-
1
-
-
70350191329
-
-
For reviews, see: a) A. Kamal, K. L. Reddy, V. Devaiah, N. Shankaraiah, M. V. Rao, Mini-Rev. Med. Chem. 2006, 6, 7189;
-
(2006)
Mini-Rev. Med. Chem.
, vol.6
, pp. 7189
-
-
Kamal, A.1
Reddy, K.L.2
Devaiah, V.3
Shankaraiah, N.4
Rao, M.V.5
-
2
-
-
0030053138
-
-
b) R. R. Wexler, W J. Greenlee, J D. Irvin, M. R. Goldberg, K. Prendergast, R. P. Smith, P. B. M. W M. Timmermans, J. Med, Chem. 1996, 39, 625-656;
-
(1996)
J. Med, Chem.
, vol.39
, pp. 625-656
-
-
Wexler, R.R.1
Greenlee, W.J.2
Irvin, J.D.3
Goldberg, M.R.4
Prendergast, K.5
Smith, R.P.6
Timmermans, P.B.M.W.M.7
-
3
-
-
0037366605
-
-
c) D. A. Horton, G. T. Bourne, M. L. Smythe, Chem. Rev. 2003, 103, 893-930.
-
(2003)
Chem. Rev.
, vol.103
, pp. 893-930
-
-
Horton, D.A.1
Bourne, G.T.2
Smythe, M.L.3
-
4
-
-
33746741042
-
-
a) Y-F. Li, G.-F. Wang, R-L. He, W-G. Huang, F-H. Zhu, HY. Gao, W Tang, Y. Luo, C-L. Feng, L.-P. Shi, Y-D. Ren, W Lu, J.-P. Zuo, J. Med, Chem. 2006, 49, 4790-4794;
-
(2006)
J. Med, Chem.
, vol.49
, pp. 4790-4794
-
-
Li, Y.-F.1
Wang, G.-F.2
He, R.-L.3
Huang, W.-G.4
Zhu, F.-H.5
Gao, H.Y.6
Tang, W.7
Luo, Y.8
Feng, C.-L.9
Shi, L.-P.10
Ren, Y.-D.11
Lu, W.12
Zuo, J.-P.13
-
5
-
-
11144220783
-
-
b) P. L. Beaulieu, Y. Bousquet, I Gauthier, I Gillard, M. Marquis, G. McKercher, C. Pellerin, S. Valois, G. Kukolj, J. Med. Chem. 2004, 47, 6884-6892;
-
(2004)
J. Med. Chem.
, vol.47
, pp. 6884-6892
-
-
Beaulieu, P.L.1
Bousquet, Y.2
Gauthier, I.3
Gillard, I.4
Marquis, M.5
McKercher, G.6
Pellerin, C.7
Valois, S.8
Kukolj, G.9
-
6
-
-
33746700189
-
-
c) S. Hiroshima, T. Suzuki, T. Ishida, S. Noji, S. Yata, I. Ando, M. Komatsu, S. Ikeda, H. Hashimoto, J. Med. Chem. 2006, 49, 4721-4736.
-
(2006)
J. Med. Chem.
, vol.49
, pp. 4721-4736
-
-
Hiroshima, S.1
Suzuki, T.2
Ishida, T.3
Noji, S.4
Yata, S.5
Ando, I.6
Komatsu, M.7
Ikeda, S.8
Hashimoto, H.9
-
7
-
-
33750531634
-
-
M. Sabat, J. C. Vanrens, M J Laufersweiler, T. A. Brugel, J. Maier, A. Golebiowski, B. De, V. Easwaran, L. C. Hsieh, R. L. Walter, M. J Mekel, A. Evdokimov, M. J. Janusz, Bioorg. Med.Chem. Lett. 2006, 16, 5973-5977.
-
(2006)
Bioorg. Med. Chem. Lett.
, vol.16
, pp. 5973-5977
-
-
Sabat, M.1
Vanrens, J.C.2
Laufersweiler, M.J.3
Brugel, T.A.4
Maier, J.5
Golebiowski, A.6
De, B.7
Easwaran, V.8
Hsieh, L.C.9
Walter, R.L.10
Mekel, M.J.11
Evdokimov, A.12
Janusz, M.J.13
-
8
-
-
0037171819
-
-
N. H. Hauel, H. Nar, H. Priepke, U. Ries, J. Stassen, W Wienen, J. Med. Chem. 2002, 45, 1757-1766.
-
(2002)
J. Med. Chem.
, vol.45
, pp. 1757-1766
-
-
Hauel, N.H.1
Nar, H.2
Priepke, H.3
Ries, U.4
Stassen, J.5
Wienen, W.6
-
9
-
-
0034005413
-
-
H. Nakano, T. Inoue, N. Kawasaki, H. Miyataka, H. Matsumoto, T. Taguchi, N. Inagaki, H. Nagai, T. Satoh, Bioorg. Med. Chem. 2000, 8, 373-380.
-
(2000)
Bioorg. Med. Chem.
, vol.8
, pp. 373-380
-
-
Nakano, H.1
Inoue, T.2
Kawasaki, N.3
Miyataka, H.4
Matsumoto, H.5
Taguchi, T.6
Inagaki, N.7
Nagai, H.8
Satoh, T.9
-
10
-
-
4143112939
-
Benzimidazoles and congeneric tricyclic compounds
-
(Eds.: A. Weissberger, E. C. Taylor), Wiley-VCH, New York
-
a) P. N. Preston, "Benzimidazoles and Congeneric Tricyclic Compounds", in 'The Chemistry of Heterocyclic Compounds (Eds.: A. Weissberger, E. C. Taylor), Wiley-VCH, New York, 1981, vol.40, pp. 6-60;
-
(1981)
The Chemistry of Heterocyclic Compounds
, vol.40
, pp. 6-60
-
-
Preston, P.N.1
-
11
-
-
84943408843
-
Imidazoles and their benzo derivatives
-
(Eds.: A. R. Katritzky, C. W Rees), Pergamon, Oxford
-
b) M. R. Grimmett, "Imidazoles and their Benzo Derivatives", in Comprehensive Heterocyclic Chemistry (Eds.: A. R. Katritzky, C. W Rees), Pergamon, Oxford, 1984, vol.5, pp. 457-487.
-
(1984)
Comprehensive Heterocyclic Chemistry
, vol.5
, pp. 457-487
-
-
Grimmett, M.R.1
-
12
-
-
64249105656
-
-
For catalytic syntheses of benzimidazoles and related cyclizations, see: a) S. Murru, B. K. Patel, J Le Bras, I Muzart, J. Org. Chem. 2009, 74, 2217-2220;
-
(2009)
J. Org. Chem.
, vol.74
, pp. 2217-2220
-
-
Murru, S.1
Patel, B.K.2
Le Bras, J.3
Muzart, I.4
-
13
-
-
49649093371
-
-
b) Z. Li, H. Sun, H. Jiang, H. Liu, Org. Lett. 2008, 10, 3263-3266;
-
(2008)
Org. Lett.
, vol.10
, pp. 3263-3266
-
-
Li, Z.1
Sun, H.2
Jiang, H.3
Liu, H.4
-
15
-
-
41949118427
-
-
Angew. Chem. Int. Ed. 2008, 47, 1932-1934;
-
(2008)
Angew. Chem. Int. Ed.
, vol.47
, pp. 1932-1934
-
-
-
16
-
-
47049109018
-
-
d) I Alen, K. Robeyns, W M. De Borggraeve, L. Van Meervelt, F. Compernolle, Tetrahedron 2008, 64, 8128-8133;
-
(2008)
Tetrahedron
, vol.64
, pp. 8128-8133
-
-
Alen, I.1
Robeyns, K.2
De Borggraeve, W.M.3
Van Meervelt, L.4
Compernolle, F.5
-
17
-
-
53549120107
-
-
e) B. Zou, Q. Yuan, D. Ma, Angew. Chem. 2007, 119, 2652-2655;
-
(2007)
Angew. Chem.
, vol.119
, pp. 2652-2655
-
-
Zou, B.1
Yuan, Q.2
Ma, D.3
-
18
-
-
34250839461
-
-
Angew. Chem. Int. Ed. 2007, 46, 2598-2601;
-
(2007)
Angew. Chem. Int. Ed.
, vol.46
, pp. 2598-2601
-
-
-
19
-
-
32144431909
-
-
f) C. Venkatesh, G. S. M. Sundram, H. IIa, H. Junjappa, J. Org. Chem. 2006, 71, 1280-1283;
-
(2006)
J. Org. Chem.
, vol.71
, pp. 1280-1283
-
-
Venkatesh, C.1
Sundram, G.S.M.2
Iia, H.3
Junjappa, H.4
-
20
-
-
0345802836
-
-
g) K. G. Nazarenko, T. I. Shyrokaya, K. V. Shvidenko, A. A. Tolmachev, Synth. Commun. 2003, 33, 4303-4311;
-
(2003)
Synth. Commun.
, vol.33
, pp. 4303-4311
-
-
Nazarenko, K.G.1
Shyrokaya, T.I.2
Shvidenko, K.V.3
Tolmachev, A.A.4
-
24
-
-
35348854372
-
-
a) S. Fujiwara, Y. Asanuma, T Shin-ike, N. Kambe, J. Org. Chem. 72, 8087-8090;
-
J. Org. Chem.
, vol.72
, pp. 8087-8090
-
-
Fujiwara, S.1
Asanuma, Y.2
Shin-ike, T.3
Kambe, N.4
-
27
-
-
1642329837
-
-
T. Saegusa, Y. Ito, K. Kobayashi, K. Hirota, H. Yoshioka, Tetrahedron Lett. 1966, 7, 6121-6124.
-
(1966)
Tetrahedron Lett.
, vol.7
, pp. 6121-6124
-
-
Saegusa, T.1
Ito, Y.2
Kobayashi, K.3
Hirota, K.4
Yoshioka, H.5
-
28
-
-
4043076940
-
-
T. Saegusa, Y. Ito, K. Kobayashi, K. Hirota, H. Yoshioka, Bull. Chem. Soc, Jpn. 1969, 42, 3310-3313.
-
(1969)
Bull. Chem. Soc, Jpn.
, vol.42
, pp. 3310-3313
-
-
Saegusa, T.1
Ito, Y.2
Kobayashi, K.3
Hirota, K.4
Yoshioka, H.5
-
29
-
-
4143116053
-
-
For recent reviews on copper-catalyzed cross-coupling reactions, see: a) S. V Ley, A. W Thomas, Angew. Chem, 2003,115, 5558-5607;
-
(2003)
Angew. Chem
, vol.115
, pp. 5558-5607
-
-
Ley, S.V.1
Thomas, A.W.2
-
30
-
-
0345708168
-
-
Angew. Chem. Int. Ed. 2003, 42, 5400-5449;
-
(2003)
Angew. Chem. Int. Ed.
, vol.42
, pp. 5400-5449
-
-
-
34
-
-
37049089244
-
-
b) A. R. Katritzky, W H. Ramer, J. N. Lam, J. Chem. Soc, Perkin Trans. 1 1987, 775-780.
-
(1987)
J. Chem. Soc, Perkin Trans.
, vol.1
, pp. 775-780
-
-
Katritzky, A.R.1
Ramer, W.H.2
Lam, J.N.3
-
35
-
-
70350205344
-
-
Article ASAP
-
For relevant reviews on transition-metal-catalyzed C-C bond formation by C.....H bond cleavage, see: a) D. A. Colby, R. G. Bergman, I A. Ellman, Chem. Rev. 2009, Article ASAP;
-
(2009)
Chem. Rev.
-
-
Colby, D.A.1
Bergman, R.G.2
Ellman, I.A.3
-
36
-
-
51649122191
-
-
b) I C. Lewis, R. G. Bergman, J. A. Ellman, Acc. Chem. Res. 2008, 41, 1013-1025;
-
(2008)
Acc. Chem. Res.
, vol.41
, pp. 1013-1025
-
-
Lewis, I.C.1
Bergman, R.G.2
Ellman, J.A.3
-
38
-
-
33846918696
-
-
d) D. Alberico, M. E. Scott, M, Lautens, Chem. Rev. 2007,107, 174-238;
-
(2007)
Chem. Rev.
, vol.107
, pp. 174-238
-
-
Alberico, D.1
Scott, M.E.2
Lautens, M.3
-
39
-
-
34250655628
-
-
e) I. V. Seregin, V. Gevorgyan, Chem. Soc, Rev. 2001,36, 1173-1193.
-
(2001)
Chem. Soc, Rev.
, vol.36
, pp. 1173-1193
-
-
Seregin, I.V.1
Gevorgyan, V.2
-
43
-
-
0037419179
-
-
d) M. W Hooper, M. Utsunomiya, J. F. Hartwig, J. Org. Chem. 2003, 68, 2861-2873.
-
(2003)
J. Org. Chem.
, vol.68
, pp. 2861-2873
-
-
Hooper, M.W.1
Utsunomiya, M.2
Hartwig, J.F.3
-
44
-
-
0000344058
-
-
a) A. G. Mistry, K. Smith, M. R. Bye, Tetrahedron Lett. 1986, ' 27, 1051-1054;
-
(1986)
Tetrahedron Lett.
, vol.27
, pp. 1051-1054
-
-
Mistry, A.G.1
Smith, K.2
Bye, M.R.3
-
45
-
-
0001492946
-
-
b) I. Kawasaki, N. Taguchi, Y. Yoneda, M. Yamashita, S. Ohta, Heterocycles 1996, 43, 1375-1379.
-
(1996)
Heterocycles
, vol.43
, pp. 1375-1379
-
-
Kawasaki, I.1
Taguchi, N.2
Yoneda, Y.3
Yamashita, M.4
Ohta, S.5
-
47
-
-
0027969825
-
-
b) G. C. Hsu, W. P. Kosar, W D. Jones, Organometallics 1994, 13, 385 396.
-
(1994)
Organometallics
, vol.13
, Issue.385
, pp. 396
-
-
Hsu, G.C.1
Kosar, W.P.2
Jones, W.D.3
-
48
-
-
70350210244
-
-
The same benzimidazole 4n was also observed as a major product in the reaction of 1-Br with 2,4,6-trimethylaniline
-
The same benzimidazole 4n was also observed as a major product in the reaction of 1-Br with 2,4,6-trimethylaniline.
-
-
-
-
50
-
-
1242318559
-
-
Z.-G. Le, Z.-C. Chen, Y. Hu, Q.-G. Zheng, Synthesis 2004, 208-210.
-
(2004)
Synthesis
, pp. 208-210
-
-
Le, Z.-G.1
Chen, Z.-C.2
Hu, Y.3
Zheng, Q.-G.4
|