A practical synthesis of trifluorophenyl R-amino acid: The key precursor for the new anti-diabetic drug sitagliptin

Chinese Chemical Letters

Volumn 20, Issue 12, 2009, Pages 1397-1399

  Zeng, Li Li ^a,b   Ding, Ying Jie ^a,b   Zhang, Gui Cheng ^a   Song, Hong Rui ^b   Hu, Wen Hui ^a  

^a GUANGZHOU INSTITUTES OF BIOMEDICINE AND HEALTH   (China)

^b SHENYANG PHARMACEUTICAL UNIVERSITY   (China)

Author keywords

Amino acid; DPP IV inhibitor; Practical synthesis; Sitagliptin

Indexed keywords

EID: 70349989935     PISSN: 10018417     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.cclet.2009.06.036     Document Type: Article

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