Synthesis and biological evaluation of 125I-nebivolol as a potential cardioselective agent for imaging β1-adrenoceptors

Journal of Radioanalytical and Nuclear Chemistry

Volumn 289, Issue 1, 2011, Pages 239-245

  Motaleb, M A ^a   Moustapha, M E ^b   Ibrahim, I T ^a  

^a Atomic Energy Authority   (Egypt)

^b BENHA UNIVERSITY   (Egypt)

Author keywords

1 adrenoceptor selectivity; 125I nebivolol; Chloramine T; Iodonium; Molecular imaging; Myocardium

Indexed keywords

BETA 1 ADRENERGIC RECEPTOR; IODINE NEBIVOLOL I 125; NEBIVOLOL; OXIDIZING AGENT; RADIOLIGAND; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CARDIOSELECTIVITY; DRUG CLEARANCE; DRUG CONCENTRATION; DRUG DISTRIBUTION; DRUG SCREENING; DRUG SELECTIVITY; DRUG SPECIFICITY; DRUG STABILITY; DRUG SYNTHESIS; DRUG UPTAKE; ELECTROPHILIC SUBSTITUTION; HEPATOBILIARY SYSTEM; ISOTOPE LABELING; KIDNEY CLEARANCE; MOLECULAR IMAGING; NONHUMAN; PH; RADIOIODINATION; RAT; SUBSTITUTION REACTION; TEMPERATURE;

EID: 79959837510     PISSN: 02365731     EISSN: 15882780     Source Type: Journal    
DOI: 10.1007/s10967-011-1069-z     Document Type: Article

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