Discovery of natural phenols as G protein-coupled receptor-35 (GPR35) agonists

ACS Medicinal Chemistry Letters

Volumn 3, Issue 2, 2012, Pages 165-169

  Deng, Huayun ^a   Hu, Haibei ^a   Ling, Shizhang ^a   Ferrie, Ann M ^a   Fang, Ye ^a  

^a Science and Technology Division   (United States)

Author keywords

biased agonism; ellagic acid; GPR35; natural phenols

Indexed keywords

7 DESHYDROXYPYROGALLIN 4 CARBOXYLIC ACID; ALPHA CYANO 4 HYDROXYCINNAMIC ACID; APIGENIN; BAICALEIN; BETA ARRESTIN; CARBOXYLIC ACID DERIVATIVE; CHRYSIN; DIOSMETIN; ELLAGIC ACID; FLAVONE DERIVATIVE; G PROTEIN COUPLED RECEPTOR; G PROTEIN COUPLED RECEPTOR 35; HEMATEST; HIERACIN; LACCACID ACID A; LAPACHOL; LOBARIC ACID; LUTEOLIN; MORIN; MYRICETIN; NATURAL PRODUCT; NIFLUMIC ACID; PHENOL DERIVATIVE; PRIMULETIN; PROTEIN INHIBITOR; QUERCETIN; SPB 05142; UNCLASSIFIED DRUG; YE 210; ZAPRINST;

ARTICLE; CONTROLLED STUDY; DRUG DESIGN; DRUG DETERMINATION; DRUG RECEPTOR BINDING; DRUG TARGETING; HUMAN; HUMAN CELL; IMMUNOASSAY; LABELING INDEX; MOLECULAR DYNAMICS; PHARMACOLOGICAL PARAMETERS; PRIORITY JOURNAL; PROTEIN TRANSPORT; STRUCTURE ACTIVITY RELATION;

EID: 84856898821     PISSN: None     EISSN: 19485875     Source Type: Journal    
DOI: 10.1021/ml2003058     Document Type: Article

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