메뉴 건너뛰기




Volumn 16, Issue 11, 2011, Pages 9386-9396

Antimicrobial prospect of newly synthesized 1,3-thiazole derivatives

Author keywords

1,3 thiazoles; Antimicrobial evaluation; benzo d thiazoles; Partition coefficient; Synthesis

Indexed keywords

ANTIINFECTIVE AGENT; THIAZOLE DERIVATIVE;

EID: 82255189882     PISSN: None     EISSN: 14203049     Source Type: Journal    
DOI: 10.3390/molecules16119386     Document Type: Article
Times cited : (46)

References (29)
  • 1
    • 0034214238 scopus 로고    scopus 로고
    • The bactericidal action of penicillin: New clues to an unsolved mystery
    • DOI 10.1016/S0966-842X(00)01762-5, PII S0966842X00017625
    • Bayles, K.W. The bactericidal action of penicillin: New clues to an unsolved mystery. Trends Microbiol. 2000, 8, 274-278. (Pubitemid 30331001)
    • (2000) Trends in Microbiology , vol.8 , Issue.6 , pp. 274-278
    • Bayles, K.W.1
  • 2
    • 0029015927 scopus 로고
    • Bacteremia due to viridans streptococci that are highly resistant to penicillin: Increase among neutropenic patients with cancer
    • Carratala, J.; Alcaide, F.; Fernandez, S.A. Bacteremia due to viridans streptococci that are highly resistant to penicillin: Increase among neutropenic patients with cancer. Clin. Infect. Dis. 1995, 20, 1169-1173.
    • (1995) Clin. Infect. Dis. , vol.20 , pp. 1169-1173
    • Carratala, J.1    Alcaide, F.2    Fernandez, S.A.3
  • 3
    • 0026780099 scopus 로고
    • Results of the National Institute of Allergy and Infectious Diseases Collaborative Clinical Trial to test the predictive value of skin testing with major and minor penicillin derivatives in hospitalized adults
    • Sogn, D.D.; Evans, R.; Shepherd, G.M. Results of the National Institute of Allergy and Infectious Diseases Collaborative Clinical Trial to test the predictive value of skin testing with major and minor penicillin derivatives in hospitalized adults. Arch. Intern. Med. 1992, 152, 1025-1032.
    • (1992) Arch. Intern. Med. , vol.152 , pp. 1025-1032
    • Sogn, D.D.1    Evans, R.2    Shepherd, G.M.3
  • 4
    • 0028939128 scopus 로고
    • Diminished Activity of Ceftizoxime in Comparison to Cefotaxime and Ceftriaxone Against Streptococcus pneumoniae
    • Haas, D.W.; Stratton, C.W.; Griffin, J.P.; Weeks, L.; Alls, S.C. Diminished Activity of Ceftizoxime in Comparison to Cefotaxime and Ceftriaxone Against Streptococcus pneumoniae. Clin. Infect. Dis. 1995, 20, 671-676.
    • (1995) Clin. Infect. Dis. , vol.20 , pp. 671-676
    • Haas, D.W.1    Stratton, C.W.2    Griffin, J.P.3    Weeks, L.4    Alls, S.C.5
  • 5
    • 0028118473 scopus 로고
    • Treatment failure with use of a third-generation cephalosporin for penicillin-resistant pneumococcal meningitis: Case report and review
    • John, C.C. Treatment Failure with Use of a Third-Generation Cephalosporin for Penicillin- Resistant Pneumococcal Meningitis: Case Report and Review. Clin. Infect. Dis. 1994, 18, 188-193. (Pubitemid 24055257)
    • (1994) Clinical Infectious Diseases , vol.18 , Issue.2 , pp. 188-193
    • John, C.C.1
  • 7
    • 1842484230 scopus 로고    scopus 로고
    • The development of the antitumour benzothiazole prodrug, phortress, as a clinical candidate
    • DOI 10.2174/0929867043455530
    • Bradshaw, T.D.; Westwell, A.D. The development of the antitumour benzothiazole prodrug, Phortress, as a clinical candidate. Curr. Med. Chem. 2004, 11, 1009-1021. (Pubitemid 38428650)
    • (2004) Current Medicinal Chemistry , vol.11 , Issue.8 , pp. 1009-1021
    • Bradshaw, T.D.1    Westwell, A.D.2
  • 8
    • 0037203997 scopus 로고    scopus 로고
    • Antitumor benzothiazoles. 16. Synthesis and pharmaceutical properties of antitumor 2-(4-aminophenyl)benzothiazole amino acid prodrugs
    • DOI 10.1021/jm011025r
    • Hutchinson, I.; Jennings, S.A.; Vishnuvajjala, B.R.; Westwell, A.D.; Stevens, M.F.G. Antitumor benzothiazoles. 16. Synthesis and pharmaceutical properties of antitumor 2-(4- aminophenyl)benzothiazole amino acid prodrugs. J. Med. Chem. 2002, 45, 744-747. (Pubitemid 34145721)
    • (2002) Journal of Medicinal Chemistry , vol.45 , Issue.3 , pp. 744-747
    • Hutchinson, I.1    Jennings, S.A.2    Vishnuvajjala, B.R.3    Westwell, A.D.4    Stevens, M.F.G.5
  • 9
    • 0035953321 scopus 로고    scopus 로고
    • Antitumor benzothiazoles. 14. Synthesis and in vitro biological properties of fluorinated 2-(4-aminophenyl)benzothiazoles
    • DOI 10.1021/jm001104n
    • Hutchinson, I.; Chua, M.S.; Browne, H.L.; Trapani, V.; Bradshaw, T.D.; Westwell, A.D.; Stevens, M.F.G. Antitumor benzothiazoles. 14. Synthesis and in vitro biological properties of fluorinated 2- (4-aminophenyl)benzothiazoles. J. Med. Chem. 2001, 44, 1446-1455. (Pubitemid 32852121)
    • (2001) Journal of Medicinal Chemistry , vol.44 , Issue.9 , pp. 1446-1455
    • Hutchinson, I.1    Chua, M.-S.2    Browne, H.L.3    Trapani, V.4    Bradshaw, T.D.5    Westwell, A.D.6    Stevens, M.F.G.7
  • 11
    • 1542285110 scopus 로고    scopus 로고
    • Synthesis and SAR of 2-arylbenzoxazoles, benzothiazoles and benzimidazoles as inhibitors of lysophosphatidic acid acyltransferase-β
    • DOI 10.1016/j.bmcl.2004.01.023, PII S0960894X04000745
    • Gong, B.Q.; Hong, F.; Kohm, C.; Bonham, L.; Klein, P. Synthesis and SAR of 2-arylbenzoxazoles, benzothiazoles and benzimidazoles as inhibitors of lysophosphatidic acid acyltransferase-beta. Bioorg. Med. Chem. Lett. 2004, 14, 1455-1459. (Pubitemid 38299428)
    • (2004) Bioorganic and Medicinal Chemistry Letters , vol.14 , Issue.6 , pp. 1455-1459
    • Gong, B.1    Hong, F.2    Kohm, C.3    Bonham, L.4    Klein, P.5
  • 12
    • 0037325622 scopus 로고    scopus 로고
    • Antitumour benzothiazoles. Part 20: 3′-cyano and 3′-alkynyl-substituted 2-(4′-aminophenyl)benzothiazoles as new potent and selective analogues
    • DOI 10.1016/S0960-894X(02)00930-7, PII S0960894X02009307
    • Hutchinson, I.; Bradshaw, T.D.; Matthews, C.S.; Stevens, M.F.G.; Westwell, A.D. Antitumour benzothiazoles. Part 20: 3'-cyano and 3'-alkynyl-substituted 2-(4'-aminophenyl)benzothiazoles as new potent and selective analogues. Bioorg. Med. Chem. Lett. 2003, 13, 471-474. (Pubitemid 36259716)
    • (2003) Bioorganic and Medicinal Chemistry Letters , vol.13 , Issue.3 , pp. 471-474
    • Hutchinson, I.1    Bradshaw, T.D.2    Matthews, C.S.3    Stevens, M.F.G.4    Westwell, A.D.5
  • 13
    • 0038745928 scopus 로고    scopus 로고
    • Synthesis and HIV-1 reverse transcriptase inhibitor activity of some 2,5,6-substituted benzoxazole, benzimidazole, benzothiazole and oxazolo (4,5-b)pyridine derivatives
    • Akbay, A.; Ören, I.; Arpaci, Ö.T.; Sener E.A.; Yalçin, I. Synthesis and HIV-1 Reverse Transcriptase Inhibitor Activity of Some 2,5,6-Substituted Benzoxazole, Benzimidazole, Benzothiazole and Oxazolo(4,5-b)pyridine Derivatives. Arzneimittel-Forsch. 2003, 53, 266-271. (Pubitemid 36535382)
    • (2003) Arzneimittel-Forschung/Drug Research , vol.53 , Issue.4 , pp. 266-271
    • Akbay, A.1    Oren, I.2    Temiz-Arpaci, O.3    Aki-Sener, E.4    Yalcin, I.5
  • 17
    • 0014603468 scopus 로고
    • Heterocyclic substituted ureas. II. Immunosuppressive and antiviral activity of benzothiazolyl- and benzoxazolylureas
    • Paget, C.J.; Kisner, K.; Stone, R.L.; DeLong, D.C. Heterocyclic substituted ureas. II. Immunosuppressive and antiviral activity of benzothiazolyl- and benzoxazolylureas. J. Med. Chem. 1969, 12, 1016-1018.
    • (1969) J. Med. Chem. , vol.12 , pp. 1016-1018
    • Paget, C.J.1    Kisner, K.2    Stone, R.L.3    Delong, D.C.4
  • 18
    • 79959581305 scopus 로고    scopus 로고
    • Synthesis, characterization, and antimicrobial evaluation of oxadiazole congeners
    • Sadek, B.; Fahelelbom, K.M.S. Synthesis, Characterization, and Antimicrobial Evaluation of Oxadiazole Congeners. Molecules 2011, 16, 4339-4347.
    • (2011) Molecules , vol.16 , pp. 4339-4347
    • Sadek, B.1    Fahelelbom, K.M.S.2
  • 19
    • 79957500537 scopus 로고    scopus 로고
    • Synthesis and antimicrobial activities of hexahydroimidazo[1,5-a] pyridinium bromides with varying benzyl substituents
    • Türkmen, H.; Ceyhan, N.; Ulkü Karabay Yavaolu, N.; Ozdemir, G.; Cetinkaya, B. Synthesis and antimicrobial activities of hexahydroimidazo[1,5-a] pyridinium bromides with varying benzyl substituents. Eur. J. Med. Chem. 2011, 46, 2895-2900.
    • (2011) Eur. J. Med. Chem. , vol.46 , pp. 2895-2900
    • Türkmen, H.1    Ceyhan, N.2    Ulkü3    Karabay Yavaolu, N.4    Ozdemir, G.5    Cetinkaya, B.6
  • 20
    • 79955048920 scopus 로고    scopus 로고
    • The antimicrobial activity of inert oligonuclear polypyridylruthenium(ii) complexes against pathogenic bacteria, including MRSA
    • Li, F.; Mulyana, Y.; Feterl, M.; Warner, J.M.; Collins, J.G.; Keene, F.R. The antimicrobial activity of inert oligonuclear polypyridylruthenium(ii) complexes against pathogenic bacteria, including MRSA. Dalton Trans. 2011, 40, 5032-5038.
    • (2011) Dalton Trans. , vol.40 , pp. 5032-5038
    • Li, F.1    Mulyana, Y.2    Feterl, M.3    Warner, J.M.4    Collins, J.G.5    Keene, F.R.6
  • 21
    • 82255161057 scopus 로고    scopus 로고
    • Quantitative structure activity relationship studies for new antimicrobial N2- substituted phenazines
    • Fahelelbom, K.M.S.; Al-Tabakha, M. Quantitative structure activity relationship studies for new antimicrobial N2- substituted phenazines. Afr. J. Pharm. Pharmacol. 2009, 3, 47-50.
    • (2009) Afr. J. Pharm. Pharmacol. , vol.3 , pp. 47-50
    • Fahelelbom, K.M.S.1    Al-Tabakha, M.2
  • 22
    • 54949087200 scopus 로고    scopus 로고
    • The effect of lipophilicity on the antibacterial activity of some 1-benzylbenzimidazole derivatives
    • Podunavac-Kuzmanović, S.O.; Cvetković, D.D.; Barn, D.J. The effect of lipophilicity on the antibacterial activity of some 1-benzylbenzimidazole derivatives. J. Serb. Chem. Soc. 2008, 73, 967-978.
    • (2008) J. Serb. Chem. Soc. , vol.73 , pp. 967-978
    • Podunavac-Kuzmanović, S.O.1    Cvetković, D.D.2    Barn, D.J.3
  • 25
    • 0013494728 scopus 로고
    • Demethylation of aryl methyl ethers by boron tribromide
    • Mcomie, J.F.W.; Watts, M.L.; West, D.E. Demethylation of aryl methyl ethers by boron tribromide. Tetrahedron 1969, 24, 2289-2292.
    • (1969) Tetrahedron , vol.24 , pp. 2289-2292
    • McOmie, J.F.W.1    Watts, M.L.2    West, D.E.3
  • 27
    • 58949083707 scopus 로고    scopus 로고
    • Naturally occurring phenolic antibacterial compounds show effectiveness against oral bacteria by a quantitative structure-activity relationship study
    • Greenberg, M.; Dodds, M.; Tian, M. Naturally occurring phenolic antibacterial compounds show effectiveness against oral bacteria by a quantitative structure-activity relationship study. J. Agric. Food Chem. 2008, 56, 11151-11156.
    • (2008) J. Agric. Food Chem. , vol.56 , pp. 11151-11156
    • Greenberg, M.1    Dodds, M.2    Tian, M.3
  • 29
    • 82255161059 scopus 로고    scopus 로고
    • Biol. Abstr., 64, 25183.
    • Biol. Abstr. , vol.64 , pp. 25183


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.