SCOPUS 정보 검색 플랫폼

Tetrahedron Letters

Volumn 53, Issue 24, 2012, Pages 3052-3055

Asymmetric synthesis of (-)-(R)-sitagliptin

(5) Davies, Stephen G a Fletcher, Ai M a Lv, Linlu a Roberts, Paul M a Thomson, James E a

a UNIVERSITY OF OXFORD (United Kingdom)

Author keywords

Asymmetric synthesis; Conjugate addition; Lithium amide; Sitagliptin

Indexed keywords

BETA AMINO ACID; ESTER; LITHIUM; SITAGLIPTIN; TRIAZOLOPYRIDAZINE DERIVATIVE;

ARTICLE; ASYMMETRIC SYNTHESIS; CATALYSIS; DIASTEREOSELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; HYDROGENOLYSIS; HYDROLYSIS; STEREOCHEMISTRY;

EID: 84861188112 PISSN: 00404039 EISSN: 18733581 Source Type: Journal
DOI: 10.1016/j.tetlet.2012.04.025 Document Type: Article

Times cited : (38)

References (58)

1
- 80053052228
- K. Mikami, S. Fuestero, M. Sánchez-Roselló, J.L. Aceña, V. Soloshonok, and A. Sorochinsky Synthesis 2011 3045
- (2011) Synthesis , pp. 3045
- Mikami, K.¹ Fuestero, S.² Sánchez-Roselló, M.³ Aceña, J.L.⁴ Soloshonok, V.⁵ Sorochinsky, A.⁶

2
- 85127635914
- CRC Press Boca Raton
- M. Suffness Taxol: Science and Applications 1995 CRC Press Boca Raton
- (1995) Taxol: Science and Applications
- Suffness, M.¹

3
- 0031040149
- E.K. Rowinsky Ann. Rev. Med. 48 1997 353
- (1997) Ann. Rev. Med. , vol.48 , pp. 353
- Rowinsky, E.K.¹

4
- 0000052734
- D. Guénard, F. Guéritte-Vogelein, and P. Potier Acc. Chem. Res. 26 1993 160
- (1993) Acc. Chem. Res. , vol.26 , pp. 160
- Guénard, D.¹ Guéritte-Vogelein, F.² Potier, P.³

5
- 0031390567
- K. Uoto, S. Ohsuki, H. Takenoshita, T. Ishiyama, S. Iimura, Y. Hirota, I. Mitsui, T. Hirofumi, and T. Soga Chem. Pharm. Bull. 45 1997 1793
- (1997) Chem. Pharm. Bull. , vol.45 , pp. 1793
- Uoto, K.¹ Ohsuki, S.² Takenoshita, H.³ Ishiyama, T.⁴ Iimura, S.⁵ Hirota, Y.⁶ Mitsui, I.⁷ Hirofumi, T.⁸ Soga, T.⁹

6
- 0031023523
- I. Ojima, J.C. Slater, P. Perea, J.M. Vieth, A. Abouabdellah, J.-P. Bégué, and R.J. Bernacki Bioorg. Med. Chem. Lett. 7 1997 133
- (1997) Bioorg. Med. Chem. Lett. , vol.7 , pp. 133
- Ojima, I.¹ Slater, J.C.² Perea, P.³ Vieth, J.M.⁴ Abouabdellah, A.⁵ Bégué, J.-P.⁶ Bernacki, R.J.⁷

7
- 0033590281
- I. Ojima, T. Wang, M. Miller, S. Lin, C.P. Borella, P. Pera, and R.J. Bernacki Bioorg. Med. Chem. Lett. 9 1999 3423
- (1999) Bioorg. Med. Chem. Lett. , vol.9 , pp. 3423
- Ojima, I.¹ Wang, T.² Miller, M.³ Lin, S.⁴ Borella, C.P.⁵ Pera, P.⁶ Bernacki, R.J.⁷

8
- 0033948409
- I. Ojima, S. Lin, J.C. Slater, T. Wang, P. Tera, R.J. Bernacki, C. Ferlini, and G. Scambia Bioorg. Med. Chem. 8 2000 1619
- (2000) Bioorg. Med. Chem. , vol.8 , pp. 1619
- Ojima, I.¹ Lin, S.² Slater, J.C.³ Wang, T.⁴ Tera, P.⁵ Bernacki, R.J.⁶ Ferlini, C.⁷ Scambia, G.⁸

9
- 0032859102
- I. Ojima, S. Lin, and T. Wang Curr. Med. Chem. 6 1999 927
- (1999) Curr. Med. Chem. , vol.6 , pp. 927
- Ojima, I.¹ Lin, S.² Wang, T.³

10
- 2342504474
- L. Kuznetsova, I.M. Ungureanu, A. Pepe, I. Zanardi, X. Wu, and I. Ojima J. Fluorine Chem. 125 2004 487
- (2004) J. Fluorine Chem. , vol.125 , pp. 487
- Kuznetsova, L.¹ Ungureanu, I.M.² Pepe, A.³ Zanardi, I.⁴ Wu, X.⁵ Ojima, I.⁶

11
- 84861197952
- The phosphate monohydrate salt of (-)-(R)-sitagliptin 1 is marketed under the name of JANUVIA™
- The phosphate monohydrate salt of (-)-(R)-sitagliptin 1 is marketed under the name of JANUVIA™.

12
- 19944427998
- D. Kim, L. Wang, M. Beconi, G.J. Eiermann, M.H. Fisher, H. He, G.J. Hickey, J.E. Kowalchick, B. Leiting, K. Lyons, F. Marsilio, M.E. McCann, R.A. Patel, A. Petrov, G. Scapin, S.B. Patel, R.S. Roy, J.K. Wu, M.J. Wyvratt, B.B. Zhang, L. Zhu, N.A. Thornberry, and A.E. Wever J. Med. Chem. 48 2005 141
- (2005) J. Med. Chem. , vol.48 , pp. 141
- Kim, D.¹ Wang, L.² Beconi, M.³ Eiermann, G.J.⁴ Fisher, M.H.⁵ He, H.⁶ Hickey, G.J.⁷ Kowalchick, J.E.⁸ Leiting, B.⁹ Lyons, K.¹⁰ Marsilio, F.¹¹ McCann, M.E.¹² Patel, R.A.¹³ Petrov, A.¹⁴ Scapin, G.¹⁵ Patel, S.B.¹⁶ Roy, R.S.¹⁷ Wu, J.K.¹⁸ Wyvratt, M.J.¹⁹ Zhang, B.B.²⁰ more..

13
- 33947690115
- N.A. Thornberry, and A.E. Weber Curr. Top. Med. Chem. 7 2007 557
- (2007) Curr. Top. Med. Chem. , vol.7 , pp. 557
- Thornberry, N.A.¹ Weber, A.E.²

14
- 79951914183
- A.A. Desai Angew. Chem., Int. Ed. 50 2011 1974
- (2011) Angew. Chem., Int. Ed. , vol.50 , pp. 1974
- Desai, A.A.¹

15
- 77954797329
- C.K. Savile, J.M. Janey, E.C. Mundorff, J.C. Moore, S. Tam, W.R. Jarvis, J.C. Colbeck, A. Krebber, F.J. Fleitz, and J. Brands Science 329 2010 305
- (2010) Science , vol.329 , pp. 305
- Savile, C.K.¹ Janey, J.M.² Mundorff, E.C.³ Moore, J.C.⁴ Tam, S.⁵ Jarvis, W.R.⁶ Colbeck, J.C.⁷ Krebber, A.⁸ Fleitz, F.J.⁹ Brands, J.¹⁰

16
- 33746916498
- A.M. Clausen, B. Dziadul, K.L. Cappuccio, M. Kaba, C. Starbuck, Y. Hsiao, and T. Dowling Org. Process Res. Dev. 10 2006 723
- (2006) Org. Process Res. Dev. , vol.10 , pp. 723
- Clausen, A.M.¹ Dziadul, B.² Cappuccio, K.L.³ Kaba, M.⁴ Starbuck, C.⁵ Hsiao, Y.⁶ Dowling, T.⁷

17
- 67649583302
- K.B. Hansen, Y. Hsiao, F. Zu, N. Rivera, A. Clausen, M. Kubryk, S. Krska, T. Rosner, B. Simmons, J. Balsells, N. Ikemoto, Y. Sun, F. Spindler, C. Malan, E.J.J. Grabowski, and J.D. Armstrong III J. Am. Chem. Soc. 131 2009 8798
- (2009) J. Am. Chem. Soc. , vol.131 , pp. 8798
- Hansen, K.B.¹ Hsiao, Y.² Zu, F.³ Rivera, N.⁴ Clausen, A.⁵ Kubryk, M.⁶ Krska, S.⁷ Rosner, T.⁸ Simmons, B.⁹ Balsells, J.¹⁰ Ikemoto, N.¹¹ Sun, Y.¹² Spindler, F.¹³ Malan, C.¹⁴ Grabowski, E.J.J.¹⁵ Armstrong Iii, J.D.¹⁶

18
- 70349989935
- L.L. Zeng, Y.J. Ding, G.C. Zhang, H.R. Song, and W.H. Hu Chin. Chem. Lett. 20 2009 1397
- (2009) Chin. Chem. Lett. , vol.20 , pp. 1397
- Zeng, L.L.¹ Ding, Y.J.² Zhang, G.C.³ Song, H.R.⁴ Hu, W.H.⁵

19
- 84861184076
- F. Te, R.X. Gao, N. Shen, and Z.X. Ding Chin. J. Synth. Chem. 18 2010 767
- (2010) Chin. J. Synth. Chem. , vol.18 , pp. 767
- Te, F.¹ Gao, R.X.² Shen, N.³ Ding, Z.X.⁴

20
- 26444512112
- K.B. Hansen, J. Balsells, S. Dreher, Y. Hsiao, M. Kubryk, M. Palucki, N. Rivera, D. Steinhuebel, J.D. Armstrong III, D. Askin, and E.J.J. Grabowski Org. Process Res. Dev. 9 2005 634
- (2005) Org. Process Res. Dev. , vol.9 , pp. 634
- Hansen, K.B.¹ Balsells, J.² Dreher, S.³ Hsiao, Y.⁴ Kubryk, M.⁵ Palucki, M.⁶ Rivera, N.⁷ Steinhuebel, D.⁸ Armstrong Iii, J.D.⁹ Askin, D.¹⁰ Grabowski, E.J.J.¹¹

21
- 77952757399
- One synthesis of (-)-(R)-sitagliptin 1 employs our diastereoselective lithium amide conjugate addition methodology, see
- One synthesis of (-)-(R)-sitagliptin 1 employs our diastereoselective lithium amide conjugate addition methodology, see: F. Liu, W. Yu, W. Ou, X. Wang, L. Ruan, Y. Li, X. Peng, X. Tao, and X. Pan J. Chem. Res. 34 2010 230
- (2010) J. Chem. Res. , vol.34 , pp. 230
- Liu, F.¹ Yu, W.² Ou, W.³ Wang, X.⁴ Ruan, L.⁵ Li, Y.⁶ Peng, X.⁷ Tao, X.⁸ Pan, X.⁹

22
- 68849088073
- D. Steinhuebel, Y. Sun, K. Matsumura, N. Sayo, and T. Saito J. Am. Chem. Soc. 131 2009 11316
- (2009) J. Am. Chem. Soc. , vol.131 , pp. 11316
- Steinhuebel, D.¹ Sun, Y.² Matsumura, K.³ Sayo, N.⁴ Saito, T.⁵

23
- 0025818883
- S.G. Davies, and O. Ichihara Tetrahedron: Asymmetry 2 1991 183
- (1991) Tetrahedron: Asymmetry , vol.2 , pp. 183
- Davies, S.G.¹ Ichihara, O.²

24
- 33746456336
- S.G. Davies, N.M. Garrido, D. Kruchinin, O. Ichihara, L.J. Kotchie, P.D. Price, A.J. Price Mortimer, A.J. Russell, and A. Smith D Tetrahedron: Asymmetry 17 2006 1793
- (2006) Tetrahedron: Asymmetry , vol.17 , pp. 1793
- Davies, S.G.¹ Garrido, N.M.² Kruchinin, D.³ Ichihara, O.⁴ Kotchie, L.J.⁵ Price, P.D.⁶ Price Mortimer, A.J.⁷ Russell, A.J.⁸ Smith, A.⁹

25
- 65549099060
- S.G. Davies, R.L. Nicholson, P.D. Price, P.M. Roberts, A.J. Russell, E.D. Savory, A.D. Smith, and J. Thomson E Tetrahedron: Asymmetry 20 2009 758
- (2009) Tetrahedron: Asymmetry , vol.20 , pp. 758
- Davies, S.G.¹ Nicholson, R.L.² Price, P.D.³ Roberts, P.M.⁴ Russell, A.J.⁵ Savory, E.D.⁶ Smith, A.D.⁷ Thomson, J.⁸

26
- 67650487269
- S.G. Davies, A.C. Garner, R.L. Nicholson, J. Osborne, P.M. Roberts, E.D. Savory, A.D. Smith, and J.E. Thomson Org. Biomol. Chem. 7 2009 2604
- (2009) Org. Biomol. Chem. , vol.7 , pp. 2604
- Davies, S.G.¹ Garner, A.C.² Nicholson, R.L.³ Osborne, J.⁴ Roberts, P.M.⁵ Savory, E.D.⁶ Smith, A.D.⁷ Thomson, J.E.⁸

27
- 84861187029
- S.G. Davies, N. Mujtaba, P.M. Roberts, A.D. Smith, and J.E. Thomson Org. Lett. 2009 1959 11
- (1959) Org. Lett. , vol.2009 , pp. 11
- Davies, S.G.¹ Mujtaba, N.² Roberts, P.M.³ Smith, A.D.⁴ Thomson, J.E.⁵

28
- 77953121876
- S.A. Bentley, S.G. Davies, J.A. Lee, P.M. Roberts, A.J. Russell, J.E. Thomson, and S.M. Toms Tetrahedron 66 2010 4604
- (2010) Tetrahedron , vol.66 , pp. 4604
- Bentley, S.A.¹ Davies, S.G.² Lee, J.A.³ Roberts, P.M.⁴ Russell, A.J.⁵ Thomson, J.E.⁶ Toms, S.M.⁷

29
- 77956266204
- E. Abraham, C.W. Bailey, T.D.W. Claridge, S.G. Davies, K.B. Ling, B. Odell, T.L. Rees, P.M. Roberts, A.J. Russell, A.D. Smith, L.J. Smith, H.R. Storr, M.J. Sweet, A.L. Thompson, J.E. Thomson, G.E. Tranter, and D.J. Watkin Tetrahedron: Asymmetry 21 2010 1797
- (2010) Tetrahedron: Asymmetry , vol.21 , pp. 1797
- Abraham, E.¹ Bailey, C.W.² Claridge, T.D.W.³ Davies, S.G.⁴ Ling, K.B.⁵ Odell, B.⁶ Rees, T.L.⁷ Roberts, P.M.⁸ Russell, A.J.⁹ Smith, A.D.¹⁰ Smith, L.J.¹¹ Storr, H.R.¹² Sweet, M.J.¹³ Thompson, A.L.¹⁴ Thomson, J.E.¹⁵ Tranter, G.E.¹⁶ Watkin, D.J.¹⁷

30
- 79951810622
- E. Abraham, T.D.W. Claridge, S.G. Davies, B. Odell, P.M. Roberts, A.J. Russell, A.D. Smith, L.J. Smith, H.R. Storr, M.J. Sweet, A.L. Thompson, J.E. Thomson, G.E. Tranter, and D.J. Watkin Tetrahedron: Asymmetry 22 2011 69
- (2011) Tetrahedron: Asymmetry , vol.22 , pp. 69
- Abraham, E.¹ Claridge, T.D.W.² Davies, S.G.³ Odell, B.⁴ Roberts, P.M.⁵ Russell, A.J.⁶ Smith, A.D.⁷ Smith, L.J.⁸ Storr, H.R.⁹ Sweet, M.J.¹⁰ Thompson, A.L.¹¹ Thomson, J.E.¹² Tranter, G.E.¹³ Watkin, D.J.¹⁴

31
- 79953165403
- E.A. Brock, S.G. Davies, J.A. Lee, P.M. Roberts, and J.E. Thomson Org. Lett. 13 2011 1594
- (2011) Org. Lett. , vol.13 , pp. 1594
- Brock, E.A.¹ Davies, S.G.² Lee, J.A.³ Roberts, P.M.⁴ Thomson, J.E.⁵

32
- 79953165311
- S.K. Bagal, S.G. Davies, A.M. Fletcher, J.A. Lee, P.M. Roberts, P.M. Scott, and J.E. Thomson Tetrahedron Lett. 52 2011 2216
- (2011) Tetrahedron Lett. , vol.52 , pp. 2216
- Bagal, S.K.¹ Davies, S.G.² Fletcher, A.M.³ Lee, J.A.⁴ Roberts, P.M.⁵ Scott, P.M.⁶ Thomson, J.E.⁷

33
- 0036070055
- For selected examples from this laboratory, see
- For selected examples from this laboratory, see: S.G. Davies, K. Iwamoto, C.A.P. Smethurst, A.D. Smith, and H. Rodríguez-Solla Synlett 2002 1146
- (2002) Synlett , pp. 1146
- Davies, S.G.¹ Iwamoto, K.² Smethurst, C.A.P.³ Smith, A.D.⁴ Rodríguez-Solla, H.⁵

34
- 0042736307
- S.G. Davies, R.J. Kelly, and A.J. Price Mortimer Chem. Commun. 2003 2132
- (2003) Chem. Commun. , pp. 2132
- Davies, S.G.¹ Kelly, R.J.² Price Mortimer, A.J.³

35
- 2542446198
- S.G. Davies, A.J. Burke, A.C. Garner, T.D. McCarthy, P.M. Roberts, A.D. Smith, H. Rodríguez-Solla, and R.J. Vickers Org. Biomol. Chem. 2 2004 1387
- (2004) Org. Biomol. Chem. , vol.2 , pp. 1387
- Davies, S.G.¹ Burke, A.J.² Garner, A.C.³ McCarthy, T.D.⁴ Roberts, P.M.⁵ Smith, A.D.⁶ Rodríguez-Solla, H.⁷ Vickers, R.J.⁸

36
- 4744346531
- S.G. Davies, J.R. Haggitt, O. Ichihara, R.J. Kelly, M.A. Leech, A.J. Price Mortimer, P.M. Roberts, and A.D. Smith Org. Biomol. Chem. 2 2004 2630
- (2004) Org. Biomol. Chem. , vol.2 , pp. 2630
- Davies, S.G.¹ Haggitt, J.R.² Ichihara, O.³ Kelly, R.J.⁴ Leech, M.A.⁵ Price Mortimer, A.J.⁶ Roberts, P.M.⁷ Smith, A.D.⁸

37
- 36148970785
- E. Abraham, J.I. Candela-Lena, S.G. Davies, M. Georgiou, R.L. Nicholson, P.M. Roberts, A.J. Russell, E.M. Sánchez-Fernández, A.D. Smith, and J.E. Thomson Tetrahedron: Asymmetry 18 2007 2510
- (2007) Tetrahedron: Asymmetry , vol.18 , pp. 2510
- Abraham, E.¹ Candela-Lena, J.I.² Davies, S.G.³ Georgiou, M.⁴ Nicholson, R.L.⁵ Roberts, P.M.⁶ Russell, A.J.⁷ Sánchez-Fernández, E.M.⁸ Smith, A.D.⁹ Thomson, J.E.¹⁰

38
- 42349103981
- E. Abraham, S.G. Davies, N.L. Millican, R.L. Nicholson, P.M. Roberts, and A.D. Smith Org. Biomol. Chem. 6 2008 1655
- (2008) Org. Biomol. Chem. , vol.6 , pp. 1655
- Abraham, E.¹ Davies, S.G.² Millican, N.L.³ Nicholson, R.L.⁴ Roberts, P.M.⁵ Smith, A.D.⁶

39
- 42349111665
- E. Abraham, E.A. Brock, J.I. Candela-Lena, S.G. Davies, M. Georgiou, R.L. Nicholson, J.H. Perkins, P.M. Roberts, A.J. Russell, E.M. Sánchez- Fernández, P.M. Scott, A.D. Smith, and J.E. Thomson Org. Biomol. Chem. 6 2008 1665
- (2008) Org. Biomol. Chem. , vol.6 , pp. 1665
- Abraham, E.¹ Brock, E.A.² Candela-Lena, J.I.³ Davies, S.G.⁴ Georgiou, M.⁵ Nicholson, R.L.⁶ Perkins, J.H.⁷ Roberts, P.M.⁸ Russell, A.J.⁹ Sánchez-Fernández, E.M.¹⁰ Scott, P.M.¹¹ Smith, A.D.¹² Thomson, J.E.¹³

40
- 70350517426
- S.G. Davies, A.M. Fletcher, P.M. Roberts, and A.D. Smith Tetrahedron 65 2009 10192
- (2009) Tetrahedron , vol.65 , pp. 10192
- Davies, S.G.¹ Fletcher, A.M.² Roberts, P.M.³ Smith, A.D.⁴

41
- 79956160271
- S.A. Bentley, S.G. Davies, J.A. Lee, P.M. Roberts, and J.E. Thomson Org. Lett. 13 2011 2544
- (2011) Org. Lett. , vol.13 , pp. 2544
- Bentley, S.A.¹ Davies, S.G.² Lee, J.A.³ Roberts, P.M.⁴ Thomson, J.E.⁵

42
- 78649785647
- S.G. Davies, O. Ichihara, P.M. Roberts, and J.E. Thomson Tetrahedron 67 2011 216
- (2011) Tetrahedron , vol.67 , pp. 216
- Davies, S.G.¹ Ichihara, O.² Roberts, P.M.³ Thomson, J.E.⁴

43
- 80255133724
- S.G. Davies, A.M. Fletcher, D.G. Hughes, J.A. Lee, P.D. Price, P.M. Roberts, A.J. Russell, A.D. Smith, J.E. Thomson, and O.M.H. Williams Tetrahedron 67 2011 9975
- (2011) Tetrahedron , vol.67 , pp. 9975
- Davies, S.G.¹ Fletcher, A.M.² Hughes, D.G.³ Lee, J.A.⁴ Price, P.D.⁵ Roberts, P.M.⁶ Russell, A.J.⁷ Smith, A.D.⁸ Thomson, J.E.⁹ Williams, O.M.H.¹⁰

44
- 80255138674
- S.G. Davies, J.A. Lee, P.M. Roberts, J.E. Thomson, and C.J. West Tetrahedron Lett. 52 2011 6477
- (2011) Tetrahedron Lett. , vol.52 , pp. 6477
- Davies, S.G.¹ Lee, J.A.² Roberts, P.M.³ Thomson, J.E.⁴ West, C.J.⁵

45
- 80054898389
- S.G. Davies, R. Huckvale, T.J.A. Lorkin, P.M. Roberts, and J.E. Thomson Tetrahedron: Asymmetry 22 2011 1591
- (2011) Tetrahedron: Asymmetry , vol.22 , pp. 1591
- Davies, S.G.¹ Huckvale, R.² Lorkin, T.J.A.³ Roberts, P.M.⁴ Thomson, J.E.⁵

46
- 84862777443
- S.G. Davies, J.A. Lee, P.M. Roberts, J.P. Stonehouse, and J.E. Thomson Tetrahedron Lett. 53 2012 1119
- (2012) Tetrahedron Lett. , vol.53 , pp. 1119
- Davies, S.G.¹ Lee, J.A.² Roberts, P.M.³ Stonehouse, J.P.⁴ Thomson, J.E.⁵

47
- 36749051660
- For selected examples from this laboratory, see
- For selected examples from this laboratory, see: T. Cailleau, J.W.B. Cooke, S.G. Davies, K.B. Ling, A. Naylor, R.L. Nicholson, P.D. Price, P.M. Roberts, A.J. Russell, A.D. Smith, and J.E. Thomson Org. Biomol. Chem. 5 2007 3922
- (2007) Org. Biomol. Chem. , vol.5 , pp. 3922
- Cailleau, T.¹ Cooke, J.W.B.² Davies, S.G.³ Ling, K.B.⁴ Naylor, A.⁵ Nicholson, R.L.⁶ Price, P.D.⁷ Roberts, P.M.⁸ Russell, A.J.⁹ Smith, A.D.¹⁰ Thomson, J.E.¹¹

48
- 59949088993
- S.G. Davies, M.J. Durbin, E.C. Goddard, P.M. Kelly, W. Kurosawa, J.A. Lee, R.L. Nicholson, P.D. Price, P.M. Roberts, A.J. Russell, P.M. Scott, and A.D. Smith Org. Biomol. Chem. 7 2009 761
- (2009) Org. Biomol. Chem. , vol.7 , pp. 761
- Davies, S.G.¹ Durbin, M.J.² Goddard, E.C.³ Kelly, P.M.⁴ Kurosawa, W.⁵ Lee, J.A.⁶ Nicholson, R.L.⁷ Price, P.D.⁸ Roberts, P.M.⁹ Russell, A.J.¹⁰ Scott, P.M.¹¹ Smith, A.D.¹²

49
- 84862907535
- S.G. Davies, J.A. Lee, P.M. Roberts, J.E. Thomson, and J. Yin Org. Lett. 14 2012 218
- (2012) Org. Lett. , vol.14 , pp. 218
- Davies, S.G.¹ Lee, J.A.² Roberts, P.M.³ Thomson, J.E.⁴ Yin, J.⁵

50
- 23844435716
- For selected examples from this laboratory, see
- For selected examples from this laboratory, see: S.G. Davies, A.C. Garner, M.J.C. Long, R.M. Morrison, P.M. Roberts, A.D. Smith, M.J. Sweet, and J.M. Withey Org. Biomol. Chem. 3 2005 2762
- (2005) Org. Biomol. Chem. , vol.3 , pp. 2762
- Davies, S.G.¹ Garner, A.C.² Long, M.J.C.³ Morrison, R.M.⁴ Roberts, P.M.⁵ Smith, A.D.⁶ Sweet, M.J.⁷ Withey, J.M.⁸

51
- 44949122583
- Y. Aye, S.G. Davies, A.C. Garner, P.M. Roberts, A.D. Smith, and J.E. Thomson Org. Biomol. Chem. 6 2008 2195
- (2008) Org. Biomol. Chem. , vol.6 , pp. 2195
- Aye, Y.¹ Davies, S.G.² Garner, A.C.³ Roberts, P.M.⁴ Smith, A.D.⁵ Thomson, J.E.⁶

52
- 47049123681
- E. Abraham, S.G. Davies, A.J. Docherty, K.B. Ling, P.M. Roberts, A.J. Russell, J.E. Thomson, and S.M. Toms Tetrahedron: Asymmetry 19 2008 1356
- (2008) Tetrahedron: Asymmetry , vol.19 , pp. 1356
- Abraham, E.¹ Davies, S.G.² Docherty, A.J.³ Ling, K.B.⁴ Roberts, P.M.⁵ Russell, A.J.⁶ Thomson, J.E.⁷ Toms, S.M.⁸

53
- 59349090568
- S.G. Davies, M.J. Durbin, S.J.S. Hartman, A. Matsuno, P.M. Roberts, A.J. Russell, A.D. Smith, J.E. Thomson, and S.M. Toms Tetrahedron: Asymmetry 19 2008 2870
- (2008) Tetrahedron: Asymmetry , vol.19 , pp. 2870
- Davies, S.G.¹ Durbin, M.J.² Hartman, S.J.S.³ Matsuno, A.⁴ Roberts, P.M.⁵ Russell, A.J.⁶ Smith, A.D.⁷ Thomson, J.E.⁸ Toms, S.M.⁹

54
- 24344501374
- S.G. Davies, A.D. Smith, and P.D. Price Tetrahedron: Asymmetry 16 2005 2833
- (2005) Tetrahedron: Asymmetry , vol.16 , pp. 2833
- Davies, S.G.¹ Smith, A.D.² Price, P.D.³

55
- 59949097919
- T.D.W. Claridge, S.G. Davies, J.A. Lee, R.L. Nicholson, P.M. Roberts, A.J. Russell, A.D. Smith, and S.M. Toms Org. Lett. 10 2008 5437
- (2008) Org. Lett. , vol.10 , pp. 5437
- Claridge, T.D.W.¹ Davies, S.G.² Lee, J.A.³ Nicholson, R.L.⁴ Roberts, P.M.⁵ Russell, A.J.⁶ Smith, A.D.⁷ Toms, S.M.⁸

56
- 0034615694
- For example, selective mono-N-deprotection has been developed by our group, see
- For example, selective mono-N-deprotection has been developed by our group, see: S.D. Bull, S.G. Davies, G. Fenton, A.W. Mulvaney, R.S. Prasad, and A.D. Smith Chem. Commun. 2000 337
- (2000) Chem. Commun. , pp. 337
- Bull, S.D.¹ Davies, S.G.² Fenton, G.³ Mulvaney, A.W.⁴ Prasad, R.S.⁵ Smith, A.D.⁶

57
- 84861197947
- S.D. Bull, S.G. Davies, G. Fenton, A.W. Mulvaney, R.S. Prasad, and A.D. Smith J. Chem. Soc., Perkin Trans. 1 2000 3965
- (2000) J. Chem. Soc., Perkin Trans. 1 , pp. 3965
- Bull, S.D.¹ Davies, S.G.² Fenton, G.³ Mulvaney, A.W.⁴ Prasad, R.S.⁵ Smith, A.D.⁶

58
- 84861187025
- Triazolopyrazine 12 was prepared according to a literature procedure, see: Ref. 5a
- Triazolopyrazine 12 was prepared according to a literature procedure, see: Ref. 5a.

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.