-
1
-
-
42549137051
-
Hormone abuse in sports: the antidoping perspective
-
O. Barroso, I. Mazzoni, and O. Rabin. Hormone abuse in sports: the antidoping perspective. Asian J.Androl. 10: 391-402 (2008).
-
(2008)
Asian J. Androl.
, vol.10
, pp. 391-402
-
-
Barroso, O.1
Mazzoni, I.2
Rabin, O.3
-
2
-
-
47749104941
-
New and old challenges of sports drug testing
-
F. Botrè. New and old challenges of sports drug testing. J.Mass. Spectrom. 43: 903-907 (2008).
-
(2008)
J. Mass. Spectrom.
, vol.43
, pp. 903-907
-
-
Botrè, F.1
-
3
-
-
84855702393
-
-
WADA. The 2009 WADA Prohibited List. (accessed April 2011)
-
WADA. The 2009 WADA Prohibited List. http://www.wadaama.org/rtecontent/document/2008_List_En.pdf (accessed April 2011).
-
-
-
-
4
-
-
84855710335
-
-
WADA. The 2009 WADA Laboratory Statistics. (accessed April 2011)
-
WADA. The 2009 WADA Laboratory Statistics. http://www.wada-ama.org/Documents/Science_Medicine/Anti-Doping_Laboratories/Lab_Statistics/WADA_2009_LaboratoryStatisticsReport_Final.pdf (accessed April 2011).
-
-
-
-
5
-
-
2942541820
-
Effects of androgenic-anabolic steroids in athletes
-
F. Hartgens and H. Kuipers. Effects of androgenic-anabolic steroids in athletes. Sports Med. 34: 513-554 (2004).
-
(2004)
Sports Med
, vol.34
, pp. 513-554
-
-
Hartgens, F.1
Kuipers, H.2
-
6
-
-
0036374401
-
Anabolic steroids
-
C. Kuhn. Anabolic steroids. Recent Prog. Horm. Res. 57: 411-434 (2002).
-
(2002)
Recent Prog. Horm. Res.
, vol.57
, pp. 411-434
-
-
Kuhn, C.1
-
7
-
-
13444306435
-
Pharmacoepidemiology of anabolic androgenic steroids: a review
-
I. Thiblin and A. Petersson. Pharmacoepidemiology of anabolic androgenic steroids: a review. Fundam. Clin. Pharmacol. 19: 27-44 (2005).
-
(2005)
Fundam. Clin. Pharmacol.
, vol.19
, pp. 27-44
-
-
Thiblin, I.1
Petersson, A.2
-
8
-
-
0034811303
-
A review of the chemistry, biological action, and clinical applications of anabolic-androgenic steroids
-
N.T. Shahidi. A review of the chemistry, biological action, and clinical applications of anabolic-androgenic steroids. Clin. Ther. 23: 1355-1390 (2001).
-
(2001)
Clin. Ther.
, vol.23
, pp. 1355-1390
-
-
Shahidi, N.T.1
-
9
-
-
3042542158
-
Tetrahydrogestrinone: discovery, synthesis, and detection in urine
-
D.H. Catlin, M.H. Sekera, B.D. Ahrens, B. Starcevic,Y.C. Chang, and C.K. Hatton. Tetrahydrogestrinone: discovery, synthesis, and detection in urine. Rapid Commun. Mass Spectrom. 18: 1245-1049 (2004).
-
(2004)
Rapid Commun. Mass Spectrom.
, vol.18
, pp. 1245-1049
-
-
Catlin, D.H.1
Sekera, M.H.2
Ahrens, B.D.3
Starcevic, B.4
Chang, Y.C.5
Hatton, C.K.6
-
10
-
-
1842434983
-
FDA warning on unapproved performance enhancer
-
FDA warning on unapproved performance enhancer. FDA Consum. 38: 4 (2004).
-
(2004)
FDA Consum
, vol.38
, pp. 4
-
-
-
11
-
-
1442357999
-
Doping by design
-
S. Ashley. Doping by design. Sci. Am. 290: 22-23 (2004).
-
(2004)
Sci. Am.
, vol.290
, pp. 22-23
-
-
Ashley, S.1
-
12
-
-
0642342092
-
Drugs in sport: no dope
-
J. Knight. Drugs in sport: no dope. Nature 426: 114-115 (2003).
-
(2003)
Nature
, vol.426
, pp. 114-115
-
-
Knight, J.1
-
13
-
-
3142599890
-
Athletes' "designer steroid" leads to widening scandal
-
W. Kondro. Athletes' "designer steroid" leads to widening scandal. Lancet 362: 1466 (2003).
-
(2003)
Lancet
, vol.362
, pp. 1466
-
-
Kondro, W.1
-
14
-
-
34547645017
-
Preventive doping control analysis: liquid and gas chromatography time-of-flight mass spectrometry for detection of designer steroids
-
C.G. Georgakopoulos, A. Vonaparti, M. Stamou, P. Kiousi, E. Lyris,Y.S. Angelis, G. Tsoupras, B.Wuest, M.W. Nielen, I. Panderi, and M. Koupparis. Preventive doping control analysis: liquid and gas chromatography time-of-flight mass spectrometry for detection of designer steroids. Rapid Commun. Mass Spectrom. 21: 2439-2446 (2007).
-
(2007)
Rapid Commun. Mass Spectrom.
, vol.21
, pp. 2439-2446
-
-
Georgakopoulos, C.G.1
Vonaparti, A.2
Stamou, M.3
Kiousi, P.4
Lyris, E.5
Angelis, Y.S.6
Tsoupras, G.7
Wuest, B.8
Nielen, M.W.9
Panderi, I.10
Koupparis, M.11
-
15
-
-
77952919521
-
Preventive doping control screening analysis of prohibited substances in human urine using rapid-resolution liquid chromatography/high-resolution time-of-flight mass spectrometry
-
A. Vonaparti, E. Lyris, Y.S. Angelis, I. Panderi, M. Koupparis, A. Tsantili-Kakoulidou, R.J. Peters, M.W. Nielen, and C. Georgakopoulos. Preventive doping control screening analysis of prohibited substances in human urine using rapid-resolution liquid chromatography/high-resolution time-of-flight mass spectrometry. Rapid Commun.Mass Spectrom. 24: 1595-1609 (2010).
-
(2010)
Rapid Commun. Mass Spectrom.
, vol.24
, pp. 1595-1609
-
-
Vonaparti, A.1
Lyris, E.2
Angelis, Y.S.3
Panderi, I.4
Koupparis, M.5
Tsantili-Kakoulidou, A.6
Peters, R.J.7
Nielen, M.W.8
Georgakopoulos, C.9
-
16
-
-
41149165250
-
Efficient approach for the comprehensive detection of unknown anabolic steroids and metabolites in human urine by liquid chromatography-electrospray-tandem mass spectrometry
-
O.J. Pozo, K. Deventer, P.VanEenoo, and F.T. Delbeke. Efficient approach for the comprehensive detection of unknown anabolic steroids and metabolites in human urine by liquid chromatography-electrospray-tandem mass spectrometry. Anal. Chem. 80: 709-720 (2008).
-
(2008)
Anal. Chem.
, vol.80
, pp. 709-720
-
-
Pozo, O.J.1
Deventer, K.2
VanEenoo, P.3
Delbeke, F.T.4
-
17
-
-
0028283503
-
Molecular mechanisms of action of steroid/thyroid receptor superfamily members
-
M.J. Tsai and B.W. O'Malley. Molecular mechanisms of action of steroid/thyroid receptor superfamily members. Annu. Rev. Biochem. 63: 451-486 (1994).
-
(1994)
Annu. Rev. Biochem.
, vol.63
, pp. 451-486
-
-
Tsai, M.J.1
O'Malley, B.W.2
-
19
-
-
0042770258
-
Structural analysis of complementary DNA and amino acid sequences of human and rat androgen receptors
-
C.S. Chang, J. Kokontis, and S.T. Liao. Structural analysis of complementary DNA and amino acid sequences of human and rat androgen receptors. Proc. Natl. Acad. Sci. USA 85: 7211-7215 (1988).
-
(1988)
Proc. Natl. Acad. Sci. USA
, vol.85
, pp. 7211-7215
-
-
Chang, C.S.1
Kokontis, J.2
Liao, S.T.3
-
20
-
-
0023929785
-
Molecular cloning of human and rat complementary DNA encoding androgen receptors
-
C.S. Chang, J. Kokontis, and S.T. Liao. Molecular cloning of human and rat complementary DNA encoding androgen receptors. Science 240: 324-326 (1988).
-
(1988)
Science
, vol.240
, pp. 324-326
-
-
Chang, C.S.1
Kokontis, J.2
Liao, S.T.3
-
21
-
-
25444496757
-
Chemistry and structural biology of androgen receptor
-
W. Gao, C.E. Bohl, and J.T. Dalton. Chemistry and structural biology of androgen receptor. Chem. Rev. 105: 3352-3370 (2005).
-
(2005)
Chem. Rev.
, vol.105
, pp. 3352-3370
-
-
Gao, W.1
Bohl, C.E.2
Dalton, J.T.3
-
22
-
-
0034937870
-
Lessons to be learned from the androgen receptor
-
A.O. Brinkmann. Lessons to be learned from the androgen receptor. Eur. J. Dermatol. 11: 301-303 (2001).
-
(2001)
Eur. J. Dermatol.
, vol.11
, pp. 301-303
-
-
Brinkmann, A.O.1
-
23
-
-
51549094259
-
Diverse roles of androgen receptor (AR) domains in AR-mediated signaling
-
F. Claessens, S. Denayer, N.Van Tilborgh, S. Kerkhofs, C. Helsen, and A. Haelens. Diverse roles of androgen receptor (AR) domains in AR-mediated signaling. Nucl. Recept. Signal 6: e008 (2008).
-
(2008)
Nucl. Recept. Signal
, vol.6
-
-
Claessens, F.1
Denayer, S.2
Van Tilborgh, N.3
Kerkhofs, S.4
Helsen, C.5
Haelens, A.6
-
24
-
-
0030925683
-
Steroid receptor interactions with heat shock protein and immunophilin chaperones
-
W.B. Pratt and D.O. Toft. Steroid receptor interactions with heat shock protein and immunophilin chaperones. Endocr. Rev. 18: 306-360 (1997).
-
(1997)
Endocr. Rev.
, vol.18
, pp. 306-360
-
-
Pratt, W.B.1
Toft, D.O.2
-
25
-
-
17544382884
-
Purification and stabilization of transcriptionally active glucocorticoid receptor
-
B.S.Warren, P. Kusk, R.G.Wolford, and G.L. Hager. Purification and stabilization of transcriptionally active glucocorticoid receptor. J. Biol. Chem. 271: 11434-11440 (1996).
-
(1996)
J. Biol. Chem.
, vol.271
, pp. 11434-11440
-
-
Warren, B.S.1
Kusk, P.2
Wolford, R.G.3
Hager, G.L.4
-
26
-
-
67349237917
-
Mechanism of androgen receptor action
-
J. Li and F. Al-Azzawi. Mechanism of androgen receptor action. Maturitas 63: 142-148 (2009).
-
(2009)
Maturitas
, vol.63
, pp. 142-148
-
-
Li, J.1
Al-Azzawi, F.2
-
27
-
-
0019869344
-
Molybdate permits resolution of untransformed glucocorticoid receptors from the transformed state
-
M.K. Dahmer, M.W. Quasney, S.T. Bissen, and W.B. Pratt. Molybdate permits resolution of untransformed glucocorticoid receptors from the transformed state. J. Biol. Chem. 256: 9401-9405 (1981).
-
(1981)
J. Biol. Chem.
, vol.256
, pp. 9401-9405
-
-
Dahmer, M.K.1
Quasney, M.W.2
Bissen, S.T.3
Pratt, W.B.4
-
28
-
-
33845414955
-
Controlling protein compartmentalization to overcome disease
-
J.R. Davis, M. Kakar, and C.S. Lim. Controlling protein compartmentalization to overcome disease. Pharm. Res. 24: 17-27 (2007).
-
(2007)
Pharm. Res.
, vol.24
, pp. 17-27
-
-
Davis, J.R.1
Kakar, M.2
Lim, C.S.3
-
29
-
-
0033279841
-
Transport between the cell nucleus and the cytoplasm
-
D. Gorlich and U. Kutay. Transport between the cell nucleus and the cytoplasm. Annu. Rev. Cell Dev. Biol. 15: 607-660 (1999).
-
(1999)
Annu. Rev. Cell Dev. Biol.
, vol.15
, pp. 607-660
-
-
Gorlich, D.1
Kutay, U.2
-
30
-
-
0030878878
-
Steroid receptor induction of gene transcription: a two-step model
-
G. Jenster, T.E. Spencer, M.M. Burcin, S.Y. Tsai, M.-J. Tsai, and B.W. O'Malley. Steroid receptor induction of gene transcription: a two-step model. Proc. Natl. Acad. Sci. USA 94: 7879-7884 (1997).
-
(1997)
Proc. Natl. Acad. Sci. USA
, vol.94
, pp. 7879-7884
-
-
Jenster, G.1
Spencer, T.E.2
Burcin, M.M.3
Tsai, S.Y.4
Tsai, M.-J.5
O'Malley, B.W.6
-
31
-
-
0036878979
-
Anabolic steroids, testosterone-precursors and virilizing androgens induce distinct activation profiles of androgen responsive promoter constructs
-
P.M. Holterhus, S. Piefke, and O. Hiort. Anabolic steroids, testosterone-precursors and virilizing androgens induce distinct activation profiles of androgen responsive promoter constructs. J. Steroid Biochem. Mol. Biol. 82: 269-275 (2002).
-
(2002)
J. Steroid Biochem. Mol. Biol.
, vol.82
, pp. 269-275
-
-
Holterhus, P.M.1
Piefke, S.2
Hiort, O.3
-
32
-
-
0039316318
-
Recruitment of octamer transcription factors to DNA by glucocorticoid receptor
-
G.G. Prefontaine, M.E. Lemieux, W. Giffin, C. Schild-Poulter, L. Pope, E. LaCasse, P. Walker, and R.J.G. Hache. Recruitment of octamer transcription factors to DNA by glucocorticoid receptor. Mol. Cell. Biol. 18: 3416-3430 (1998).
-
(1998)
Mol. Cell. Biol.
, vol.18
, pp. 3416-3430
-
-
Prefontaine, G.G.1
Lemieux, M.E.2
Giffin, W.3
Schild-Poulter, C.4
Pope, L.5
LaCasse, E.6
Walker, P.7
Hache, R.J.G.8
-
33
-
-
0027249002
-
Steroid hormone receptors: interaction with deoxyribonucleic acid and transcription factors
-
M. Truss and M. Beato. Steroid hormone receptors: interaction with deoxyribonucleic acid and transcription factors. Endocr. Rev. 14: 459-479 (1993).
-
(1993)
Endocr. Rev.
, vol.14
, pp. 459-479
-
-
Truss, M.1
Beato, M.2
-
34
-
-
77953254302
-
Effect of anabolicandrogenic steroids and glucocorticoids on the kinetics of hAR and hGR nucleocytoplasmic translocation
-
A.B. Cadwallader, D.E. Rollins, and C.S. Lim. Effect of anabolicandrogenic steroids and glucocorticoids on the kinetics of hAR and hGR nucleocytoplasmic translocation. Mol. Pharm. 7: 689-698 (2010).
-
(2010)
Mol. Pharm.
, vol.7
, pp. 689-698
-
-
Cadwallader, A.B.1
Rollins, D.E.2
Lim, C.S.3
-
36
-
-
0346027209
-
The mechanisms of androgen effects on body composition: mesenchymal pluripotent cell as the target of androgen action
-
S. Bhasin, W.E. Taylor, R. Singh, J. Artaza, I. Sinha-Hikim, R. Jasuja, H. Choi, and N.F. Gonzalez-Cadavid. The mechanisms of androgen effects on body composition: mesenchymal pluripotent cell as the target of androgen action. J. Gerontol. A Biol. Sci. Med. Sci. 58: M1103-1110 (2003).
-
(2003)
J. Gerontol. A Biol. Sci. Med. Sci.
, vol.58
-
-
Bhasin, S.1
Taylor, W.E.2
Singh, R.3
Artaza, J.4
Sinha-Hikim, I.5
Jasuja, R.6
Choi, H.7
Gonzalez-Cadavid, N.F.8
-
39
-
-
6344291192
-
Androgen receptor in human skeletal muscle and cultured muscle satellite cells: up-regulation by androgen treatment
-
I. Sinha-Hikim,W.E. Taylor, N.F. Gonzalez-Cadavid,W. Zheng, and S. Bhasin. Androgen receptor in human skeletal muscle and cultured muscle satellite cells: up-regulation by androgen treatment. J. Clin. Endocrinol. Metab. 89: 5245-5255 (2004).
-
(2004)
J. Clin. Endocrinol. Metab.
, vol.89
, pp. 5245-5255
-
-
Sinha-Hikim, I.1
Taylor, W.E.2
Gonzalez-Cadavid, N.F.3
Zheng, W.4
Bhasin, S.5
-
40
-
-
0036298091
-
Testosterone-induced increase in muscle size in healthy young men is associated with muscle fiber hypertrophy
-
I. Sinha-Hikim, J. Artaza, L.Woodhouse, N. Gonzalez-Cadavid, A.B. Singh, M.I. Lee, T.W. Storer, R. Casaburi, R. Shen, and S. Bhasin. Testosterone-induced increase in muscle size in healthy young men is associated with muscle fiber hypertrophy. Am. J. Physiol. Endocrinol. Metab. 283: E154-164 (2002).
-
(2002)
Am. J. Physiol. Endocrinol. Metab.
, vol.283
-
-
Sinha-Hikim, I.1
Artaza, J.2
Woodhouse, L.3
Gonzalez-Cadavid, N.4
Singh, A.B.5
Lee, M.I.6
Storer, T.W.7
Casaburi, R.8
Shen, R.9
Bhasin, S.10
-
41
-
-
29344440814
-
Testosterone inhibits adipogenic differentiation in 3T3-L1 cells: nuclear translocation of androgen receptor complex with beta-catenin and T-cell factor 4 may bypass canonicalWnt signaling to down-regulate adipogenic transcription factors
-
R. Singh, J.N. Artaza,W.E. Taylor, M. Braga, X. Yuan, N.F. Gonzalez-Cadavid, and S. Bhasin. Testosterone inhibits adipogenic differentiation in 3T3-L1 cells: nuclear translocation of androgen receptor complex with beta-catenin and T-cell factor 4 may bypass canonicalWnt signaling to down-regulate adipogenic transcription factors. Endocrinology 147: 141-154 (2006).
-
(2006)
Endocrinology
, vol.147
, pp. 141-154
-
-
Singh, R.1
Artaza, J.N.2
Taylor, W.E.3
Braga, M.4
Yuan, X.5
Gonzalez-Cadavid, N.F.6
Bhasin, S.7
-
42
-
-
0242468434
-
Androgens stimulate myogenic differentiation and inhibit adipogenesis in C3H 10T1/2 pluripotent cells through an androgen receptor-mediated pathway
-
R. Singh, J.N. Artaza, W.E. Taylor, N.F. Gonzalez-Cadavid, and S. Bhasin. Androgens stimulate myogenic differentiation and inhibit adipogenesis in C3H 10T1/2 pluripotent cells through an androgen receptor-mediated pathway. Endocrinology 144: 5081-5088 (2003).
-
(2003)
Endocrinology
, vol.144
, pp. 5081-5088
-
-
Singh, R.1
Artaza, J.N.2
Taylor, W.E.3
Gonzalez-Cadavid, N.F.4
Bhasin, S.5
-
43
-
-
42549164768
-
The physiological and pharmacological basis for the ergogenic effects of androgens in elite sports
-
K. Choong, K.M. Lakshman, and S. Bhasin. The physiological and pharmacological basis for the ergogenic effects of androgens in elite sports. Asian J. Androl. 10: 351-363 (2008).
-
(2008)
Asian J. Androl.
, vol.10
, pp. 351-363
-
-
Choong, K.1
Lakshman, K.M.2
Bhasin, S.3
-
44
-
-
22544451284
-
Androgen regulation of satellite cell function
-
Y. Chen, J.D. Zajac, and H.E. MacLean. Androgen regulation of satellite cell function. J. Endocrinol. 186: 21-31 (2005).
-
(2005)
J. Endocrinol.
, vol.186
, pp. 21-31
-
-
Chen, Y.1
Zajac, J.D.2
MacLean, H.E.3
-
45
-
-
0024595381
-
Satellite cell proliferation and increase in the number ofmyonuclei induced by testosterone in the levator ani muscle of the adult female rat
-
Y. Joubert and C. Tobin. Satellite cell proliferation and increase in the number ofmyonuclei induced by testosterone in the levator ani muscle of the adult female rat. Dev. Biol. 131: 550-557 (1989).
-
(1989)
Dev. Biol.
, vol.131
, pp. 550-557
-
-
Joubert, Y.1
Tobin, C.2
-
46
-
-
0038678058
-
Testosteroneinduced muscle hypertrophy is associated with an increase in satellite cell number in healthy, young men
-
I. Sinha-Hikim, S.M. Roth, M.I. Lee, and S. Bhasin. Testosteroneinduced muscle hypertrophy is associated with an increase in satellite cell number in healthy, young men. Am. J. Physiol. Endocrinol. Metab. 285: E197-E205 (2003).
-
(2003)
Am. J. Physiol. Endocrinol. Metab.
, vol.285
-
-
Sinha-Hikim, I.1
Roth, S.M.2
Lee, M.I.3
Bhasin, S.4
-
47
-
-
0030008005
-
Testosterone up-regulates androgen receptors and decreases differentiation of porcine myogenic satellite cells in vitro
-
M. Doumit, D.R. Cook, and R.A. Merkel. Testosterone up-regulates androgen receptors and decreases differentiation of porcine myogenic satellite cells in vitro. Endocrinology 137: 1385-1394 (1996).
-
(1996)
Endocrinology
, vol.137
, pp. 1385-1394
-
-
Doumit, M.1
Cook, D.R.2
Merkel, R.A.3
-
48
-
-
37349118115
-
Androgen receptor (AR) coregulators: a diversity of functions converging on and regulating the AR transcriptional complex
-
H.V. Heemers and D.J. Tindall. Androgen receptor (AR) coregulators: a diversity of functions converging on and regulating the AR transcriptional complex. Endocr. Rev. 28: 778-808 (2007).
-
(2007)
Endocr. Rev.
, vol.28
, pp. 778-808
-
-
Heemers, H.V.1
Tindall, D.J.2
-
49
-
-
15544371000
-
Ligand control of coregulator recruitment to nuclear receptors
-
K.W. Nettles and G.L. Greene. Ligand control of coregulator recruitment to nuclear receptors. Annu. Rev. Physiol. 67: 309-333 (2005).
-
(2005)
Annu. Rev. Physiol.
, vol.67
, pp. 309-333
-
-
Nettles, K.W.1
Greene, G.L.2
-
50
-
-
0345859565
-
The roles of sex steroid receptor coregulators in cancer
-
X. Gao, B.W. Loggie, and Z. Nawaz. The roles of sex steroid receptor coregulators in cancer. Mol. Cancer 1: 1-7 (2002).
-
(2002)
Mol. Cancer
, vol.1
, pp. 1-7
-
-
Gao, X.1
Loggie, B.W.2
Nawaz, Z.3
-
51
-
-
33646138016
-
Comparison of crystal structures of human androgen receptor ligand-binding domain complexed with various agonists reveals molecular determinants responsible for binding affinity
-
K. Pereira de Jesus-Tran, P.L. Cote, L. Cantin, J. Blanchet, F. Labrie, and R. Breton. Comparison of crystal structures of human androgen receptor ligand-binding domain complexed with various agonists reveals molecular determinants responsible for binding affinity. Protein Sci. 15: 987-999 (2006).
-
(2006)
Protein Sci
, vol.15
, pp. 987-999
-
-
Pereira de Jesus-Tran, K.1
Cote, P.L.2
Cantin, L.3
Blanchet, J.4
Labrie, F.5
Breton, R.6
-
52
-
-
0037621919
-
Dissociation of steroid receptor coactivator 1 and nuclear receptor corepressor recruitment to the human glucocorticoid receptor by modification of the ligand-receptor interface: the role of tyrosine 735
-
A. Stevens, H. Garside, A. Berry, C. Waters, A. White, and D. Ray. Dissociation of steroid receptor coactivator 1 and nuclear receptor corepressor recruitment to the human glucocorticoid receptor by modification of the ligand-receptor interface: the role of tyrosine 735. Mol. Endocrinol. 17: 845-859 (2003).
-
(2003)
Mol. Endocrinol.
, vol.17
, pp. 845-859
-
-
Stevens, A.1
Garside, H.2
Berry, A.3
Waters, C.4
White, A.5
Ray, D.6
-
53
-
-
0032213219
-
Structure and specificity of nuclear receptor-coactivator interactions
-
B.D. Darimont, R.L. Wagner, J.W. Apriletti, M.R. Stallcup, P.J. Kushner, J.D. Baxter, R.J. Fletterick, and K.R. Yamamoto. Structure and specificity of nuclear receptor-coactivator interactions. Genes Dev. 12: 3343-3356 (1998).
-
(1998)
Genes Dev
, vol.12
, pp. 3343-3356
-
-
Darimont, B.D.1
Wagner, R.L.2
Apriletti, J.W.3
Stallcup, M.R.4
Kushner, P.J.5
Baxter, J.D.6
Fletterick, R.J.7
Yamamoto, K.R.8
-
54
-
-
20044394709
-
The molecular mechanisms of coactivator utilization in ligand-dependent transactivation by the androgen receptor
-
E. Estebanez-Perpina, J.M. Moore, E. Mar, E. Delgado-Rodrigues, P. Nguyen, J.D. Baxter, B.M. Buehrer, P. Webb, R.J. Fletterick, and R.K. Guy. The molecular mechanisms of coactivator utilization in ligand-dependent transactivation by the androgen receptor. J. Biol. Chem. 280: 8060-8068 (2005).
-
(2005)
J. Biol. Chem.
, vol.280
, pp. 8060-8068
-
-
Estebanez-Perpina, E.1
Moore, J.M.2
Mar, E.3
Delgado-Rodrigues, E.4
Nguyen, P.5
Baxter, J.D.6
Buehrer, B.M.7
Webb, P.8
Fletterick, R.J.9
Guy, R.K.10
-
55
-
-
19344376991
-
Recognition and accommodation at the androgen receptor coactivator binding interface
-
E. Hur, S.J. Pfaff, E.S. Payne, H. Grøn, B.M. Buehrer, and R.J. Fletterick. Recognition and accommodation at the androgen receptor coactivator binding interface. PLoS Biol. 2: E274 (2004).
-
(2004)
PLoS Biol
, vol.2
-
-
Hur, E.1
Pfaff, S.J.2
Payne, E.S.3
Grøn, H.4
Buehrer, B.M.5
Fletterick, R.J.6
-
56
-
-
0036219918
-
Androgen receptor (AR) coregulators: an overview
-
C.A. Heinlein and C. Chang. Androgen receptor (AR) coregulators: an overview. Endocr. Rev. 23: 175-200 (2002).
-
(2002)
Endocr. Rev.
, vol.23
, pp. 175-200
-
-
Heinlein, C.A.1
Chang, C.2
-
58
-
-
0346496776
-
Androgens
-
10th ed., J.G. Hardman, L.E. Limbird, and A.G. Gilman, Eds. McGraw-Hill, New York, NY
-
P. Snyder. Androgens. In Goodman and Gilman's The Pharmacological Basis of Therapeutics, 10th ed., J.G. Hardman, L.E. Limbird, and A.G. Gilman, Eds. McGraw-Hill, New York, NY, 2001, pp 1635-1648.
-
(2001)
Goodman and Gilman's The Pharmacological Basis of Therapeutics
, pp. 1635-1648
-
-
Snyder, P.1
-
59
-
-
0029987681
-
Metabolism of anabolic androgenic steroids
-
W. Schanzer. Metabolism of anabolic androgenic steroids. Clin. Chem. 42: 1001-1020 (1996).
-
(1996)
Clin. Chem.
, vol.42
, pp. 1001-1020
-
-
Schanzer, W.1
-
61
-
-
0027346409
-
Exercise and inhibition of glucocorticoid-induced muscle atrophy
-
R.C. Hickson and J.R. Marone. Exercise and inhibition of glucocorticoid-induced muscle atrophy. Exerc. Sport Sci. Rev. 21: 135-167 (1993).
-
(1993)
Exerc. Sport Sci. Rev.
, vol.21
, pp. 135-167
-
-
Hickson, R.C.1
Marone, J.R.2
-
62
-
-
0016622562
-
Interaction of anabolic steroids with glucocorticoid receptor sites in rat muscle cytosol
-
M. Mayer and F. Rosen. Interaction of anabolic steroids with glucocorticoid receptor sites in rat muscle cytosol. Am. J. Physiol. 229: 1381-1386 (1975).
-
(1975)
Am. J. Physiol.
, vol.229
, pp. 1381-1386
-
-
Mayer, M.1
Rosen, F.2
-
66
-
-
84855664859
-
-
(accessed June 2010)
-
http://anabolicminds.com/forum/steroids/9989-vida-textandrogens. html (accessed June 2010).
-
-
-
-
67
-
-
84855664860
-
-
(accessed June 2010)
-
http://www.demonoid.com/files/details/1643294/008522825736/(accessed June 2010).
-
-
-
-
68
-
-
44349157577
-
Pharmacology of anabolic steroids
-
A.T. Kicman. Pharmacology of anabolic steroids. Br. J. Pharmacol. 154: 502-521 (2008).
-
(2008)
Br. J. Pharmacol.
, vol.154
, pp. 502-521
-
-
Kicman, A.T.1
-
69
-
-
67549142234
-
Nonsteroidal selective androgen receptor modulators (SARMs): dissociating the anabolic and androgenic activities of the androgen receptor for therapeutic benefit
-
M.L. Mohler, C.E. Bohl, A. Jones, C.C. Coss, R. Narayanan, Y. He, D.J. Hwang, J.T. Dalton, and D.D. Miller. Nonsteroidal selective androgen receptor modulators (SARMs): dissociating the anabolic and androgenic activities of the androgen receptor for therapeutic benefit. J. Med. Chem. 52: 3597-3617 (2009).
-
(2009)
J. Med. Chem.
, vol.52
, pp. 3597-3617
-
-
Mohler, M.L.1
Bohl, C.E.2
Jones, A.3
Coss, C.C.4
Narayanan, R.5
He, Y.6
Hwang, D.J.7
Dalton, J.T.8
Miller, D.D.9
-
70
-
-
0032489326
-
Discovery of nonsteroidal androgens
-
J.T. Dalton, A. Mukherjee, Z. Zhu, L. Kirkovsky, and D.D. Miller. Discovery of nonsteroidal androgens. Biochem. Biophys. Res. Commun. 244: 1-4 (1998).
-
(1998)
Biochem. Biophys. Res. Commun.
, vol.244
, pp. 1-4
-
-
Dalton, J.T.1
Mukherjee, A.2
Zhu, Z.3
Kirkovsky, L.4
Miller, D.D.5
-
71
-
-
59049096464
-
Selective androgen receptor modulators in preclinical and clinical development
-
R. Narayanan, M.L. Mohler, C.E. Bohl, D.D. Miller, and J.T. Dalton. Selective androgen receptor modulators in preclinical and clinical development. Nucl. Recept. Signal 6: e010 (2008).
-
(2008)
Nucl. Recept. Signal
, vol.6
-
-
Narayanan, R.1
Mohler, M.L.2
Bohl, C.E.3
Miller, D.D.4
Dalton, J.T.5
-
72
-
-
1842627842
-
Pharmacokinetics of S-3-(4-acetylamino-phenoxy)-2-hydroxy-2-methyl-N-(4-nitro-3-trifluoromethyl-phenyl)-propionamide in rats, a non-steroidal selective androgen receptor modulator
-
J.D. Kearbey, D.Wu,W. Gao, D.D. Miller, and J.T. Dalton. Pharmacokinetics of S-3-(4-acetylamino-phenoxy)-2-hydroxy-2-methyl-N-(4-nitro-3-trifluoromethyl-phenyl)-propionamide in rats, a non-steroidal selective androgen receptor modulator. Xenobiotica 34: 273-280 (2004).
-
(2004)
Xenobiotica
, vol.34
, pp. 273-280
-
-
Kearbey, J.D.1
Wu, D.2
Gao, W.3
Miller, D.D.4
Dalton, J.T.5
-
73
-
-
22544467523
-
Discovery and therapeutic promise of selective androgen receptor modulators
-
J. Chen, J. Kim, and J.T. Dalton. Discovery and therapeutic promise of selective androgen receptor modulators. Mol. Interv. 5: 173-188 (2005).
-
(2005)
Mol. Interv.
, vol.5
, pp. 173-188
-
-
Chen, J.1
Kim, J.2
Dalton, J.T.3
-
74
-
-
77449160132
-
Synthetic anabolic agents: steroids and nonsteroidal selective androgen receptor modulators
-
M. Thevis and W. Schänzer. Synthetic anabolic agents: steroids and nonsteroidal selective androgen receptor modulators. Handb. Exp. Pharmacol. 195: 99-126 (2010).
-
(2010)
Handb. Exp. Pharmacol.
, vol.195
, pp. 99-126
-
-
Thevis, M.1
Schänzer, W.2
-
75
-
-
18044371228
-
Androgen receptor-cofactor interactions as targets for new drug discovery
-
C.Y. Chang and D.P. McDonnell. Androgen receptor-cofactor interactions as targets for new drug discovery. Trends Pharmacol. Sci. 26: 225-228 (2005).
-
(2005)
Trends Pharmacol. Sci.
, vol.26
, pp. 225-228
-
-
Chang, C.Y.1
McDonnell, D.P.2
-
76
-
-
82855178424
-
-
WADA. The 2010 Prohibited List. International Standard.WADA, Montreal, QC, Canada
-
WADA. TheWorld Anti-Doping Code. The 2010 Prohibited List. International Standard.WADA, Montreal, QC, Canada, 2010.
-
(2010)
TheWorld Anti-Doping Code
-
-
-
77
-
-
47749101721
-
Mass spectrometry of selective androgen receptor modulators
-
M. Thevis and W. Schanzer. Mass spectrometry of selective androgen receptor modulators. J. Mass Spectrom. 43: 865-876 (2008).
-
(2008)
J. Mass Spectrom.
, vol.43
, pp. 865-876
-
-
Thevis, M.1
Schanzer, W.2
-
78
-
-
40849120748
-
Aryl-propionamide-derived selective androgen receptor modulators: liquid chromatography-tandem mass spectrometry characterization of the in vitro synthesized metabolites for doping control purposes
-
T. Kuuranne, A. Leinonen, W. Schanzer, M. Kamber, R. Kostiainen, and M. Thevis. Aryl-propionamide-derived selective androgen receptor modulators: liquid chromatography-tandem mass spectrometry characterization of the in vitro synthesized metabolites for doping control purposes. Drug Metab. Dispos. 36: 571-581 (2008).
-
(2008)
Drug Metab. Dispos.
, vol.36
, pp. 571-581
-
-
Kuuranne, T.1
Leinonen, A.2
Schanzer, W.3
Kamber, M.4
Kostiainen, R.5
Thevis, M.6
-
79
-
-
42449084465
-
Determination of benzimidazoleand bicyclic hydantoin-derived selective androgen receptor antagonists and agonists in human urine using LC-MS/MS
-
M. Thevis, M. Kohler, A. Thomas, J. Maurer, N. Schlorer, M. Kamber, and W. Schanzer. Determination of benzimidazoleand bicyclic hydantoin-derived selective androgen receptor antagonists and agonists in human urine using LC-MS/MS. Anal. Bioanal. Chem. 391: 251-261 (2008).
-
(2008)
Anal. Bioanal. Chem.
, vol.391
, pp. 251-261
-
-
Thevis, M.1
Kohler, M.2
Thomas, A.3
Maurer, J.4
Schlorer, N.5
Kamber, M.6
Schanzer, W.7
-
80
-
-
65749089277
-
Emerging drugs: mechanism of action, mass spectrometry and doping control analysis
-
M. Thevis, A. Thomas, M. Kohler, S. Beuck, and W. Schanzer. Emerging drugs: mechanism of action, mass spectrometry and doping control analysis. J.Mass Spectrom. 44: 442-460 (2009).
-
(2009)
J. Mass Spectrom.
, vol.44
, pp. 442-460
-
-
Thevis, M.1
Thomas, A.2
Kohler, M.3
Beuck, S.4
Schanzer, W.5
-
81
-
-
57349182202
-
Illicit organogenesis: methods and substances of doping and manipulation
-
M. Thevis and W. Schanzer. Illicit organogenesis: methods and substances of doping and manipulation. Organogenesis 4: 264-271 (2008).
-
(2008)
Organogenesis
, vol.4
, pp. 264-271
-
-
Thevis, M.1
Schanzer, W.2
-
82
-
-
37649023920
-
New drugs and methods of doping and manipulation
-
M. Thevis, M. Kohler, and W. Schanzer. New drugs and methods of doping and manipulation. Drug Discov. Today 13: 59-66 (2008).
-
(2008)
Drug Discov. Today
, vol.13
, pp. 59-66
-
-
Thevis, M.1
Kohler, M.2
Schanzer, W.3
-
83
-
-
34247386771
-
Analysis of a challenging subset of World Anti-Doping Agency-banned steroids and antiestrogens by LC-MS-MS
-
C.R. Borges, N. Miller, M. Shelby, M. Hansen, C. White, M.H. Slawson, K. Monti, and D.J. Crouch. Analysis of a challenging subset of World Anti-Doping Agency-banned steroids and antiestrogens by LC-MS-MS. J. Anal. Toxicol. 31: 125-131 (2007).
-
(2007)
J. Anal. Toxicol.
, vol.31
, pp. 125-131
-
-
Borges, C.R.1
Miller, N.2
Shelby, M.3
Hansen, M.4
White, C.5
Slawson, M.H.6
Monti, K.7
Crouch, D.J.8
-
84
-
-
33846624349
-
A general screening method for doping agents in human urine by solid phase extraction and liquid chromatography/time-of-flight mass spectrometry
-
M. Kolmonen, A. Leinonen, A. Pelander, and I. Ojanperä. A general screening method for doping agents in human urine by solid phase extraction and liquid chromatography/time-of-flight mass spectrometry. Anal. Chim. Acta 585: 94-102 (2007).
-
(2007)
Anal. Chim. Acta
, vol.585
, pp. 94-102
-
-
Kolmonen, M.1
Leinonen, A.2
Pelander, A.3
Ojanperä, I.4
-
85
-
-
37649013598
-
Application of fast gas chromatography/mass spectrometry for the rapid screening of synthetic anabolic steroids and other drugs in anti-doping analysis
-
M. Mazzarino, M. Orengia, and F. Botre. Application of fast gas chromatography/mass spectrometry for the rapid screening of synthetic anabolic steroids and other drugs in anti-doping analysis. Rapid Commun. Mass Spectrom. 21: 4117-4124 (2007).
-
(2007)
Rapid Commun. Mass Spectrom.
, vol.21
, pp. 4117-4124
-
-
Mazzarino, M.1
Orengia, M.2
Botre, F.3
-
86
-
-
34748883693
-
Development and validation of a qualitative screening method for the detection of exogenous anabolic steroids in urine by liquid chromatography-tandem mass spectrometry
-
O.J. Pozo, P. Van Eenoo, K. Deventer, and F.T. Delbeke. Development and validation of a qualitative screening method for the detection of exogenous anabolic steroids in urine by liquid chromatography-tandem mass spectrometry. Anal. Bioanal. Chem. 389: 1209-1224 (2007).
-
(2007)
Anal. Bioanal. Chem.
, vol.389
, pp. 1209-1224
-
-
Pozo, O.J.1
Van Eenoo, P.2
Deventer, K.3
Delbeke, F.T.4
-
87
-
-
37549025787
-
In vitro bioassays for androgens and their diagnostic applications
-
P. Roy, M. Alevizaki, and I. Huhtaniemi. In vitro bioassays for androgens and their diagnostic applications. Hum. Reprod.Update 14: 73-82 (2008).
-
(2008)
Hum. Reprod. Update
, vol.14
, pp. 73-82
-
-
Roy, P.1
Alevizaki, M.2
Huhtaniemi, I.3
-
88
-
-
61849096693
-
Validation and application of a yeast bioassay for screening androgenic activity in calf urine and feed
-
T.F. Bovee, G. Bor, H.H. Heskamp, J.J. Lasaroms, M.B. Sanders, and M.W. Nielen. Validation and application of a yeast bioassay for screening androgenic activity in calf urine and feed. Anal. Chim. Acta 637: 225-234 (2009).
-
(2009)
Anal. Chim. Acta
, vol.637
, pp. 225-234
-
-
Bovee, T.F.1
Bor, G.2
Heskamp, H.H.3
Lasaroms, J.J.4
Sanders, M.B.5
Nielen, M.W.6
-
89
-
-
35648992471
-
A new highly specific and robust yeast androgen bioassay for the detection of agonists and antagonists
-
T.F. Bovee, R.J. Helsdingen, A.R. Hamers, M.B. van Duursen, M.W. Nielen, and R.L. Hoogenboom. A new highly specific and robust yeast androgen bioassay for the detection of agonists and antagonists. Anal. Bioanal. Chem. 389: 1549-1558 (2007).
-
(2007)
Anal. Bioanal. Chem.
, vol.389
, pp. 1549-1558
-
-
Bovee, T.F.1
Helsdingen, R.J.2
Hamers, A.R.3
van Duursen, M.B.4
Nielen, M.W.5
Hoogenboom, R.L.6
-
90
-
-
72449170947
-
SERMs and SARMs: detection of their activities with yeast based bioassays
-
T.F. Bovee, M. Thevis, A.R. Hamers, A.A. Peijnenburg, M.W. Nielen, and W.G. Schoonen. SERMs and SARMs: detection of their activities with yeast based bioassays. J. Steroid Biochem. Mol. Biol. 118: 85-92 (2009).
-
(2009)
J. Steroid Biochem. Mol. Biol.
, vol.118
, pp. 85-92
-
-
Bovee, T.F.1
Thevis, M.2
Hamers, A.R.3
Peijnenburg, A.A.4
Nielen, M.W.5
Schoonen, W.G.6
-
91
-
-
0031105822
-
Evaluation of chemicals with endocrine modulating activity in a yeast-based steroid hormone receptor gene transcription assay
-
K.W. Gaido, L.S. Leonard, S. Lovell, J.C. Gould, D. Babai, C.J. Portier, and D.P. McDonnell. Evaluation of chemicals with endocrine modulating activity in a yeast-based steroid hormone receptor gene transcription assay. Toxicol. Appl. Pharmacol. 143: 205-212 (1997).
-
(1997)
Toxicol. Appl. Pharmacol.
, vol.143
, pp. 205-212
-
-
Gaido, K.W.1
Leonard, L.S.2
Lovell, S.3
Gould, J.C.4
Babai, D.5
Portier, C.J.6
McDonnell, D.P.7
-
92
-
-
0037377230
-
Novel yeast bioassay system for detection of androgenic and antiandrogenic compounds
-
H.J. Lee, Y.S. Lee, H.B. Kwon, and K. Lee. Novel yeast bioassay system for detection of androgenic and antiandrogenic compounds. Toxicol. In Vitro 17: 237-244 (2003).
-
(2003)
Toxicol. In Vitro
, vol.17
, pp. 237-244
-
-
Lee, H.J.1
Lee, Y.S.2
Kwon, H.B.3
Lee, K.4
-
93
-
-
23744463526
-
Bioluminescent yeast assays for detecting estrogenic and androgenic activity in different matrices
-
P. Leskinen, E. Michelini, D. Picard, M. Karp, and M.Virta. Bioluminescent yeast assays for detecting estrogenic and androgenic activity in different matrices. Chemosphere 61: 259-266 (2005).
-
(2005)
Chemosphere
, vol.61
, pp. 259-266
-
-
Leskinen, P.1
Michelini, E.2
Picard, D.3
Karp, M.4
Virta, M.5
-
94
-
-
0345201750
-
A yeast screen system for aromatase inhibitors and ligands for androgen receptor: yeast cells transformed with aromatase and androgen receptor
-
P. Mak, F.D. Cruz, and S. Chen. A yeast screen system for aromatase inhibitors and ligands for androgen receptor: yeast cells transformed with aromatase and androgen receptor. Environ. Health Perspect. 107: 855-860 (1999).
-
(1999)
Environ. Health Perspect.
, vol.107
, pp. 855-860
-
-
Mak, P.1
Cruz, F.D.2
Chen, S.3
-
95
-
-
15944402750
-
A new recombinant cell-based bioluminescent assay for sensitive androgen-like compound detection
-
E. Michelini, P. Leskinen, M.Virta, M. Karp, and A. Roda. A new recombinant cell-based bioluminescent assay for sensitive androgen-like compound detection. Biosens. Bioelectron. 20: 2261-2267 (2005).
-
(2005)
Biosens. Bioelectron.
, vol.20
, pp. 2261-2267
-
-
Michelini, E.1
Leskinen, P.2
Virta, M.3
Karp, M.4
Roda, A.5
-
96
-
-
25444452108
-
Recombinant cell-based bioluminescence assay for androgen bioactivity determination in clinical samples
-
E. Michelini, M. Magliulo, P. Leskinen, M. Virta, M. Karp, and A. Roda. Recombinant cell-based bioluminescence assay for androgen bioactivity determination in clinical samples. Clin. Chem. 51: 1995-1998 (2005).
-
(2005)
Clin. Chem.
, vol.51
, pp. 1995-1998
-
-
Michelini, E.1
Magliulo, M.2
Leskinen, P.3
Virta, M.4
Karp, M.5
Roda, A.6
-
97
-
-
0025997048
-
An androgen-inducible expression system for Saccharomyces cerevisiae
-
I.J. Purvis, D. Chotai, C.W. Dykes, D.B. Lubahn, F.S. French, E.M. Wilson, and A.N. Hobden. An androgen-inducible expression system for Saccharomyces cerevisiae. Gene 106: 35-42 (1991).
-
(1991)
Gene
, vol.106
, pp. 35-42
-
-
Purvis, I.J.1
Chotai, D.2
Dykes, C.W.3
Lubahn, D.B.4
French, F.S.5
Wilson, E.M.6
Hobden, A.N.7
-
98
-
-
0031656115
-
Several environmental oestrogens are also anti-androgens
-
P. Sohoni and J.P. Sumpter. Several environmental oestrogens are also anti-androgens. J. Endocrinol. 158: 327-339 (1998).
-
(1998)
J. Endocrinol.
, vol.158
, pp. 327-339
-
-
Sohoni, P.1
Sumpter, J.P.2
-
99
-
-
46749138616
-
Detection of anabolic steroid abuse using a yeast transactivation system
-
O. Zierau, S. Lehmann, G. Vollmer, W. Schanzer, and P. Diel. Detection of anabolic steroid abuse using a yeast transactivation system. Steroids 73: 1143-1147 (2008).
-
(2008)
Steroids
, vol.73
, pp. 1143-1147
-
-
Zierau, O.1
Lehmann, S.2
Vollmer, G.3
Schanzer, W.4
Diel, P.5
-
100
-
-
37549066675
-
Androgen receptor transactivation assay using green fluorescent protein as a reporter
-
V. Beck, E. Reiter, and A. Jungbauer. Androgen receptor transactivation assay using green fluorescent protein as a reporter. Anal. Biochem. 373: 263-271 (2008).
-
(2008)
Anal. Biochem.
, vol.373
, pp. 263-271
-
-
Beck, V.1
Reiter, E.2
Jungbauer, A.3
-
101
-
-
0035499955
-
Development of an androgen reporter gene assay (AR-LUX) utilizing a human cell line with an endogenously regulated androgen receptor
-
B.M. Blankvoort, E.M. de Groene, A.P. van Meeteren-Kreikamp, R.F.Witkamp, R.J. Rodenburg, and J.M. Aarts. Development of an androgen reporter gene assay (AR-LUX) utilizing a human cell line with an endogenously regulated androgen receptor. Anal. Biochem. 298: 93-102 (2001).
-
(2001)
Anal. Biochem.
, vol.298
, pp. 93-102
-
-
Blankvoort, B.M.1
de Groene, E.M.2
van Meeteren-Kreikamp, A.P.3
Witkamp, R.F.4
Rodenburg, R.J.5
Aarts, J.M.6
-
102
-
-
33751551690
-
Circulating bioactive androgens in midlife women
-
J. Chen, M.R. Sowers, F.M. Moran, D.S. McConnell, N.A. Gee, G.A. Greendale, C. Whitehead, S.E. Kasim-Karakas, and B.L. Lasley. Circulating bioactive androgens in midlife women. J. Clin. Endocrinol. Metab. 91: 4387-4394 (2006).
-
(2006)
J. Clin. Endocrinol. Metab.
, vol.91
, pp. 4387-4394
-
-
Chen, J.1
Sowers, M.R.2
Moran, F.M.3
McConnell, D.S.4
Gee, N.A.5
Greendale, G.A.6
Whitehead, C.7
Kasim-Karakas, S.E.8
Lasley, B.L.9
-
103
-
-
0037333156
-
Tibolone is not converted by human aromatase to 7alpha-methyl-17alpha-ethynylestradiol (7alpha-MEE): analyses with sensitive bioassays for estrogens and androgens and with LC-MSMS
-
M.E. de Gooyer, H.M. Oppers-Tiemissen, D. Leysen, H.A. Verheul, and H.J. Kloosterboer. Tibolone is not converted by human aromatase to 7alpha-methyl-17alpha-ethynylestradiol (7alpha-MEE): analyses with sensitive bioassays for estrogens and androgens and with LC-MSMS. Steroids 68: 235-243 (2003).
-
(2003)
Steroids
, vol.68
, pp. 235-243
-
-
de Gooyer, M.E.1
Oppers-Tiemissen, H.M.2
Leysen, D.3
Verheul, H.A.4
Kloosterboer, H.J.5
-
104
-
-
61849083471
-
Detection of anabolic androgenic steroid abuse in doping control using mammalian reporter gene bioassays
-
C.J. Houtman, S.S. Sterk, M.P. van de Heijning, A. Brouwer, R.W. Stephany, B. van der Burg, and E. Sonneveld. Detection of anabolic androgenic steroid abuse in doping control using mammalian reporter gene bioassays. Anal. Chim. Acta 637: 247-258 (2009).
-
(2009)
Anal. Chim. Acta
, vol.637
, pp. 247-258
-
-
Houtman, C.J.1
Sterk, S.S.2
van de Heijning, M.P.3
Brouwer, A.4
Stephany, R.W.5
van der Burg, B.6
Sonneveld, E.7
-
105
-
-
77955868810
-
Biological analysis of endocrine-disrupting compounds in Tunisian sewage treatment plants
-
W. Mnif, S. Dagnino, A. Escande, A. Pillon, H. Fenet, E. Gomez, C. Casellas, M.J. Duchesne, G. Hernandez-Raquet,V. Cavaillès, P. Balaguer, and A. Bartegi. Biological analysis of endocrine-disrupting compounds in Tunisian sewage treatment plants. Arch. Environ. Contam. Toxicol. 59(1): 1-12 (2010).
-
(2010)
Arch. Environ. Contam. Toxicol.
, vol.59
, Issue.1
, pp. 1-12
-
-
Mnif, W.1
Dagnino, S.2
Escande, A.3
Pillon, A.4
Fenet, H.5
Gomez, E.6
Casellas, C.7
Duchesne, M.J.8
Hernandez-Raquet, G.9
Cavaillès, V.10
Balaguer, P.11
Bartegi, A.12
-
106
-
-
34248593017
-
Antiandrogenic activity of norgestimate in a human androgen-dependent stable-transfected cell line
-
F. Paris, F. Rabeolina, P. Balaguer, A. Bacquet, and C. Sultan. Antiandrogenic activity of norgestimate in a human androgen-dependent stable-transfected cell line. Gynecol. Endocrinol. 23: 193-197 (2007).
-
(2007)
Gynecol. Endocrinol.
, vol.23
, pp. 193-197
-
-
Paris, F.1
Rabeolina, F.2
Balaguer, P.3
Bacquet, A.4
Sultan, C.5
-
107
-
-
0036174089
-
A new recombinant cell bioassay for ultrasensitive determination of serum estrogenic bioactivity in children
-
F. Paris, N. Servant, B. Terouanne, P. Balaguer, J.C. Nicolas, and C. Sultan. A new recombinant cell bioassay for ultrasensitive determination of serum estrogenic bioactivity in children. J. Clin. Endocrinol. Metab. 87: 791-797 (2002).
-
(2002)
J. Clin. Endocrinol. Metab.
, vol.87
, pp. 791-797
-
-
Paris, F.1
Servant, N.2
Terouanne, B.3
Balaguer, P.4
Nicolas, J.C.5
Sultan, C.6
-
108
-
-
0037203496
-
Evaluation of androgenic bioactivity in human serum by recombinant cell line: preliminary results
-
F. Paris, N. Servant, B. Terouanne, and C. Sultan. Evaluation of androgenic bioactivity in human serum by recombinant cell line: preliminary results. Mol. Cell Endocrinol. 198: 123-129 (2002).
-
(2002)
Mol. Cell Endocrinol.
, vol.198
, pp. 123-129
-
-
Paris, F.1
Servant, N.2
Terouanne, B.3
Sultan, C.4
-
109
-
-
0035037647
-
Novel assay for determination of androgen bioactivity in human serum
-
T. Raivio, J.J. Palvimo, L. Dunkel, S.Wickman, and O.A. Janne. Novel assay for determination of androgen bioactivity in human serum. J. Clin. Endocrinol. Metab. 86: 1539-1544 (2001).
-
(2001)
J. Clin. Endocrinol. Metab.
, vol.86
, pp. 1539-1544
-
-
Raivio, T.1
Palvimo, J.J.2
Dunkel, L.3
Wickman, S.4
Janne, O.A.5
-
110
-
-
33748064349
-
Determination of androgen bioactivity in human serum samples using a recombinant cell based in vitro bioassay
-
P. Roy, S. Franks, M. Read, and I.T. Huhtaniemi. Determination of androgen bioactivity in human serum samples using a recombinant cell based in vitro bioassay. J. Steroid Biochem.Mol. Biol. 101: 68-77 (2006).
-
(2006)
J. Steroid Biochem. Mol. Biol.
, vol.101
, pp. 68-77
-
-
Roy, P.1
Franks, S.2
Read, M.3
Huhtaniemi, I.T.4
-
111
-
-
1842785912
-
Screening of some anti-androgenic endocrine disruptors using a recombinant cell-based in vitro bioassay
-
P. Roy, H. Salminen, P. Koskimies, J. Simola, A. Smeds, P. Saukko, and I.T. Huhtaniemi. Screening of some anti-androgenic endocrine disruptors using a recombinant cell-based in vitro bioassay. J. Steroid Biochem.Mol. Biol. 88: 157-166 (2004).
-
(2004)
J. Steroid Biochem. Mol. Biol.
, vol.88
, pp. 157-166
-
-
Roy, P.1
Salminen, H.2
Koskimies, P.3
Simola, J.4
Smeds, A.5
Saukko, P.6
Huhtaniemi, I.T.7
-
112
-
-
12344265705
-
Development of androgen- and estrogen-responsive bioassays, members of a panel of human cell line-based highly selective steroid-responsive bioassays
-
E. Sonneveld, H.J. Jansen, J.A. Riteco, A. Brouwer and B. van der Burg. Development of androgen- and estrogen-responsive bioassays, members of a panel of human cell line-based highly selective steroid-responsive bioassays. Toxicol. Sci. 83: 136-148 (2005).
-
(2005)
Toxicol. Sci.
, vol.83
, pp. 136-148
-
-
Sonneveld, E.1
Jansen, H.J.2
Riteco, J.A.3
Brouwer, A.4
van der Burg, B.5
-
113
-
-
29544439001
-
Comparison of in vitro and in vivo screening models for androgenic and estrogenic activities
-
E. Sonneveld, J.A. Riteco, H.J. Jansen, B. Pieterse, A. Brouwer, W.G. Schoonen, and B. van der Burg. Comparison of in vitro and in vivo screening models for androgenic and estrogenic activities. Toxicol. Sci. 89: 173-187 (2006).
-
(2006)
Toxicol. Sci.
, vol.89
, pp. 173-187
-
-
Sonneveld, E.1
Riteco, J.A.2
Jansen, H.J.3
Pieterse, B.4
Brouwer, A.5
Schoonen, W.G.6
van der Burg, B.7
-
114
-
-
0037379703
-
Mutation of the androgen receptor at amino acid 708 (Gly-->Ala) abolishes partial agonist activity of steroidal antiandrogens
-
B. Terouanne, P. Nirdé, F. Rabenoelina,W. Bourguet, C. Sultan, and G. Auzou. Mutation of the androgen receptor at amino acid 708 (Gly-->Ala) abolishes partial agonist activity of steroidal antiandrogens. Mol. Pharmacol. 63: 791-798 (2003).
-
(2003)
Mol. Pharmacol.
, vol.63
, pp. 791-798
-
-
Terouanne, B.1
Nirdé, P.2
Rabenoelina, F.3
Bourguet, W.4
Sultan, C.5
Auzou, G.6
-
115
-
-
56249084597
-
Androgen receptor functional analyses by high throughput imaging: determination of ligand, cell cycle, and mutation-specific effects
-
A.T. Szafran, M. Szwarc, M. Marcelli, and M.A. Mancini. Androgen receptor functional analyses by high throughput imaging: determination of ligand, cell cycle, and mutation-specific effects. PLoS One 3: e3605 (2008).
-
(2008)
PLoS One
, vol.3
-
-
Szafran, A.T.1
Szwarc, M.2
Marcelli, M.3
Mancini, M.A.4
-
116
-
-
31444441045
-
Transfection with steroid-responsive reporter constructs shows glucocorticoid rather than androgen responsiveness in cultured Sertoli cells
-
E. Denolet, K.D. Gendt, J.V. Swinnen, G. Verrijdt, L. Deboel, T. Roskams, and G. Verhoeven. Transfection with steroid-responsive reporter constructs shows glucocorticoid rather than androgen responsiveness in cultured Sertoli cells. J. Steroid Biochem. Mol. Biol. 98: 164-173 (2006).
-
(2006)
J. Steroid Biochem. Mol. Biol.
, vol.98
, pp. 164-173
-
-
Denolet, E.1
Gendt, K.D.2
Swinnen, J.V.3
Verrijdt, G.4
Deboel, L.5
Roskams, T.6
Verhoeven, G.7
-
117
-
-
0036192083
-
A novel cell line, MDA-kb2, that stably expresses an androgenand glucocorticoid-responsive reporter for the detection of hormone receptor agonists and antagonists
-
V.S. Wilson, K. Bobseine, C.R. Lambright, and L.E. Gray, Jr. A novel cell line, MDA-kb2, that stably expresses an androgenand glucocorticoid-responsive reporter for the detection of hormone receptor agonists and antagonists. Toxicol. Sci. 66: 69-81 (2002).
-
(2002)
Toxicol. Sci.
, vol.66
, pp. 69-81
-
-
Wilson, V.S.1
Bobseine, K.2
Lambright, C.R.3
Gray Jr., L.E.4
-
118
-
-
40749093681
-
Detailed functional studies on androgen receptor mild mutations demonstrate their association with male infertility
-
D. Zuccarello, A. Ferlin, C. Vinanzi, E. Prana, A. Garolla, L. Callewaert, F. Claessens, A.O. Brinkmann, and C. Foresta. Detailed functional studies on androgen receptor mild mutations demonstrate their association with male infertility. Clin. Endocrinol. (Oxf.) 68: 580-588 (2008).
-
(2008)
Clin. Endocrinol. (Oxf.)
, vol.68
, pp. 580-588
-
-
Zuccarello, D.1
Ferlin, A.2
Vinanzi, C.3
Prana, E.4
Garolla, A.5
Callewaert, L.6
Claessens, F.7
Brinkmann, A.O.8
Foresta, C.9
-
119
-
-
0029778413
-
The androgen-specific probasin response element 2 interacts differentially with androgen and glucocorticoid receptors
-
F. Claessens, P. Alen, A. Devos, B. Peeters, G. Verhoeven, and W. Rombauts. The androgen-specific probasin response element 2 interacts differentially with androgen and glucocorticoid receptors. J. Biol. Chem. 271: 19013-19016 (1996).
-
(1996)
J. Biol. Chem.
, vol.271
, pp. 19013-19016
-
-
Claessens, F.1
Alen, P.2
Devos, A.3
Peeters, B.4
Verhoeven, G.5
Rombauts, W.6
-
120
-
-
0034993267
-
Selective DNA binding by the androgen receptor as a mechanism for hormonespecific gene regulation
-
F. Claessens, G. Verrijdt, E. Schoenmakers, A. Haelens, B. Peeters, G. Verhoeven and W. Rombauts. Selective DNA binding by the androgen receptor as a mechanism for hormonespecific gene regulation. J. Steroid Biochem. Mol. Biol. 76: 23-30 (2001).
-
(2001)
J. Steroid Biochem. Mol. Biol.
, vol.76
, pp. 23-30
-
-
Claessens, F.1
Verrijdt, G.2
Schoenmakers, E.3
Haelens, A.4
Peeters, B.5
Verhoeven, G.6
Rombauts, W.7
-
121
-
-
0034697122
-
Differences in DNA binding characteristics of the androgen and glucocorticoid receptors can determine hormone-specific responses
-
E. Schoenmakers, G. Verrijdt, B. Peeters, G. Verhoeven, W. Rombauts, and F. Claessens. Differences in DNA binding characteristics of the androgen and glucocorticoid receptors can determine hormone-specific responses. J. Biol. Chem. 275: 12290-12297 (2000).
-
(2000)
J. Biol. Chem.
, vol.275
, pp. 12290-12297
-
-
Schoenmakers, E.1
Verrijdt, G.2
Peeters, B.3
Verhoeven, G.4
Rombauts, W.5
Claessens, F.6
-
122
-
-
0033305722
-
Androgen specificity of a response unit upstream of the human secretory component gene is mediated by differential receptor binding to an essential androgen response element
-
G. Verrijdt, E. Schoenmakers, P. Alen, A. Haelens, B. Peeters, W. Rombauts, and F. Claessens. Androgen specificity of a response unit upstream of the human secretory component gene is mediated by differential receptor binding to an essential androgen response element. Mol. Endocrinol. 13: 1558-1570 (1999).
-
(1999)
Mol. Endocrinol.
, vol.13
, pp. 1558-1570
-
-
Verrijdt, G.1
Schoenmakers, E.2
Alen, P.3
Haelens, A.4
Peeters, B.5
Rombauts, W.6
Claessens, F.7
-
123
-
-
0034697359
-
Change of specificity mutations in androgen-selective enhancers. Evidence for a role of differential DNA binding by the androgen receptor
-
G. Verrijdt, E. Schoenmakers, A. Haelens, B. Peeters, G. Verhoeven, W. Rombauts, and F. Claessens. Change of specificity mutations in androgen-selective enhancers. Evidence for a role of differential DNA binding by the androgen receptor. J. Biol. Chem. 275: 12298-12305 (2000).
-
(2000)
J. Biol. Chem.
, vol.275
, pp. 12298-12305
-
-
Verrijdt, G.1
Schoenmakers, E.2
Haelens, A.3
Peeters, B.4
Verhoeven, G.5
Rombauts, W.6
Claessens, F.7
-
124
-
-
0037809279
-
Dynamic shuttling and intranuclear mobility of nuclear hormone receptors
-
P. Maruvada, C.T. Baumann, G.L. Hager, and P.M. Yen. Dynamic shuttling and intranuclear mobility of nuclear hormone receptors. J. Biol. Chem. 278: 12425-12432 (2003).
-
(2003)
J. Biol. Chem.
, vol.278
, pp. 12425-12432
-
-
Maruvada, P.1
Baumann, C.T.2
Hager, G.L.3
Yen, P.M.4
-
125
-
-
0037372002
-
Molecular determinants of glucocorticoid receptor mobility in living cells: the importance of ligand affinity
-
M.J. Schaaf and J.A. Cidlowski. Molecular determinants of glucocorticoid receptor mobility in living cells: the importance of ligand affinity. Mol. Cell Biol. 23: 1922-1934 (2003).
-
(2003)
Mol. Cell Biol.
, vol.23
, pp. 1922-1934
-
-
Schaaf, M.J.1
Cidlowski, J.A.2
-
126
-
-
7244247363
-
Estrogen response element-dependent regulation of transcriptional activation of estrogen receptors alpha and beta by coactivators and corepressors
-
C.M. Klinge, S.C. Jernigan, K.A. Mattingly, K.E. Risinger, and J. Zhang. Estrogen response element-dependent regulation of transcriptional activation of estrogen receptors alpha and beta by coactivators and corepressors. J. Mol. Endocrinol. 33: 387-410 (2004).
-
(2004)
J. Mol. Endocrinol.
, vol.33
, pp. 387-410
-
-
Klinge, C.M.1
Jernigan, S.C.2
Mattingly, K.A.3
Risinger, K.E.4
Zhang, J.5
-
127
-
-
0033618510
-
Peptide antagonists of the human estrogen receptor
-
J.D. Norris, L.A. Paige, D.J. Christensen, C.Y. Chang, M.R. Huacani, D. Fan, P.T. Hamilton, D.M. Fowlkes, and D.P. McDonnell. Peptide antagonists of the human estrogen receptor. Science 285: 744-746 (1999).
-
(1999)
Science
, vol.285
, pp. 744-746
-
-
Norris, J.D.1
Paige, L.A.2
Christensen, D.J.3
Chang, C.Y.4
Huacani, M.R.5
Fan, D.6
Hamilton, P.T.7
Fowlkes, D.M.8
McDonnell, D.P.9
-
128
-
-
0032807750
-
A novel role for helix 12 of retinoid X receptor in regulating repression
-
J. Zhang, X. Hu, and M.A. Lazar. A novel role for helix 12 of retinoid X receptor in regulating repression. Mol. Cell Biol. 19: 6448-6457 (1999).
-
(1999)
Mol. Cell Biol.
, vol.19
, pp. 6448-6457
-
-
Zhang, J.1
Hu, X.2
Lazar, M.A.3
-
129
-
-
70350602531
-
Comparison of in vitro hormone activities of selected phthalates using reporter gene assays
-
O. Shen, G. Du, H. Sun,W.Wu, Y. Jiang, L. Song, and X.Wang. Comparison of in vitro hormone activities of selected phthalates using reporter gene assays. Toxicol. Lett. 191: 9-14 (2009).
-
(2009)
Toxicol. Lett.
, vol.191
, pp. 9-14
-
-
Shen, O.1
Du, G.2
Sun, H.3
Wu, W.4
Jiang, Y.5
Song, L.6
Wang, X.7
-
130
-
-
0142211276
-
Identification and characterization of a ligand-regulated nuclear export signal in androgen receptor
-
A.J. Saporita, Q. Zhang, N. Navai, Z. Dincer, J. Hahn, X. Cai, and Z.Wang. Identification and characterization of a ligand-regulated nuclear export signal in androgen receptor. J. Biol. Chem. 278: 41998-42005 (2003).
-
(2003)
J. Biol. Chem.
, vol.278
, pp. 41998-42005
-
-
Saporita, A.J.1
Zhang, Q.2
Navai, N.3
Dincer, Z.4
Hahn, J.5
Cai, X.6
Wang, Z.7
-
131
-
-
0034663560
-
A natural sequence consisting of overlapping glucocorticoid-responsive elements mediates glucocorticoid, but not androgen, regulation of gene expression
-
C. Massaad, M. Garlatti, E.M. Wilson, F. Cadepond, and R. Barouki. A natural sequence consisting of overlapping glucocorticoid-responsive elements mediates glucocorticoid, but not androgen, regulation of gene expression. Biochem. J. 350 Pt 1: 123-129 (2000).
-
(2000)
Biochem. J.
, vol.350
, Issue.PART 1
, pp. 123-129
-
-
Massaad, C.1
Garlatti, M.2
Wilson, E.M.3
Cadepond, F.4
Barouki, R.5
-
132
-
-
67449092061
-
Regulation of activities of steroid hormone receptors by tibolone and its primary metabolites
-
A. Escande, N. Servant, F. Rabenoelina, G. Auzou, H. Kloosterboer, V. Cavailles, P. Balaguer, and T. Maudelonde. Regulation of activities of steroid hormone receptors by tibolone and its primary metabolites. J. Steroid Biochem.Mol. Biol. 116: 8-14 (2009).
-
(2009)
J. Steroid Biochem. Mol. Biol.
, vol.116
, pp. 8-14
-
-
Escande, A.1
Servant, N.2
Rabenoelina, F.3
Auzou, G.4
Kloosterboer, H.5
Cavailles, V.6
Balaguer, P.7
Maudelonde, T.8
-
133
-
-
0242351903
-
Antiandrogenic activity of the phytoestrogens naringenin, 6-(1,1-dimethylallyl)naringenin and 8-prenylnaringenin
-
O. Zierau, C. Morrissey, R.W. Watson, P. Schwab, S. Kolba, P. Metz, and G. Vollmer. Antiandrogenic activity of the phytoestrogens naringenin, 6-(1,1-dimethylallyl)naringenin and 8-prenylnaringenin. Planta Med. 69: 856-858 (2003).
-
(2003)
Planta Med
, vol.69
, pp. 856-858
-
-
Zierau, O.1
Morrissey, C.2
Watson, R.W.3
Schwab, P.4
Kolba, S.5
Metz, P.6
Vollmer, G.7
-
134
-
-
0343851745
-
A stable prostatic bioluminescent cell line to investigate androgen and antiandrogen effects
-
B. Terouanne, B. Tahiri, V. Georget, C. Belon, N. Poujol, C. Avances, F. Orio, Jr., P. Balaguer, and C. Sultan. A stable prostatic bioluminescent cell line to investigate androgen and antiandrogen effects. Mol. Cell Endocrinol. 160: 39-49 (2000).
-
(2000)
Mol. Cell Endocrinol.
, vol.160
, pp. 39-49
-
-
Terouanne, B.1
Tahiri, B.2
Georget, V.3
Belon, C.4
Poujol, N.5
Avances, C.6
Orio Jr., F.7
Balaguer, P.8
Sultan, C.9
-
135
-
-
0002302132
-
Adrenocorticotropic hormone; adrenocortical steroids and their synthetic analogs; inhibitors of the synthesis and actions of adrenocortical hormones
-
10th ed., J.G. Hardman, L.E. Limbird, and A.G. Gilman, Eds. McGraw-Hill, New York, NY
-
B.P. Schimmer and K.L. Parker. Adrenocorticotropic hormone; adrenocortical steroids and their synthetic analogs; inhibitors of the synthesis and actions of adrenocortical hormones. In Goodman and Gilman's The Pharmacological Basis of Therapeutics, 10th ed., J.G. Hardman, L.E. Limbird, and A.G. Gilman, Eds. McGraw-Hill, New York, NY, 2001, pp 1649-1677.
-
(2001)
Goodman and Gilman's The Pharmacological Basis of Therapeutics
, pp. 1649-1677
-
-
Schimmer, B.P.1
Parker, K.L.2
|