메뉴 건너뛰기




Volumn 339, Issue 3, 2011, Pages 952-958

Effects of ranolazine on cloned cardiac Kv4.3 potassium channels

Author keywords

[No Author keywords available]

Indexed keywords

POTASSIUM CHANNEL KV4.3; RANOLAZINE; SHAL POTASSIUM CHANNEL; UNCLASSIFIED DRUG;

EID: 81555204275     PISSN: 00223565     EISSN: 15210103     Source Type: Journal    
DOI: 10.1124/jpet.111.184176     Document Type: Article
Times cited : (5)

References (47)
  • 3
    • 4344577023 scopus 로고    scopus 로고
    • Electrophysiological effects of ranolazine, a novel antianginal agent with antiarrhythmic properties
    • DOI 10.1161/01.CIR.0000139333.83620.5D
    • Antzelevitch C, Belardinelli L, Zygmunt AC, Burashnikov A, Di Diego JM, Fish JM, Cordeiro JM, and Thomas G (2004b) Electrophysiological effects of ranolazine, a novel antianginal agent with antiarrhythmic properties. Circulation 110:904-910. (Pubitemid 39136212)
    • (2004) Circulation , vol.110 , Issue.8 , pp. 904-910
    • Antzelevitch, C.1    Belardinelli, L.2    Zygmunt, A.C.3    Burashnikov, A.4    Di, D.J.M.5    Fish, J.M.6    Cordeiro, J.M.7    Thomas, G.8
  • 4
    • 0032494172 scopus 로고    scopus 로고
    • Functional knockout of the transient outward current, long-QT syndrome, and cardiac remodeling in mice expressing a dominant-negative Kv4 α subunit
    • Barry DM, Xu H, Schuessler RB, and Nerbonne JM (1998) Functional knockout of the transient outward current, long-QT syndrome, and cardiac remodeling in mice expressing a dominant-negative Kv4 α subunit. Circ Res 83:560-567. (Pubitemid 28411058)
    • (1998) Circulation Research , vol.83 , Issue.5 , pp. 560-567
    • Barry, D.M.1    Xu, H.2    Schuessler, R.B.3    Nerbonne, J.M.4
  • 5
    • 0020624782 scopus 로고
    • Lidocaine block of cardiac sodium channels
    • Bean BP, Cohen CJ, and Tsien RW (1983) Lidocaine block of cardiac sodium channels.J Gen Physiol 81:613-642.
    • (1983) J Gen Physiol , vol.81 , pp. 613-642
    • Bean, B.P.1    Cohen, C.J.2    Tsien, R.W.3
  • 7
    • 2342605426 scopus 로고    scopus 로고
    • Blockers of the Kv1.5 channel for the treatment ofatrial arrhythmias
    • Brendel J and Peukert S (2003) Blockers of the Kv1.5 channel for the treatment ofatrial arrhythmias. Curr Med Chem Cardiovasc Hematol Agents 1:273-287.
    • (2003) Curr Med Chem Cardiovasc Hematol Agents , vol.1 , pp. 273-287
    • Brendel, J.1    Peukert, S.2
  • 8
    • 0025263891 scopus 로고
    • Molecular mechanisms of local anesthesia:a review
    • Butterworth JF 4th and Strichartz GR (1990) Molecular mechanisms of local anesthesia:a review. Anesthesiology 72:711-734.
    • (1990) Anesthesiology , vol.72 , pp. 711-734
    • Butterworth IV, J.F.1    Strichartz, G.R.2
  • 9
    • 0038630449 scopus 로고    scopus 로고
    • Effects of flecainide and quinidine on Kv4.2 currents: Voltage dependence and role of S6 valines
    • DOI 10.1038/sj.bjp.0705199
    • Caballero R, Pourrier M, Schram G, Delpón E, Tamargo J, and Nattel S (2003) Effects of flecainide and quinidine on Kv4.2 currents: voltage dependence and role of S6 valines. Br J Pharmacol 138:1475-1484. (Pubitemid 36609643)
    • (2003) British Journal of Pharmacology , vol.138 , Issue.8 , pp. 1475-1484
    • Caballero, R.1    Pourrier, M.2    Schram, G.3    Delpon, E.4    Tamargo, J.5    Nattel, S.6
  • 10
    • 0036885781 scopus 로고    scopus 로고
    • Measuring antianginal drug efficacy using exercise testing for chronic angina: Improved exercise performance with ranolazine, a pFOX inhibitor
    • Chaitman BR (2002) Measuring antianginal drug efficacy using exercise testing for chronic angina: improved exercise performance with ranolazine, a pFOX inhibitor.Curr Probl Cardiol 27:527-555.
    • (2002) Curr Probl Cardiol , vol.27 , pp. 527-555
    • Chaitman, B.R.1
  • 11
    • 33744455453 scopus 로고    scopus 로고
    • Ranolazine for the treatment of chronic angina and potential use in other cardiovascular conditions
    • Chaitman BR (2006) Ranolazine for the treatment of chronic angina and potential use in other cardiovascular conditions. Circulation 113:2462-2472.
    • (2006) Circulation , vol.113 , pp. 2462-2472
    • Chaitman, B.R.1
  • 12
    • 0015016070 scopus 로고
    • Voltage clamp studies of a transient outward membrane current in gastropod neural somata
    • Connor JA and Stevens CF (1971) Voltage clamp studies of a transient outward membrane current in gastropod neural somata. J Physiol 213:21-30.
    • (1971) J Physiol , vol.213 , pp. 21-30
    • Connor, J.A.1    Stevens, C.F.2
  • 13
    • 0016792109 scopus 로고
    • Mechanism of frequency-dependent inhibition of sodium currents in frog myelinated nerve by the lidocaine derivative GEA
    • Courtney KR (1975) Mechanism of frequency-dependent inhibition of sodium currents in frog myelinated nerve by the lidocaine derivative GEA. J Pharmacol ExpTher 195:225-236.
    • (1975) J Pharmacol ExpTher , vol.195 , pp. 225-236
    • Courtney, K.R.1
  • 16
    • 9444282030 scopus 로고    scopus 로고
    • Interaction of ropivacaine with cloned cardiac Kv4.3/KChIP2.2 complexes
    • Friederich P and Solth A (2004) Interaction of ropivacaine with cloned cardiac Kv4.3/KChIP2.2 complexes. Anesthesiology 101:1347-1356. (Pubitemid 39564991)
    • (2004) Anesthesiology , vol.101 , Issue.6 , pp. 1347-1356
    • Friederich, P.1    Solth, A.2
  • 17
    • 34447250066 scopus 로고    scopus 로고
    • Regional and tissue specific transcript signatures of ion channel genes in the non-diseased human heart
    • DOI 10.1113/jphysiol.2006.126714
    • Gaborit N, Le Bouter S, Szuts V, Varro A, Escande D, Nattel S, and Demolombe S (2007) Regional and tissue specific transcript signatures of ion channel genes inthe non-diseased human heart. J Physiol 582:675-693. (Pubitemid 47040552)
    • (2007) Journal of Physiology , vol.582 , Issue.2 , pp. 675-693
    • Gaborit, N.1    Le, B.S.2    Szuts, V.3    Varro, A.4    Escande, D.5    Nattel, S.6    Demolombe, S.7
  • 18
    • 0025222445 scopus 로고
    • Mechanisms of potassium channel block in rat alveolar epithelial cells
    • Jacobs ER and DeCoursey TE (1990) Mechanisms of potassium channel block in rat alveolar epithelial cells. J Pharmacol Exp Ther 255:459-472.
    • (1990) J Pharmacol Exp Ther , vol.255 , pp. 459-472
    • Jacobs, E.R.1    DeCoursey, T.E.2
  • 19
    • 0023695849 scopus 로고
    • Lidocaine blocks Na, Ca and K currents of chick ventricular myocytes
    • Josephson IR (1988) Lidocaine blocks Na, Ca and K currents of chick ventricular myocytes. J Mol Cell Cardiol 20:593-604.
    • (1988) J Mol Cell Cardiol , vol.20 , pp. 593-604
    • Josephson, I.R.1
  • 20
    • 0034710954 scopus 로고    scopus 로고
    • Channel structure and drug-induced cardiac arrhythmias
    • Kass RS and Cabo C (2000) Channel structure and drug-induced cardiac arrhythmias.Proc Natl Acad Sci U S A 97:11683-11684.
    • (2000) Proc Natl Acad Sci U S A , vol.97 , pp. 11683-11684
    • Kass, R.S.1    Cabo, C.2
  • 21
    • 79952148405 scopus 로고    scopus 로고
    • Inhibition of Kv4.3 by genistein via a tyrosine phosphorylation- independent mechanism
    • Kim HJ, Ahn HS, Choi BH, and Hahn SJ (2011) Inhibition of Kv4.3 by genistein via a tyrosine phosphorylation-independent mechanism. Am J Physiol Cell Physiol 300:C567-C575.
    • (2011) Am J Physiol Cell Physiol , vol.300
    • Kim, H.J.1    Ahn, H.S.2    Choi, B.H.3    Hahn, S.J.4
  • 22
    • 0022551421 scopus 로고
    • Modulation of aminopyridine block of potassium currents in squid axon
    • Kirsch GE, Yeh JZ, and Oxford GS (1986) Modulation of aminopyridine block of potassium currents in squid axon. Biophys J 50:637-644. (Pubitemid 16028171)
    • (1986) Biophysical Journal , vol.50 , Issue.4 , pp. 637-644
    • Kirsch, G.E.1    Yeh, J.Z.2    Oxford, G.S.3
  • 23
    • 0021364788 scopus 로고
    • Combined effects of hypoxia, hyperkalemia and acidosis on membrane action potential and excitability of guinea-pig ventricular muscle
    • DOI 10.1016/S0022-2828(84)80591-X
    • Kodama I, Wilde A, Janse MJ, Durrer D, and Yamada K (1984) Combined effects of hypoxia, hyperkalemia and acidosis on membrane action potential and excitability of guinea-pig ventricular muscle. J Mol Cell Cardiol 16:247-259. (Pubitemid 14168016)
    • (1984) Journal of Molecular and Cellular Cardiology , vol.16 , Issue.3 , pp. 247-259
    • Kodama, I.1    Wilde, A.2    Janse, M.J.3
  • 25
    • 0141723313 scopus 로고    scopus 로고
    • The antianginal agent trimetazidine does not exert its functional benefit via inhibition of mitochondrial long-chain 3-ketoacyl coenzyme A thiolase
    • MacInnes A, Fairman DA, Binding P, Rhodes J, Wyatt MJ, Phelan A, Haddock PS, and Karran EH (2003) The antianginal agent trimetazidine does not exert its functional benefit via inhibition of mitochondrial long-chain 3-ketoacyl coenzyme A thiolase. Circ Res 93:e26-32.
    • (2003) Circ Res , vol.93
    • MacInnes, A.1    Fairman, D.A.2    Binding, P.3    Rhodes, J.4    Wyatt, M.J.5    Phelan, A.6    Haddock, P.S.7    Karran, E.H.8
  • 26
    • 0031971168 scopus 로고    scopus 로고
    • Ranolazine: A novel metabolic modulator for the treatment of angina
    • DOI 10.1016/S0306-3623(97)00301-7, PII S0306362397003017
    • McCormack JG, Stanley WC, and Wolff AA (1998) Ranolazine: a novel metabolic modulator for the treatment of angina. Gen Pharmacol 30:639-645. (Pubitemid 28167764)
    • (1998) General Pharmacology , vol.30 , Issue.5 , pp. 639-645
    • McCormack, J.G.1    Stanley, W.C.2    Wolff, A.A.3
  • 27
    • 0034213745 scopus 로고    scopus 로고
    • + channel diversity in the mammalian myocardium
    • + channel diversity in the mammalian myocardium. J Physiol 525:285-298.
    • (2000) J Physiol , vol.525 , pp. 285-298
    • Nerbonne, J.M.1
  • 29
    • 0032983310 scopus 로고    scopus 로고
    • A controlled trial with a novel anti-lschemic agent, ranolazine, in chronic stable angina pectoris that is responsive to conventional antianginal agents
    • DOI 10.1016/S0002-9149(99)00190-3, PII S0002914999001903
    • Pepine CJ and Wolff AA (1999) A controlled trial with a novel anti-ischemic agent, ranolazine, in chronic stable angina pectoris that is responsive to conventional antianginal agents. Ranolazine Study Group. Am J Cardiol 84:46-50. (Pubitemid 29307639)
    • (1999) American Journal of Cardiology , vol.84 , Issue.1 , pp. 46-50
    • Pepine, C.J.1    Wolff, A.A.2
  • 31
  • 34
    • 0028325440 scopus 로고
    • + channel blocking actions of flecainide compared with those of propafenone and quinidine in adult rat ventricular myocytes
    • + channel blocking actions of flecainide compared with those of propafenone and quinidine in adult rat ventricular myocytes. J Pharmacol Exp Ther 269:66-74.
    • (1994) J Pharmacol Exp Ther , vol.269 , pp. 66-74
    • Slawsky, M.T.1    Castle, N.A.2
  • 35
    • 0033017643 scopus 로고    scopus 로고
    • Structure and function of cardiac potassium channels
    • Snyders DJ (1999) Structure and function of cardiac potassium channels. Cardiovasc Res 42:377-390.
    • (1999) Cardiovasc Res , vol.42 , pp. 377-390
    • Snyders, D.J.1
  • 36
    • 0027321972 scopus 로고
    • A rapidly activating and slowly inactivating potassium channel cloned from human heart. Functional analysis after stable mammalian cell culture expression
    • Snyders DJ, Tamkun MM, and Bennett PB (1993) A rapidly activating and slowly inactivating potassium channel cloned from human heart. Functional analysis after stable mammalian cell culture expression. J Gen Physiol 101:513-543. (Pubitemid 23123420)
    • (1993) Journal of General Physiology , vol.101 , Issue.4 , pp. 513-543
    • Snyders, D.J.1    Tamkun, M.M.2    Bennett, P.B.3
  • 37
    • 0029130666 scopus 로고
    • Determinants of antiarrhythmic drug action. Electrostatic and hydrophobic components of block of the human cardiac hKv1.5 channel
    • Snyders DJ and Yeola SW (1995) Determinants of antiarrhythmic drug action. Electrostatic and hydrophobic components of block of the human cardiac hKv1.5 channel. Circ Res 77:575-583.
    • (1995) Circ Res , vol.77 , pp. 575-583
    • Snyders, D.J.1    Yeola, S.W.2
  • 38
    • 26244468710 scopus 로고    scopus 로고
    • V401I
    • DOI 10.1097/00000542-200510000-00018
    • Solth A, Siebrands CC, and Friederich P (2005) Inhibition of Kv4.3/KChIP2.2 channels by bupivacaine and its modulation by the pore mutation Kv4.3V401I. Anesthesiology 103:796-804. (Pubitemid 41415528)
    • (2005) Anesthesiology , vol.103 , Issue.4 , pp. 796-804
    • Solth, A.1    Siebrands, C.C.2    Friederich, P.3
  • 41
    • 40849140980 scopus 로고    scopus 로고
    • + channel isoforms by ranolazine
    • DOI 10.1124/mol.107.041541
    • Wang GK, Calderon J, and Wang SY (2008) State- and use-dependent block of muscle Nav1.4 and neuronal Nav1.7 voltage-gated Na- channel isoforms by ranolazine. Mol Pharmacol 73:940-948. (Pubitemid 351397898)
    • (2008) Molecular Pharmacology , vol.73 , Issue.3 , pp. 940-948
    • Ging, K.W.1    Calderon, J.2    Wang, S.-Y.3
  • 42
    • 0028838977 scopus 로고
    • Effects of flecainide, quinidine, and 4-aminopyridine on transient outward and ultrarapid delayed rectifier currents in human atrial myocytes
    • Wang Z, Fermini B, and Nattel S (1995) Effects of flecainide, quinidine, and 4-aminopyridine on transient outward and ultrarapid delayed rectifier currents in human atrial myocytes. J Pharmacol Exp Ther 272:184-196.
    • (1995) J Pharmacol Exp Ther , vol.272 , pp. 184-196
    • Wang, Z.1    Fermini, B.2    Nattel, S.3
  • 45
    • 73449119314 scopus 로고    scopus 로고
    • Voltage-gated potassium channels as therapeutic targets
    • Wulff H, Castle NA, and Pardo LA (2009) Voltage-gated potassium channels as therapeutic targets. Nat Rev Drug Discov 8:982-1001.
    • (2009) Nat Rev Drug Discov , vol.8 , pp. 982-1001
    • Wulff, H.1    Castle, N.A.2    Pardo, L.A.3
  • 46
    • 0017089418 scopus 로고
    • Dynamics of aminopyridine block of potassium channels in squid axon membrane
    • Yeh JZ, Oxford GS, Wu CH, and Narahashi T (1976) Dynamics of aminopyridine block of potassium channels in squid axon membrane. J Gen Physiol 68:519-535.
    • (1976) J Gen Physiol , vol.68 , pp. 519-535
    • Yeh, J.Z.1    Oxford, G.S.2    Wu, C.H.3    Narahashi, T.4
  • 47
    • 64549138059 scopus 로고    scopus 로고
    • Modulation of major voltage- And ligand-gated ion channels in cultured neurons of the rat inferior colliculus by lidocaine
    • Yu M and Chen L (2008) Modulation of major voltage- and ligand-gated ion channels in cultured neurons of the rat inferior colliculus by lidocaine. Acta Pharmacol Sin 29:1409-1418.
    • (2008) Acta Pharmacol Sin , vol.29 , pp. 1409-1418
    • Yu, M.1    Chen, L.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.