFFICACY; DRUG POTENCY; GENE TRANSLOCATION; MOLECULAR PROBE; PHYSIOLOGY;

ANTI-INFLAMMATORY AGENTS; ARRESTINS; BIOLOGICAL ASSAY; DOSE-RESPONSE RELATIONSHIP, DRUG; HT29 CELLS; HUMANS; LIGANDS; PROTEIN TRANSPORT; RECEPTORS, G-PROTEIN-COUPLED; RECOMBINANT FUSION PROTEINS; SIGNAL TRANSDUCTION; STRUCTURE-ACTIVITY RELATIONSHIP; THIOPHENES;

EID: 84861577281     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2012.04.057     Document Type: Article

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