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Journal of Biological Inorganic Chemistry

Volumn 15, Issue 4, 2010, Pages 591-599

Design, synthesis, and evaluation of cyclofenil derivatives for potential SPECT imaging agents

(6) Zhu, Hua a,b Huang, Liliang a,b Zhang, Yuanqing a,b Xu, Xiaoping a,b Sun, Yanhong a Shen, Yu Mei a,c

a SHANGHAI INSTITUTE OF APPLIED PHYSICS (China)

b INSTITUTE OF GEOLOGY AND GEOPHYSICS (China)

c Chinese National Human Genome Center at Shanghai (China)

Author keywords

Cyclofenil; Estrogen receptor; Nonsteroidal; Radiolabeling; Tricarbonyl rhenium

Indexed keywords

CONTRAST MEDIUM; ESTROGEN RECEPTOR; TRICARBONYL RHENIUM COMPLEX; TRICARBONYL TECHNETIUM CYCLOFENIL COMPLEX; UNCLASSIFIED DRUG;

ALKYLATION; ARTICLE; BINDING AFFINITY; CHEMICAL ANALYSIS; CHEMICAL BINDING; DRUG DESIGN; DRUG PURITY; DRUG STABILITY; DRUG SYNTHESIS; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; PRIORITY JOURNAL; RADIOCHEMISTRY; SINGLE PHOTON EMISSION COMPUTER TOMOGRAPHY; SYNTHESIS;

BREAST NEOPLASMS; CYCLOFENIL; DRUG DESIGN; DRUG STABILITY; HUMANS; LIGANDS; OCTANOLS; ORGANOTECHNETIUM COMPOUNDS; RECEPTORS, ESTROGEN; RHENIUM; TOMOGRAPHY, EMISSION-COMPUTED, SINGLE-PHOTON; WATER;

EID: 77953356765 PISSN: 09498257 EISSN: None Source Type: Journal
DOI: 10.1007/s00775-010-0627-0 Document Type: Article

Times cited : (16)

References (50)

1
- 0033096995
- Gao H, Katzenellenbogen JA, Garg R, Hansch C (1999) Chem Rev 99:723-744
- (1999) Chem Rev , vol.99 , pp. 723-744
- Gao, H.¹ Katzenellenbogen, J.A.² Garg, R.³ Hansch, C.⁴

2
- 0038111022
- Zhang W, Andersson S, Cheng G, Simpson ER, Warner M, Gustafsson JA (2003) FEBS Lett 546:17-24
- (2003) FEBS Lett , vol.546 , pp. 17-24
- Zhang, W.¹ Andersson, S.² Cheng, G.³ Simpson, E.R.⁴ Warner, M.⁵ Gustafsson, J.A.⁶

3
- 0030579801
- Kuiper G, Enmark E, Pelto-Huikko M, Nilsson S, Gustafsson JA (1996) Proc Natl Acad Sci USA 93:5925-5930
- (1996) Proc Natl Acad Sci USA , vol.93 , pp. 5925-5930
- Kuiper, G.¹ Enmark, E.² Pelto-Huikko, M.³ Nilsson, S.⁴ Gustafsson, J.A.⁵

4
- 0035866760
- Roger P, Sahla ME, Makela S, Gustafsson JA, Baldet P, Rochefort H (2000) Cancer Res 61:2537-2541
- (2000) Cancer Res , vol.61 , pp. 2537-2541
- Roger, P.¹ Sahla, M.E.² Makela, S.³ Gustafsson, J.A.⁴ Baldet, P.⁵ Rochefort, H.⁶

5
- 18344363175
- Palmieri C, Cheng GJ, Saji S, Zelada-Hedman WarriA, Weihua Z, Noorden SV, Wahlstrom T, Coombes RC, Warner M, Gustafsson JA (2002) Endocr Relat Cancer 9:1-13
- (2002) Endocr Relat Cancer , vol.9 , pp. 1-13
- Palmieri, C.¹ Cheng, G.J.² Saji, S.³ WarriA, Z.-H.⁴ Weihua, Z.⁵ Noorden, S.V.⁶ Wahlstrom, T.⁷ Coombes, R.C.⁸ Warner, M.⁹ Gustafsson, J.A.¹⁰

6
- 77953356031
- Speirs V, Carder PJ, Lansdown MR (2002) Br J Cancer 87:688689
- (2002) Br J Cancer , vol.87 , pp. 688689
- Speirs, V.¹ Carder, P.J.² Lansdown, M.R.³

7
- 0036161026
- Omoto Y, Kobayashi S, Inoue S, Ogawa S, Toyama T, Yamashita H, Muramatsu M, Gustafsson JA, Iwase H (2002) Eur J Cancer 38:380-386
- (2002) Eur J Cancer , vol.38 , pp. 380-386
- Omoto, Y.¹ Kobayashi, S.² Inoue, S.³ Ogawa, S.⁴ Toyama, T.⁵ Yamashita, H.⁶ Muramatsu, M.⁷ Gustafsson, J.A.⁸ Iwase, H.⁹

8
- 0019378715
- Katzenellenbogen JA, Senderoff SG, McElvany KD, Brien HA Jr, Welch MJ (1981) J Nucl Med 22:42-47
- (1981) J Nucl Med , vol.22 , pp. 42-47
- Katzenellenbogen, J.A.¹ Senderoff, S.G.² McElvany, K.D.³ Brien Jr., H.A.⁴ Welch, M.J.⁵

9
- 0020001918
- McElvany KD, Katzenellenbogen JA, Shafer KE, Siegel BA, Senderoff SG, Welch MJ (1982) J Nucl Med 23:425-430
- (1982) J Nucl Med , vol.23 , pp. 425-430
- McElvany, K.D.¹ Katzenellenbogen, J.A.² Shafer, K.E.³ Siegel, B.A.⁴ Senderoff, S.G.⁵ Welch, M.J.⁶

10
- 0031961153
- Rijks LJ, Bos JC, Doremalenl PA, Boer GJ, Bruin K, Doornbos T, Vekemans JA, Posthumus MA, Janssen AG (1998) Royen Nucl Med Biol 25:411-421
- (1998) Royen Nucl Med Biol , vol.25 , pp. 411-421
- Rijks, L.J.¹ Bos, J.C.² Doremalenl, P.A.³ Boer, G.J.⁴ Bruin, K.⁵ Doornbos, T.⁶ Vekemans, J.A.⁷ Posthumus, Ma.⁸ Janssen, A.G.⁹

11
- 0025251173
- Pomper MG, Brocklin H, Thieme AM, Thomas KD, Kiesewetter KE, Carlson KE, Mathias CJ, Welch MJ, Katzenellenbogen JA (1990) J Med Chem 33:3143-3155
- (1990) J Med Chem , vol.33 , pp. 3143-3155
- Pomper, M.G.¹ Brocklin, H.² Thieme, A.M.³ Thomas, K.D.⁴ Kiesewetter, K.E.⁵ Carlson, K.E.⁶ Mathias, C.J.⁷ Welch, M.J.⁸ Katzenellenbogen, J.A.⁹

12
- 0036026463
- Seimbille Y, Brocklin H, Lier JE (2002) J Chem Soc Perkin Trans 20:2275-2281
- (2002) J Chem Soc Perkin Trans , vol.20 , pp. 2275-2281
- Seimbille, Y.¹ Brocklin, H.² Lier, J.E.³

13
- 0027336501
- VanBrocklin HF, Carlson KE, Katzenellenbogen JA, Welch MJ (1993) J Med Chem 36:1619-1629
- (1993) J Med Chem , vol.36 , pp. 1619-1629
- VanBrocklin, H.F.¹ Carlson, K.E.² Katzenellenbogen, J.A.³ Welch, M.J.⁴

14
- 0242266521
- Luyt G, Bigott HM, Welch MJ, Katzenellenbogen JA (2003) Bioorg Med Chem 11:4977-4989
- (2003) Bioorg Med Chem , vol.11 , pp. 4977-4989
- Luyt, G.¹ Bigott, H.M.² Welch, M.J.³ Katzenellenbogen, J.A.⁴

15
- 0029145533
- Top S, Hafa HE, Vessieres A, Quivy J, Vaissermann J, Hughes DW, McGlinchey MJ, Mornon JP, Thoreau E, Jaouen G (1995) J Am Chem Soc 117:8372-8380
- (1995) J Am Chem Soc , vol.117 , pp. 8372-8380
- Top, S.¹ Hafa, H.E.² Vessieres, A.³ Quivy, J.⁴ Vaissermann, J.⁵ Hughes, D.W.⁶ McGlinchey, M.J.⁷ Mornon, J.P.⁸ Thoreau, E.⁹ Jaouen, G.¹⁰

16
- 0345440144
- Skaddan MB, Wust FR, Katzenellenbogen JA (1999) J Org Chem 64:8108-8121
- (1999) J Org Chem , vol.64 , pp. 8108-8121
- Skaddan, M.B.¹ Wust, F.R.² Katzenellenbogen, J.A.³

17
- 0041336761
- Arterburn JB, Corona C, Rao KV, Carlson KE, Katzenellenbogen JA (2003) J Org Chem 68:7063-7070
- (2003) J Org Chem , vol.68 , pp. 7063-7070
- Arterburn, J.B.¹ Corona, C.² Rao, K.V.³ Carlson, K.E.⁴ Katzenellenbogen, J.A.⁵

18
- 0028013557
- Bergmann KE, Landvatter SW, Rocque PG, Carlson KE, Welch MJ, Katzenellenbogen JA (1994) Nucl Med Biol 21:25-39
- (1994) Nucl Med Biol , vol.21 , pp. 25-39
- Bergmann, K.E.¹ Landvatter, S.W.² Rocque, P.G.³ Carlson, K.E.⁴ Welch, M.J.⁵ Katzenellenbogen, J.A.⁶

19
- 0036973248
- Lashley MR, Niedzinski EJ, Rogers JM, Denison MS, Nantz MH (2002) Bioorg Med Chem 10:4075-4082
- (2002) Bioorg Med Chem , vol.10 , pp. 4075-4082
- Lashley, M.R.¹ Niedzinski, E.J.² Rogers, J.M.³ Denison, M.S.⁴ Nantz, M.H.⁵

20
- 0041620649
- Lee KC, Moon BS, Lee JH, Chung KH, Katzenellenbogen JA, Chi DY (2003) Bioorg Med Chem 11:3649-3658
- (2003) Bioorg Med Chem , vol.11 , pp. 3649-3658
- Lee, K.C.¹ Moon, B.S.² Lee, J.H.³ Chung, K.H.⁴ Katzenellenbogen, J.A.⁵ Chi, D.Y.⁶

21
- 77953360920
- Yang DJ, Li C, Kuang LR, Price JE, Buzdar AU, Tansey W, Cheriff A, Gretzer M, Kim EE, Wallace S (1994) Life Sci 55:5367
- (1994) Life Sci , vol.55 , pp. 5367
- Yang, D.J.¹ Li, C.² Kuang, L.R.³ Price, J.E.⁴ Buzdar, A.U.⁵ Tansey, W.⁶ Cheriff, A.⁷ Gretzer, M.⁸ Kim, E.E.⁹ Wallace, S.¹⁰

22
- 0036375102
- McDonnell DP, Connor CE, Wijayaratne A, Chang CY, Norris JD (2002) Recent Prog Horm Res 27:295-316
- (2002) Recent Prog Horm Res , vol.27 , pp. 295-316
- McDonnell, D.P.¹ Connor, C.E.² Wijayaratne, A.³ Chang, C.Y.⁴ Norris, J.D.⁵

23
- 0033368173
- Silfen SL, Ciaccia AV, Bryant HU (1999) Climacteric 2:268-283
- (1999) Climacteric , vol.2 , pp. 268-283
- Silfen, S.L.¹ Ciaccia, A.V.² Bryant, H.U.³

24
- 33646123780
- Seo JW, Comminos JS, Chi DY, Kim DW, Carlson KE, Katzenellenbogen JA (2006) J Med Chem 49:2496-2511
- (2006) J Med Chem , vol.49 , pp. 2496-2511
- Seo, J.W.¹ Comminos, J.S.² Chi, D.Y.³ Kim, D.W.⁴ Carlson, K.E.⁵ Katzenellenbogen, J.A.⁶

25
- 34248149419
- Seo JW, Chi DY, Dence CS, Welch MJ (2007) Nucl Med Biol 34:383-390
- (2007) Nucl Med Biol , vol.34 , pp. 383-390
- Seo, J.W.¹ Chi, D.Y.² Dence, C.S.³ Welch, M.J.⁴

26
- 39649117151
- Gao MZ, Wang M, Mock BH, Miller KD, Sledge GW, Hutchins GD, Zheng QH (2008) Appl Radia Isotopes 66:523-529
- (2008) Appl Radia Isotopes , vol.66 , pp. 523-529
- Gao, M.Z.¹ Wang, M.² Mock, B.H.³ Miller, K.D.⁴ Sledge, G.W.⁵ Hutchins, G.D.⁶ Zheng, Q.H.⁷

27
- 33748216792
- Schwochau K (1994) Angew Chem Int Ed Engl 33:2258-2267
- (1994) Angew Chem Int Ed Engl , vol.33 , pp. 2258-2267
- Schwochau, K.¹

28
- 0033198735
- Pike AC, Brzozowski AM, Hubbard RE, Bonn T, Thorsell AG, Engstrom O, Ljunggren J, Gustafsson J, Carlquist M (1999) EMBO J 18:4608-4618
- (1999) EMBO J , vol.18 , pp. 4608-4618
- Pike, A.C.¹ Brzozowski, A.M.² Hubbard, R.E.³ Bonn, T.⁴ Thorsell, A.G.⁵ Engstrom, O.⁶ Ljunggren, J.⁷ Gustafsson, J.⁸ Carlquist, M.⁹

29
- 0030969731
- Jacques G, Maryse F, Tiiu O, Christophe DJ, Michel P (1997) J Med Chem 40:1104-1111
- (1997) J Med Chem , vol.40 , pp. 1104-1111
- Jacques, G.¹ Maryse, F.² Tiiu, O.³ Christophe, D.J.⁴ Michel, P.⁵

30
- 0345358448
- Muthyala RS, Carlson KE, Katzenellenbogen JA (2003) Bioorg Med Chem Lett 13:4485-4488
- (2003) Bioorg Med Chem Lett , vol.13 , pp. 4485-4488
- Muthyala, R.S.¹ Carlson, K.E.² Katzenellenbogen, J.A.³

31
- 33751005875
- Kim SH, Katzenellenbogen JA (2006) Angew Chem Int Ed 45:7243-7248
- (2006) Angew Chem Int Ed , vol.45 , pp. 7243-7248
- Kim, S.H.¹ Katzenellenbogen, J.A.²

32
- 58849105986
- Bartholoma M, Valliant J, Maresca KP, Babich J, Zubieta J (2009) Chem Commun 493-512
- (2009) Chem Commun , pp. 493-512
- Bartholoma, M.¹ Valliant, J.² Maresca, Kp.³ Babich, J.⁴ Zubieta, J.⁵

33
- 67650602179
- Jennings LE, Long NJ (2009) Chem Commun 3511-3524
- (2009) Chem Commun , pp. 3511-3524
- Jennings, L.E.¹ Long, N.J.²

34
- 70349136310
- Maresca KP, Hiller SM, Femia FJ, Zimmerman CN, Levadala MK, Banerjee SR, Hicks J, Sundararajan C, Valliant J, Zubieta J, Eckelman WC, Joyal JL, Babich JW (2009) Bioconjug Chem 20:1625-1633
- (2009) Bioconjug Chem , vol.20 , pp. 1625-1633
- Maresca, Kp.¹ Hiller, S.M.² Femia, F.J.³ Zimmerman, C.N.⁴ Levadala, M.K.⁵ Banerjee, S.R.⁶ Hicks, J.⁷ Sundararajan, C.⁸ Valliant, J.⁹ Zubieta, J.¹⁰ Eckelman, W.C.¹¹ Joyal, J.L.¹² Babich, J.W.¹³

35
- 0034836075
- Alberto R, Ortner K, Wheatley N, Schibli R, Schubiger PA (2001) J Am Chem Soc 123:3135-3136
- (2001) J Am Chem Soc , vol.123 , pp. 3135-3136
- Alberto, R.¹ Ortner, K.² Wheatley, N.³ Schibli, R.⁴ Schubiger, P.A.⁵

36
- 0001454913
- Alberto R, Schibli R, EgIi A, Schubiger PA, Herrmann WA, Artus G, Abram U, Kaden TA (1995) J Organomet Chem 493:119-127
- (1995) J Organomet Chem , vol.493 , pp. 119-127
- Alberto, R.¹ Schibli, R.² EgIi, A.³ Schubiger, P.A.⁴ Herrmann, W.A.⁵ Artus, G.⁶ Abram, U.⁷ Kaden, T.A.⁸

37
- 0015902629
- Katzenellenbogen JA, Johnson HJ, Myers HN (1973) Biochemistry 12:4085-4092
- (1973) Biochemistry , vol.12 , pp. 4085-4092
- Katzenellenbogen, J.A.¹ Johnson, H.J.² Myers, H.N.³

38
- 0030734795
- Carlson KE, Choi I, Gee A, Katzenellenbogen BS, Katzenellenbogen JA (1997) Biochemistry 36:14897-14905
- (1997) Biochemistry , vol.36 , pp. 14897-14905
- Carlson, K.E.¹ Choi, I.² Gee, A.³ Katzenellenbogen, B.S.⁴ Katzenellenbogen, J.A.⁵

39
- 0035996627
- Seimbille Y, Rousseau J, Benard F, Morin C, Ali H, Avvakumov G, Hammond GL, Lier JE (2002) Steroids 67:765-775
- (2002) Steroids , vol.67 , pp. 765-775
- Seimbille, Y.¹ Rousseau, J.² Benard, F.³ Morin, C.⁴ Ali, H.⁵ Avvakumov, G.⁶ Hammond, G.L.⁷ Lier, J.E.⁸

40
- 0032511351
- Alberto R, Schibli R, EgIi A, Schubiger PA (1998) J Am Chem Soc 120:7987-7988
- (1998) J Am Chem Soc , vol.120 , pp. 7987-7988
- Alberto, R.¹ Schibli, R.² EgIi, A.³ Schubiger, P.A.⁴

41
- 33646933762
- Muller C, Schubiger PA, Schibli R (2006) Bioconjug Chem 17:797-806
- (2006) Bioconjug Chem , vol.17 , pp. 797-806
- Muller, C.¹ Schubiger, P.A.² Schibli, R.³

42
- 77953362256
- Muller C, Schubiger PA, Schibli R (2007) Nucl Med Bio 34:595601
- (2007) Nucl Med Bio , vol.34 , pp. 595601
- Muller, C.¹ Schubiger, P.A.² Schibli, R.³

43
- 33747472945
- Pillarsetty N, Cai S, Ageyeva L, Finn RD, Blasberg RG (2006) J Med Chem 49:5377-5381
- (2006) J Med Chem , vol.49 , pp. 5377-5381
- Pillarsetty, N.¹ Cai, S.² Ageyeva, L.³ Finn, R.D.⁴ Blasberg, R.G.⁵

44
- 16644397119
- Alberto AR, Abram U, Hegetschweiler K, Gramlich V, Schubiger PA (1994) J Chem Soc Dalton Trans 19:2815-2820
- (1994) J Chem Soc Dalton Trans , vol.19 , pp. 2815-2820
- Alberto, A.R.¹ Abram, U.² Hegetschweiler, K.³ Gramlich, V.⁴ Schubiger, P.A.⁵

45
- 0031059270
- Anstead GM, Carlson KE, Katzenellenbogen JA (1997) Steroids 62:268-303
- (1997) Steroids , vol.62 , pp. 268-303
- Anstead, G.M.¹ Carlson, K.E.² Katzenellenbogen, J.A.³

46
- 0345567604
- Grese TA, Sluka JP, Bryant HU, Cullinan GJ, Glasebrook AL, Jones CD, Matsumoto K, Palkowitz AD, Sato M, Termine JD, Winter MA, Yang NN, Dodge JA (1997) Proc Natl Acad Sci USA 94:14105-14110
- (1997) Proc Natl Acad Sci USA , vol.94 , pp. 14105-14110
- Grese, T.A.¹ Sluka, J.P.² Bryant, H.U.³ Cullinan, G.J.⁴ Glasebrook, A.L.⁵ Jones, C.D.⁶ Matsumoto, K.⁷ Palkowitz, A.D.⁸ Sato, M.⁹ Termine, J.D.¹⁰ Winter, Ma.¹¹ Yang, N.N.¹² Dodge, J.A.¹³

47
- 0002089528
- Abel EW, Ouell KG, Osborne AG, Pain HM, Sik V, Hursthouse MB, Malik KMA (1994) J Chem Soc Dalton Trans 3441-3449
- (1994) J Chem Soc Dalton Trans , pp. 3441-3449
- Abel, E.W.¹ Ouell, K.G.² Osborne, A.G.³ Pain, H.M.⁴ Sik, V.⁵ Hursthouse, M.B.⁶ Malik, K.M.A.⁷

48
- 77953360784
- Gamelin DR, George MW, Glyn P, Grevek FW, Schaffner K, Turner JJ (1995) Inorg Chem 33:3250-4246
- (1995) Inorg Chem , vol.33 , pp. 3250-4246
- Gamelin, D.R.¹ George, M.W.² Glyn, P.³ Grevek, F.W.⁴ Schaffner, K.⁵ Turner, J.J.⁶

49
- 0025785380
- Levesque C, Merand Y, Dufour JM, Labrie C, Labrie F (1991) J Med Chem 34:1624-1630
- (1991) J Med Chem , vol.34 , pp. 1624-1630
- Levesque, C.¹ Merand, Y.² Dufour, J.M.³ Labrie, C.⁴ Labrie, F.⁵

50
- 44849115355
- Nayak TK, Hathaway HJ, Ramesh C, Arterburn JB, Dai DH, Sklar LA, Norenberg JP, Prossnitz ER (2008) J Nucl Med 49:978-986
- (2008) J Nucl Med , vol.49 , pp. 978-986
- Nayak, T.K.¹ Hathaway, H.J.² Ramesh, C.³ Arterburn, J.B.⁴ Dai, D.H.⁵ Sklar, L.A.⁶ Norenberg, J.P.⁷ Prossnitz, E.R.⁸

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