Pharmacology and selectivity of various natural and synthetic bombesin related peptide agonists for human and rat bombesin receptors differs

Peptides

Volumn 32, Issue 8, 2011, Pages 1685-1699

  Uehara, Hirotsugu ^a   González, Nieves ^a   Sancho, Veronica ^a   Mantey, Samuel A ^a   Nuche Berenguer, Bernardo ^a   Pradhan, Tapas ^a   Coy, David H ^b   Jensen, Robert T ^a  

^a NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES   (United States)

^b TULANE UNIVERSITY HEALTH SCIENCES CENTER   (United States)

Author keywords

Bombesin; Bombesin receptor; BRS 3; Gastrin releasing peptide; Gastrin releasing peptide receptor; Neuromedin B; Neuromedin B receptor; Peptide mediated cytotoxicity; PRRT; Satiety; Tumor imaging

Indexed keywords

ALYTESIN; BETA ALANINE; BOMBESIN; BOMBESIN DERIVATIVE; BOMBESIN RECEPTOR; GASTRIN RELEASING PEPTIDE DERIVATIVE; GASTRIN RELEASING PEPTIDE RECEPTOR; GASTRIN RELEASING PEPTIDE[14-27]; LITORIN; NEUROMEDIN B; NEUROMEDIN B[1-30]; NEUROMEDIN C; PHOSPHOLIPASE C; PHYLLOLITORIN; PSEUDOPHRYNE GUNTHERI LITORIN LIKE PEPTIDE; RANATENSIN; ROHDEI LITORIN; SYNTHETIC PEPTIDE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CELL ACTIVATION; CONCENTRATION RESPONSE; CONTROLLED STUDY; ENZYME ACTIVITY; HUMAN; HUMAN CELL; LIGAND BINDING; MOUSE; NONHUMAN; PHARMACOPHORE; PRIORITY JOURNAL; PROTEIN EXPRESSION; RAT; RECEPTOR AFFINITY; RECEPTOR BINDING;

3T3 CELLS; ANIMALS; CELL LINE, TUMOR; HUMANS; LIGANDS; MICE; MICE, INBRED BALB C; PEPTIDES; RATS; RECEPTORS, BOMBESIN; TRANSFECTION;

BOVINE RESPIRATORY SYNCYTIAL VIRUS; MAMMALIA; RATTUS; RODENTIA;

EID: 80051550769     PISSN: 01969781     EISSN: 18735169     Source Type: Journal    
DOI: 10.1016/j.peptides.2011.06.017     Document Type: Article

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