Catalysis and inhibition of Mycobacterium tuberculosis methionine aminopeptidase

Journal of Medicinal Chemistry

Volumn 53, Issue 3, 2010, Pages 1329-1337

  Lu, Jing Ping ^a   Chai, Sergio C ^a   Ye, Qi Zhuang ^a  

^a INDIANA UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

APOENZYME; COBALT; FERROUS ION; MANGANESE; METAL ION; METHIONYL AMINOPEPTIDASE; NICKEL;

ARTICLE; CATALYSIS; CELL GROWTH; CRYSTAL STRUCTURE; DRUG INHIBITION; DRUG STRUCTURE; ESCHERICHIA COLI; GENE; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; PLASMID; X RAY CRYSTALLOGRAPHY;

AMINOPEPTIDASES; APOENZYMES; BINDING SITES; CATALYSIS; CATIONS, DIVALENT; CRYSTALLOGRAPHY, X-RAY; ENZYME INHIBITORS; ESCHERICHIA COLI; FERRIC COMPOUNDS; GENETIC COMPLEMENTATION TEST; MODELS, MOLECULAR; MOLECULAR STRUCTURE; MYCOBACTERIUM TUBERCULOSIS; PROTEIN BINDING; PROTEIN CONFORMATION; RECOMBINANT PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP; SUBSTRATE SPECIFICITY;

EID: 77249109358     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm901624n     Document Type: Article

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