Synthesis and SAR of 2-arylbenzoxazoles, benzothiazoles and benzimidazoles as inhibitors of lysophosphatidic acid acyltransferase-β

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 6, 2004, Pages 1455-1459

  Gong, Baoqing ^a   Hong, Feng ^a   Kohm, Cory ^a   Bonham, Lynn ^a   Klein, Peter ^a  

^a Cell Therapeutics Inc   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ACYLTRANSFERASE; ANTINEOPLASTIC AGENT; BENZIMIDAZOLE DERIVATIVE; BENZOTHIAZOLE DERIVATIVE; BENZOXAZOLE DERIVATIVE; LYSOPHOSPHATIDIC ACID;

ARTICLE; CELL PROLIFERATION; DRUG EFFECT; DRUG IDENTIFICATION; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IN VITRO STUDY; NONHUMAN; STRUCTURE ACTIVITY RELATION; TUMOR CELL;

ACYLTRANSFERASES; BENZIMIDAZOLES; BENZOTHIAZOLES; BENZOXAZOLES; CELL LINE, TUMOR; ENZYME INHIBITORS; HUMANS; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

EID: 1542285110     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.01.023     Document Type: Article

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