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Volumn 276, Issue 1, 2001, Pages 495-504

Tyrosine 220 in the 5th transmembrane domain of the neuromedin B receptor is critical for the high selectivity of the peptoid antagonist PD168368

(6) Tokita, Kenji a Hocart, Simon J b Katsuno, Tatsuro a Mantey, Samuel A a Coy, David H b Jensen, Robert T a

a NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES (United States)

b TULANE UNIVERSITY HEALTH SCIENCES CENTER (United States)

Author keywords

[No Author keywords available]

Indexed keywords

G PROTEIN COUPLED RECEPTOR; GASTRIN RELEASING PEPTIDE; HORMONE RECEPTOR BLOCKING AGENT; HYDROXYL GROUP; MEMBRANE PROTEIN; NEUROHORMONE; NEUROMEDIN B; NEUROMEDIN B RECEPTOR ANTAGONIST; PD 168368; PHENYLALANINE; TYROSINE; UNCLASSIFIED DRUG;

AMINO ACID SUBSTITUTION; ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SPECIFICITY; HYDROGEN BOND; MOUSE; NONHUMAN; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN PROTEIN INTERACTION; RECEPTOR AFFINITY; RECEPTOR SENSITIVITY; SITE DIRECTED MUTAGENESIS; TISSUE SPECIFICITY;

3T3 CELLS; AMINO ACID SEQUENCE; AMINO ACID SUBSTITUTION; ANIMALS; BINDING SITES; INDOLES; MICE; MODELS, MOLECULAR; MOLECULAR SEQUENCE DATA; MUTAGENESIS, SITE-DIRECTED; NEUROKININ B; PEPTIDES; PEPTOIDS; POINT MUTATION; PROTEIN BINDING; PROTEIN CONFORMATION; PROTEIN STRUCTURE, TERTIARY; PYRIDINES; RECEPTORS, BOMBESIN; RECOMBINANT FUSION PROTEINS; SUBSTRATE SPECIFICITY; TRANSFECTION; TYROSINE;

ANIMALIA;

EID: 0035808449 PISSN: 00219258 EISSN: None Source Type: Journal
DOI: 10.1074/jbc.M006059200 Document Type: Article

Times cited : (28)

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