메뉴 건너뛰기




Volumn 37, Issue 7, 2010, Pages 727-740

Fluorine-18 radiopharmaceuticals beyond [18F]FDG for use in oncology and neurosciences

Author keywords

[No Author keywords available]

Indexed keywords

1 FLUORO 3 (2 NITRO 1 IMIDAZOLYL) 2 PROPANOL F 18; 3' FLUOROTHYMIDINE F 18; 6 FLUORODOPA F 18; AMINO ACID OXIDASE; BORON; CARBON 11; FLUORINE 18; FLUOROCHOLINE F 18; FLUORODEOXYGLUCOSE F 18; FLUOROTYROSINE F 18; PHOSPHORUS DERIVATIVE; SILICON; SODIUM FLUORIDE F 18; TRACER; UNCLASSIFIED DRUG;

EID: 77956991351     PISSN: 09698051     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.nucmedbio.2010.04.185     Document Type: Review
Times cited : (115)

References (105)
  • 1
    • 0017540177 scopus 로고
    • 18F-labeled 2-deoxy-2-fluoro-d-glucose as radiopharmaceutical for measuring regional myocardial glucose metabolism in vivo: tissue distribution and imaging studies in animals
    • 18F-labeled 2-deoxy-2-fluoro-d-glucose as radiopharmaceutical for measuring regional myocardial glucose metabolism in vivo: tissue distribution and imaging studies in animals. J Nucl Med 1977, 18:990-996.
    • (1977) J Nucl Med , vol.18 , pp. 990-996
    • Gallagher, B.M.1    Ansari, A.2    Atkins, H.3    Casella, V.4    Christman, D.R.5    Fowler, J.S.6
  • 2
    • 0022885139 scopus 로고
    • 18F]-fluoro-2-deoxy-d-glucose using aminopolyether supported nucleophilic substitution
    • 18F]-fluoro-2-deoxy-d-glucose using aminopolyether supported nucleophilic substitution. J Nucl Med 1986, 27:235-238.
    • (1986) J Nucl Med , vol.27 , pp. 235-238
    • Hamacher, K.1    Coenen, H.H.2    Stöcklin, G.3
  • 3
    • 79960733448 scopus 로고    scopus 로고
    • U.S.Department of Health and Human Services Food and Drug Administration Center for Drug Evaluation and Research (CDER)
    • U.S.Department of Health and Human Services Food and Drug Administration Center for Drug Evaluation and Research (CDER) Guidance: PET drugs-current good manufacturing practice (CGMP): December 2009 http://www.fda.gov/downloads/Drugs/GuidanceComplianceRegulatoryInformation/Guidances/ucm070306.pdf.
    • Guidance: PET drugs-current good manufacturing practice (CGMP): December 2009
  • 4
    • 34848871896 scopus 로고    scopus 로고
    • 18F-Labelled positron emission tomographic radiopharmaceuticals in oncology: an overview of radiochemistry and mechanism of tumor localization
    • 18F-Labelled positron emission tomographic radiopharmaceuticals in oncology: an overview of radiochemistry and mechanism of tumor localization. Sem Nucl Med 2007, 37:400-419.
    • (2007) Sem Nucl Med , vol.37 , pp. 400-419
    • Vallabhasojula, S.1
  • 5
    • 34249282333 scopus 로고    scopus 로고
    • Molecular imaging agents for clinical positron emission tomography in oncology other than fluorodeoxyglucose (FDG): applications, limitations and potential
    • Mercer J.R. Molecular imaging agents for clinical positron emission tomography in oncology other than fluorodeoxyglucose (FDG): applications, limitations and potential. J Pharm Pharmaceut Sci 2007, 10:180-202.
    • (2007) J Pharm Pharmaceut Sci , vol.10 , pp. 180-202
    • Mercer, J.R.1
  • 6
    • 77956991876 scopus 로고    scopus 로고
    • Radioisotope products and their availability
    • International Atomic Energy Agency
    • International Atomic Energy Agency Radioisotope products and their availability. Nuclear Technology Review 2010, 36. http://www-govatom.iaea.org/DocumentDetails.asp?Language=English&Path=f:/websites/govatom/govatomdocs/govdoc/2010/gov-2010-05/gov2010-5.doc.
    • (2010) Nuclear Technology Review , pp. 36
  • 11
    • 77957015504 scopus 로고    scopus 로고
    • International Atomic Energy Agency. [18F]Fluorodeoxyglucose (FDG): guidance for facility, production and quality control. IAEA Radioisotopes and Radiopharmaceuticals Series 3: [in press]
    • International Atomic Energy Agency. [18F]Fluorodeoxyglucose (FDG): guidance for facility, production and quality control. IAEA Radioisotopes and Radiopharmaceuticals Series 3: [in press].
  • 16
    • 0033059817 scopus 로고    scopus 로고
    • Calculation of positron range and its effect on the fundamental limit of positron emission tomography system spatial resolution
    • Levin C.S., Hoffman E.J. Calculation of positron range and its effect on the fundamental limit of positron emission tomography system spatial resolution. Phys Med Biol 1999, 44:781-791.
    • (1999) Phys Med Biol , vol.44 , pp. 781-791
    • Levin, C.S.1    Hoffman, E.J.2
  • 20
    • 0030810879 scopus 로고    scopus 로고
    • F-18 labeled fluorine gas for synthesis of tracer molecules
    • Bergman J., Solin O. F-18 labeled fluorine gas for synthesis of tracer molecules. Nucl Med Biol 1997, 24:677-683.
    • (1997) Nucl Med Biol , vol.24 , pp. 677-683
    • Bergman, J.1    Solin, O.2
  • 21
    • 0003002385 scopus 로고
    • Regiospecific aromatic fluorodemetallation of group IVb metalloarenes using elemental fluorine or acetyl hypofluorite
    • Coenen H.H., Moerlein S.M. Regiospecific aromatic fluorodemetallation of group IVb metalloarenes using elemental fluorine or acetyl hypofluorite. J Fluor Chem 1987, 36:63-75.
    • (1987) J Fluor Chem , vol.36 , pp. 63-75
    • Coenen, H.H.1    Moerlein, S.M.2
  • 25
    • 73249138886 scopus 로고    scopus 로고
    • Teflon radiolysis as the major source of carrier in fluorine-18
    • Berridge M.S., Apana S.M., Hersh J.M. Teflon radiolysis as the major source of carrier in fluorine-18. J Label Comp Radiopharm 2009, 52:543-548.
    • (2009) J Label Comp Radiopharm , vol.52 , pp. 543-548
    • Berridge, M.S.1    Apana, S.M.2    Hersh, J.M.3
  • 26
    • 33845592524 scopus 로고    scopus 로고
    • 2 reactions catalyzed by protic solvents: Facile fluorination for isotopic labeling of diagnostic molecules
    • 2 reactions catalyzed by protic solvents: Facile fluorination for isotopic labeling of diagnostic molecules. J Am Chem Soc 2006, 128:16394-16397.
    • (2006) J Am Chem Soc , vol.128 , pp. 16394-16397
    • Kim, D.W.1    Ahn, D.S.2    Oh, Y.H.3    Lee, S.4    Kil, H.S.5    Oh, S.J.6
  • 28
    • 44849114508 scopus 로고    scopus 로고
    • Springer, P.A. Schubiger, L. Lehmann, M. Friebe (Eds.)
    • PET Chemistry 2007, Springer. P.A. Schubiger, L. Lehmann, M. Friebe (Eds.).
    • (2007) PET Chemistry
  • 29
    • 36249019306 scopus 로고    scopus 로고
    • 18F-fluoroalkyl agents: synthesis, reactivity and application for development of PET-ligands in molecular imaging
    • 18F-fluoroalkyl agents: synthesis, reactivity and application for development of PET-ligands in molecular imaging. Curr Top Med Chem 2007, 7:1817-1828.
    • (2007) Curr Top Med Chem , vol.7 , pp. 1817-1828
    • Zhang, M.R.1    Suzuki, K.2
  • 30
    • 0028471146 scopus 로고
    • 18F]fluorobenzoate and its application to the labeling of a monoclonal antibody fragment
    • 18F]fluorobenzoate and its application to the labeling of a monoclonal antibody fragment. Bioconjug Chem 1994, 5:352-356.
    • (1994) Bioconjug Chem , vol.5 , pp. 352-356
    • Vaidyanathan, G.1    Zalutsky, R.2
  • 31
    • 0029945878 scopus 로고    scopus 로고
    • A comparative study of NCA fluorine-18 labelling of proteins via acylation and photochemical conjugation
    • Wester H.J., Hamacher K., Stoecklin G. A comparative study of NCA fluorine-18 labelling of proteins via acylation and photochemical conjugation. Nucl Med Biol 1996, 23:365-372.
    • (1996) Nucl Med Biol , vol.23 , pp. 365-372
    • Wester, H.J.1    Hamacher, K.2    Stoecklin, G.3
  • 34
    • 0037099395 scopus 로고    scopus 로고
    • A stepwise Huisgen cycloaddition process: copper(I)-catalyzed regioselective "ligation" of azides and terminal alkynes
    • Rostovtsev V.V., Green L.G., Folkin V.V., Sharpless B.K. A stepwise Huisgen cycloaddition process: copper(I)-catalyzed regioselective "ligation" of azides and terminal alkynes. Angew Chem Int Ed 2002, 41:2596-2599.
    • (2002) Angew Chem Int Ed , vol.41 , pp. 2596-2599
    • Rostovtsev, V.V.1    Green, L.G.2    Folkin, V.V.3    Sharpless, B.K.4
  • 38
    • 29144528086 scopus 로고    scopus 로고
    • Multistep synthesis of a radiolabeled imaging probe using integrated microfluidics
    • Lee C.C., Sui G., Elizarov A., Shu C.J., Shin Y.S., Dooley A.N., et al. Multistep synthesis of a radiolabeled imaging probe using integrated microfluidics. Science 2005, 16:1793-1796.
    • (2005) Science , vol.16 , pp. 1793-1796
    • Lee, C.C.1    Sui, G.2    Elizarov, A.3    Shu, C.J.4    Shin, Y.S.5    Dooley, A.N.6
  • 44
    • 77957003947 scopus 로고    scopus 로고
    • Special Issue on 'positron emission tomography with fluorine-18 agents other than fluorodeoxyglucose'
    • Special Issue on 'positron emission tomography with fluorine-18 agents other than fluorodeoxyglucose'. Sem Nucl Med 2007, 37:399-488.
    • (2007) Sem Nucl Med , vol.37 , pp. 399-488
  • 45
    • 34848895720 scopus 로고    scopus 로고
    • 18F-Fluoride positron emission tomography and positron emission tomography/computed tomography
    • 18F-Fluoride positron emission tomography and positron emission tomography/computed tomography. Sem Nucl Med 2007, 462-469.
    • (2007) Sem Nucl Med , pp. 462-469
    • Even-Sapir, E.1    Mishani, E.2    Flusser, G.3    Metser, U.R.4
  • 46
    • 70449523074 scopus 로고    scopus 로고
    • 18F]sodium fluoride for injection, USP to address the technetium-99m isotope shortage
    • 18F]sodium fluoride for injection, USP to address the technetium-99m isotope shortage. Appl Radiat Isot 2010, 117-119.
    • (2010) Appl Radiat Isot , pp. 117-119
    • Hockley, B.G.1    Scott, J.H.2
  • 52
    • 33847291423 scopus 로고    scopus 로고
    • 18F-fluorocyclobutane-1-carboxylic acid with PET/CT in prostate carcinoma
    • 18F-fluorocyclobutane-1-carboxylic acid with PET/CT in prostate carcinoma. J Nucl Med 2007, 48:56-63.
    • (2007) J Nucl Med , vol.48 , pp. 56-63
    • Schuster, D.M.1    Votaw, J.R.2    Nieh, P.T.3
  • 59
    • 0001976894 scopus 로고    scopus 로고
    • Automated synthesis of fluorine-18 labeled choline analogue: 2-fluoroetheyl-dimethyl-2-oxyethylammonium
    • Hara T., Yuasa M. Automated synthesis of fluorine-18 labeled choline analogue: 2-fluoroetheyl-dimethyl-2-oxyethylammonium. J Nucl Med 1997, 38(Supplement):44P.
    • (1997) J Nucl Med , vol.38 , Issue.SUPPL.
    • Hara, T.1    Yuasa, M.2
  • 62
    • 0036172994 scopus 로고    scopus 로고
    • 18F-fluoroethylcholine for cancer imaging with PET: synthesis, biochemistry, and prostate cancer imaging
    • 18F-fluoroethylcholine for cancer imaging with PET: synthesis, biochemistry, and prostate cancer imaging. J Nucl Med 2002, 43:187-199.
    • (2002) J Nucl Med , vol.43 , pp. 187-199
    • Hara, T.1    Kosaka, N.2    Kishi, H.3
  • 69
    • 0024551844 scopus 로고
    • 18F]fluoro-1-(2-nitro-1-imidazolyl)-2-propanol. A potential PET agent for detecting hypoxic but viable tissues
    • 18F]fluoro-1-(2-nitro-1-imidazolyl)-2-propanol. A potential PET agent for detecting hypoxic but viable tissues. Int J Radiat Appl Instrum [A] 1989, 40:117-126.
    • (1989) Int J Radiat Appl Instrum [A] , vol.40 , pp. 117-126
    • Hwang, D.R.1    Dence, C.S.2    Bonasera, T.A.3    Welch, M.J.4
  • 75
    • 0030272778 scopus 로고    scopus 로고
    • The use of 3-methoxymethyl-16 beta, 17 beta-epiestriol-O-cyclic sulfone as the precursor in the synthesis of F-18 16 alpha-fluoroestradiol
    • Lim J.L., Zheng L., Berridge M.S., Tewson T.J. The use of 3-methoxymethyl-16 beta, 17 beta-epiestriol-O-cyclic sulfone as the precursor in the synthesis of F-18 16 alpha-fluoroestradiol. Nucl Med Biol 1996, 23:911-915.
    • (1996) Nucl Med Biol , vol.23 , pp. 911-915
    • Lim, J.L.1    Zheng, L.2    Berridge, M.S.3    Tewson, T.J.4
  • 76
    • 18244428952 scopus 로고    scopus 로고
    • 18F]FHBG): a new potential imaging agent for viral infection and gene therapy using PET
    • 18F]FHBG): a new potential imaging agent for viral infection and gene therapy using PET. Nucl Med Biol 1998, 25:175-180.
    • (1998) Nucl Med Biol , vol.25 , pp. 175-180
    • Alauddin, M.M.1    Conti, P.S.2
  • 77
    • 77957007226 scopus 로고    scopus 로고
    • Springer-Verlag London Limited
    • Wagner H.N. Brain Imaging 2009, Springer-Verlag London Limited.
    • (2009) Brain Imaging
    • Wagner, H.N.1
  • 80
    • 0028964653 scopus 로고
    • 18F]fluoropropyl)-2,3-dimethoxybenzamide as an improved dopamine D-2 receptor tracer
    • 18F]fluoropropyl)-2,3-dimethoxybenzamide as an improved dopamine D-2 receptor tracer. Nucl Med Biol 1995, 22:283-296.
    • (1995) Nucl Med Biol , vol.22 , pp. 283-296
    • Mukherjee, J.1    Yang, Z.Y.2    Das, M.K.3    Brown, T.4
  • 87
    • 0029981856 scopus 로고    scopus 로고
    • 18F]DOPA-PET and clinical study of the rate of the progression in Parkinson's disease
    • 18F]DOPA-PET and clinical study of the rate of the progression in Parkinson's disease. Brain 1996, 119:585-591.
    • (1996) Brain , vol.119 , pp. 585-591
    • Morrish, P.K.1    Sawle, G.V.2    Brooks, D.J.3
  • 88
    • 0842286829 scopus 로고    scopus 로고
    • The sensitivity of 18-fluorodopa positron emission tomography and magnetic resonance imaging in Parkinson's disease
    • Heiss W.D., Hilker R. The sensitivity of 18-fluorodopa positron emission tomography and magnetic resonance imaging in Parkinson's disease. Eur J Neurol 2004, 11:5-12.
    • (2004) Eur J Neurol , vol.11 , pp. 5-12
    • Heiss, W.D.1    Hilker, R.2
  • 94
    • 0026355999 scopus 로고
    • Fluorine-18-altanserin: a radioligand for the study of serotonin receptors with PET: radiolabeling and in vivo biologic behavior in rats
    • Lemaire C., Cantineau R., Guillaume M., Plenevaux A., Christiaens L. Fluorine-18-altanserin: a radioligand for the study of serotonin receptors with PET: radiolabeling and in vivo biologic behavior in rats. J Nucl Med 1991, 32:2266-2272.
    • (1991) J Nucl Med , vol.32 , pp. 2266-2272
    • Lemaire, C.1    Cantineau, R.2    Guillaume, M.3    Plenevaux, A.4    Christiaens, L.5
  • 95
    • 33846889762 scopus 로고    scopus 로고
    • 18F]MPPF as a tool for the in vivo imaging of 5-HT1A receptors in animal and human brain
    • 18F]MPPF as a tool for the in vivo imaging of 5-HT1A receptors in animal and human brain. Neuropharmacol 2007, 52:695-707.
    • (2007) Neuropharmacol , vol.52 , pp. 695-707
    • Aznavour, N.1    Zimmer, L.2
  • 99
    • 0642310756 scopus 로고    scopus 로고
    • 18F-CPFPX, a novel adenosine A1 receptor ligand: in vitro autoradiography and high-resolution small animal PET
    • 18F-CPFPX, a novel adenosine A1 receptor ligand: in vitro autoradiography and high-resolution small animal PET. J Nucl Med 2003, 44:1682-1689.
    • (2003) J Nucl Med , vol.44 , pp. 1682-1689
    • Bauer, A.1    Holschbach, M.H.2    Cremer, M.3    Weber, S.4    Boy, C.5    Shah, N.J.6
  • 100
    • 0035893245 scopus 로고    scopus 로고
    • Binding characteristics of radiofluorinated 6-dialkylamino-2-naphthylethylidene derivatives as positron emission tomography imaging probes for beta-amyloid plaques in Alzheimer's disease
    • Agdeppa E.D., Kepe V., Liu J., Flores-Torres S., Satyamurthy N., Petric A., et al. Binding characteristics of radiofluorinated 6-dialkylamino-2-naphthylethylidene derivatives as positron emission tomography imaging probes for beta-amyloid plaques in Alzheimer's disease. J Neurosci 2001, 21:RC189.
    • (2001) J Neurosci , vol.21
    • Agdeppa, E.D.1    Kepe, V.2    Liu, J.3    Flores-Torres, S.4    Satyamurthy, N.5    Petric, A.6
  • 102
    • 77956998284 scopus 로고    scopus 로고
    • Molecular Imaging and Contrast Agent Database (MICAD) [database online]. Bethesda (MD): National Library of Medicine (US). [accessed on 23rd April]
    • Molecular Imaging and Contrast Agent Database (MICAD) [database online]. Bethesda (MD): National Library of Medicine (US). [accessed on 23rd April 2010]. http://micad.nih.gov.
    • (2010)
  • 104
    • 68249144167 scopus 로고    scopus 로고
    • Radiopharmaceuticals, drug development and pharmaceuticals regulations in Europe
    • Salvadori P.A. Radiopharmaceuticals, drug development and pharmaceuticals regulations in Europe. Current Radiopharmaceuticals 2008, 1:7-11.
    • (2008) Current Radiopharmaceuticals , vol.1 , pp. 7-11
    • Salvadori, P.A.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.