Molecular determinants of tissue selectivity in estrogen receptor modulators

Proceedings of the National Academy of Sciences of the United States of America

Volumn 94, Issue 25, 1997, Pages 14105-14110

  Grese, Timothy A ^a   Sluka, James P ^a   Bryant, Henry U ^a   Cullinan, George J ^a   Glasebrook, Andrew L ^a   Jones, Charles D ^a   Matsumoto, Ken ^a   Palkowitz, Alan D ^a   Sato, Masahiko ^a   Termine, John D ^a   Winter, Mark A ^a   Yang, Na N ^a   Dodge, Jeffrey A ^a  

^a ELI LILLY AND COMPANY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ESTRADIOL; ESTROGEN RECEPTOR; RALOXIFENE; STILBENE; TAMOXIFEN;

ARTICLE; BINDING AFFINITY; GENETIC TRANSCRIPTION; HYPOTHESIS; LIGAND BINDING; PRIORITY JOURNAL; PROTEIN CONFORMATION; RECEPTOR BINDING; STRUCTURE ACTIVITY RELATION; TISSUE SPECIFICITY; TRANSCRIPTION REGULATION;

ANIMALS; CELL LINE; ESTRADIOL CONGENERS; ESTROGEN ANTAGONISTS; FEMALE; LIGANDS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; PIPERIDINES; PROTEIN CONFORMATION; RALOXIFENE; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, ESTROGEN; STRUCTURE-ACTIVITY RELATIONSHIP; TAMOXIFEN; THERMODYNAMICS; TISSUE DISTRIBUTION; UTERUS;

EID: 0345567604     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.94.25.14105     Document Type: Article

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