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European Journal of Organic Chemistry

Volumn , Issue 30, 2009, Pages 5215-5223

Synthesis of new trifluoromethylated hydroxyethylamine-based scaffolds

(5) Philippe, Christine a Milcent, Thierry a Ngoc, Tam Nguyen Thi a Crousse, Benoit a Bonnet Delpon, Daniéle a

a UNIVERSITÉ PARIS SUD (France)

Author keywords

Amino acids; Epoxides; Fluorine; Hydroxyethylamine; Peptidomimetics; Protease

Indexed keywords

EID: 70350159246 PISSN: 1434193X EISSN: 10990690 Source Type: Journal
DOI: 10.1002/ejoc.200900578 Document Type: Article

Times cited : (10)

References (48)

1
- 0034628448
- D. Leung, G. Abbenante, D. P. Fairlie, J. Med. Chem. 2000, 43, 305-341.
- (2000) J. Med. Chem. , vol.43 , pp. 305-341
- Leung, D.¹ Abbenante, G.² Fairlie, D.P.³

2
- 0035179667
- A. K. Ghosh, G. Bilcer, G. Schutz, Synthesis 2001, 15, 2203-2229.
- (2001) Synthesis , vol.15 , pp. 2203-2229
- Ghosh, A.K.¹ Bilcer, G.² Schutz, G.³

3
- 1542374135
- C. S. T. Oost, M. Brewer, M. Goodnough, W. Tepp, E. A. Johnson, D. H. Rich, Pept. Sci. 2003, 71, 602-619.
- (2003) Pept. Sci. , vol.71 , pp. 602-619
- Oost, C.S.T.¹ Brewer, M.² Goodnough, M.³ Tepp, W.⁴ Johnson, E.A.⁵ Rich, D.H.⁶

4
- 23644450055
- D. Muthas, D. Noteberg, Y. A. Sabnis, E. Hamelink, L. Vrang, B. Samuelsson, A. Karlen, A. Hallberg, Bioorg. Med. Chem. 2005, 13, 5371-5390.
- (2005) Bioorg. Med. Chem. , vol.13 , pp. 5371-5390
- Muthas, D.¹ Noteberg, D.² Sabnis, Y.A.³ Hamelink, E.⁴ Vrang, L.⁵ Samuelsson, B.⁶ Karlen, A.⁷ Hallberg, A.⁸

5
- 0037468420
- D. Noteberg, E. Hamelink, J. Hulten, M. Wahlgren, L. Vrang, B. Samuelsson, A. Hallberg, J. Med. Chem. 2003, 46, 734-746.
- (2003) J. Med. Chem. , vol.46 , pp. 734-746
- Noteberg, D.¹ Hamelink, E.² Hulten, J.³ Wahlgren, M.⁴ Vrang, L.⁵ Samuelsson, B.⁶ Hallberg, A.⁷

6
- 0033594354
- T. S. Haque, A. G. Skillman, C. E. Lee, H. Habashita, I. Y Gluzman, T. J. A. Ewing, D. E. Goldberg, I. D. Kuntz, J. A. Ellman, J. Med. Chem. 1999, 42, 1428-1440.
- (1999) J. Med. Chem. , vol.42 , pp. 1428-1440
- Haque, T.S.¹ Skillman, A.G.² Lee, C.E.³ Habashita, H.⁴ Gluzman, I.Y.⁵ Ewing, T.J.A.⁶ Goldberg, D.E.⁷ Kuntz, I.D.⁸ Ellman, J.A.⁹

7
- 0141787013
- D. Nöteberg, W. Schaal, E. Hamelink, L. Vrang, M. Lahred, J. Comb. Chem. 2003, 5, 456-464.
- (2003) J. Comb. Chem. , vol.5 , pp. 456-464
- Nöteberg, D.¹ Schaal, W.² Hamelink, E.³ Vrang, L.⁴ Lahred, M.⁵

8
- 33746147381
- R. M. McConnell, A. W. Green, C. J. Trana, M. S. McConnell, J. F. Lindley, K. Sayyar, W. E. Godwin, S. E. Hatfield, Med. Chem. 2006, 2, 27-38.
- (2006) Med. Chem. , vol.2 , pp. 27-38
- McConnell, R.M.¹ Green, A.W.² Trana, C.J.³ McConnell, M.S.⁴ Lindley, J.F.⁵ Sayyar, K.⁶ Godwin, W.E.⁷ Hatfield, S.E.⁸

9
- 44949137244
- N. Charrier, B. Clarke, L. Cutler, E. Demont, C. Dingwall, R. Dunsdon, P. East, J. Hawkins, C. Howes, I. Hussain, P. Jeffrey, G. Maile, R. Matico, J. Mosley, A. Naylor, A. Brien, S. Redshaw, P. Rowland, V. Soleil, K. J. Smith, S. Sweitzer, P. Theobald, D. Vesey, D. S. Walter, G. Wayne, J. Med. Chem. 2008, 51, 3313-3317.
- (2008) J. Med. Chem. , vol.51 , pp. 3313-3317
- Charrier, N.¹ Clarke, B.² Cutler, L.³ Demont, E.⁴ Dingwall, C.⁵ Dunsdon, R.⁶ East, P.⁷ Hawkins, J.⁸ Howes, C.⁹ Hussain, I.¹⁰ Jeffrey, P.¹¹ Maile, G.¹² Matico, R.¹³ Mosley, J.¹⁴ Naylor, A.¹⁵ Brien, A.¹⁶ Redshaw, S.¹⁷ Rowland, P.¹⁸ Soleil, V.¹⁹ Smith, K.J.²⁰ more..

10
- 33845648379
- J. N. Freskos, Y. M. Fobian, T E. Benson, M, J. Bienkowski, D. L. Brown, T. L. Emmons, R. Heintz, A. Laborde, J. J. McDonald, B. V. Mischke, J. M. Molyneaux, J. B. Moon, P. B. Mullins, D. B. Prince, D. J. Paddock, A. G. Tomasselli, G. Winterrowd, Bioorg. Med. Chem. Lett. 2007, 17, 73-77.
- (2007) Bioorg. Med. Chem. Lett. , vol.17 , pp. 73-77
- Freskos, J.N.¹ Fobian, Y.M.² Benson, T.E.³ Bienkowski, J.⁴ Brown, D.L.⁵ Emmons, T.L.⁶ Heintz, R.⁷ Laborde, A.⁸ McDonald, J.J.⁹ Mischke, B.V.¹⁰ Molyneaux, J.M.¹¹ Moon, J.B.¹² Mullins, P.B.¹³ Prince, D.B.¹⁴ Paddock, D.J.¹⁵ Tomasselli, A.G.¹⁶ Winterrowd, G.¹⁷

11
- 33845602981
- J. N. Freskos, Y. M. Fobian, T. E. Benson, J. B. Moon, M. J. Bienkowski, D. L. Brown, T. L. Emmons, R. Heintz, A. Laborde, J. J. McDonald, B. V. Mischke, J. M. Molyneaux, P. B. Mullins, D. B. Prince, D. J. Paddock, A. G. Tomasselli, G. Winterrowd, Bioorg. Med. Chem. Lett. 2007, 17, 78-81.
- (2007) Bioorg. Med. Chem. Lett. , vol.17 , pp. 78-81
- Freskos, J.N.¹ Fobian, Y.M.² Benson, T.E.³ Moon, J.B.⁴ Bienkowski, M.J.⁵ Brown, D.L.⁶ Emmons, T.L.⁷ Heintz, R.⁸ Laborde, A.⁹ McDonald, J.J.¹⁰ Mischke, B.V.¹¹ Molyneaux, J.M.¹² Mullins, P.B.¹³ Prince, D.B.¹⁴ Paddock, D.J.¹⁵ Tomasselli, A.G.¹⁶ Winterrowd, G.¹⁷

12
- 33847368052
- M. C Maillard, R. K. Horn, T. E. Benson, J. B. Moon, S. Mamo, M. Bienkowski, A. G. Tomasselli, D. D. Woods, D. B. Prince, D. J. Paddock, T. L. Emmons, J. A. Trucker, M. S. Dappen, L. Brogley, E. D. Thorsett, N. Jewett, S. Sinha, V. John, J. Med. Chem. 2007, 50, 776-781.
- (2007) J. Med. Chem. , vol.50 , pp. 776-781
- Maillard, M.C.¹ Horn, R.K.² Benson, T.E.³ Moon, J.B.⁴ Mamo, S.⁵ Bienkowski, M.⁶ Tomasselli, A.G.⁷ Woods, D.D.⁸ Prince, D.B.⁹ Paddock, D.J.¹⁰ Emmons, T.L.¹¹ Trucker, J.A.¹² Dappen, M.S.¹³ Brogley, L.¹⁴ Thorsett, E.D.¹⁵ Jewett, N.¹⁶ Sinha, S.¹⁷ John, V.¹⁸

13
- 42949127288
- M. Sani, A. Volonterio, M. Zanda, Chem Med Chem 2007, 2, 1693-1700.
- (2007) Chem MedChem , vol.2 , pp. 1693-1700
- Sani, M.¹ Volonterio, A.² Zanda, M.³

14
- 37849047198
- H. Meng, K. Kumar, J. Am. Chem. Soc. 2007, 129, 1561515622.
- (2007) J. Am. Chem. Soc. , vol.129 , pp. 1561515622
- Meng, H.¹ Kumar, K.²

15
- 0026775845
- I. Ojima, K. Kato, F. A. Jameison, J. Conway, Bioorg. Med. Chem. Lett. 1992, 2, 219-222.
- (1992) Bioorg. Med. Chem. Lett. , vol.2 , pp. 219-222
- Ojima, I.¹ Kato, K.² Jameison, F.A.³ Conway, J.⁴

16
- 0025997192
- I. Ojima, F. A. Jameison, Bioorg. Med. Chem. Lett. 1991, 7, 581-584.
- (1991) Bioorg. Med. Chem. Lett. , vol.7 , pp. 581-584
- Ojima, I.¹ Jameison, F.A.²

17
- 33746356860
- J. P. Bégué, D. Bonnet-Delpon, J. Fluorine Chem. 2006, 127, 992-1012.
- (2006) J. Fluorine Chem. , vol.127 , pp. 992-1012
- Bégué, J.P.¹ Bonnet-Delpon, D.²

18
- 33645454126
- C. Isanbor, D. O'Hagan, J. Fluorine. Chem. 2006, 127, 303-319.
- (2006) J. Fluorine. Chem. , vol.127 , pp. 303-319
- Isanbor, C.¹ O'Hagan, D.²

19
- 33746372978
- K. L. Kirk, J. Fluorine Chem. 2006, 127, 1013-1029.
- (2006) J. Fluorine Chem. , vol.127 , pp. 1013-1029
- Kirk, K.L.¹

20
- 84890169857
- John Wiley & Sons, Hoboken
- J. P. Bégué, D. Bonnet-Delpon, Bioorganic and Medicinal Chemistry of Fluorine, John Wiley & Sons, Hoboken, 2008.
- (2008) Bioorganic and Medicinal Chemistry of Fluorine
- Bégué, J.P.¹ Bonnet-Delpon, D.²

21
- 84891565619
- Wiley-VCH, Weinheim
- P. Kirsch, Modern Fluoroorganic Chemistry: Synthesis Reactivity, Applications, Wiley-VCH, Weinheim, 2004.
- (2004) Modern Fluoroorganic Chemistry: Synthesis Reactivity, Applications
- Kirsch, P.¹

22
- 11244267140
- M. Zanda, New J. Chem. 2004, 28, 1401-1411.
- (2004) New J. Chem. , vol.28 , pp. 1401-1411
- Zanda, M.¹

23
- 12344252565
- N. T. N. Tarn, G. Magueur, M. Ourevitch, B. Crousse, J. P. Bégué, D. Bonnet-Delpon, J. Org. Chem. 2005, 70, 699-702.
- (2005) J. Org. Chem. , vol.70 , pp. 699-702
- Tarn, N.T.N.¹ Magueur, G.² Ourevitch, M.³ Crousse, B.⁴ Bégué, J.P.⁵ Bonnet-Delpon, D.⁶

24
- 0030580414
- D. M. Hodgson, A. R. Gibbs, G. P. Lee, Tetrahedron 1996, 52, 14361-14384.
- (1996) Tetrahedron , vol.52 , pp. 14361-14384
- Hodgson, D.M.¹ Gibbs, A.R.² Lee, G.P.³

25
- 0000830825
- R. M. Hanson, Chem. Rev. 1991, 91, 437-475.
- (1991) Chem. Rev. , vol.91 , pp. 437-475
- Hanson, R.M.¹

26
- 0012543140
- K. Fagnou, M. Lautens, Org. Lett. 2000, 2, 2319-2321.
- (2000) Org. Lett. , vol.2 , pp. 2319-2321
- Fagnou, K.¹ Lautens, M.²

27
- 0033534609
- G. Sekar, V. K. Singh, J. Org. Chem. 1999, 64, 287-289.
- (1999) J. Org. Chem. , vol.64 , pp. 287-289
- Sekar, G.¹ Singh, V.K.²

28
- 0037423323
- R. H. Fan, X. L. Hou, J. Org. Chem. 2003, 68, 726-730.
- (2003) J. Org. Chem. , vol.68 , pp. 726-730
- Fan, R.H.¹ Hou, X.L.²

29
- 40049096344
- A. Procopio, M. Gaspari, M. Nardi, M. Oliverio, O. Rosati, Tetrahedron Lett. 2008, 49, 2289-2293.
- (2008) Tetrahedron Lett. , vol.49 , pp. 2289-2293
- Procopio, A.¹ Gaspari, M.² Nardi, M.³ Oliverio, M.⁴ Rosati, O.⁵

30
- 0034613328
- U. Das, B. Crousse, V. Kesavan, D. Bonnet-Delpon, J. P. Bégué, J. Org. Chem. 2000, 65, 6749-6751.
- (2000) J. Org. Chem. , vol.65 , pp. 6749-6751
- Das, U.¹ Crousse, B.² Kesavan, V.³ Bonnet-Delpon, D.⁴ Bégué, J.P.⁵

31
- 24044486238
- N. Azizi, M. R. Saidi, Org. Lett. 2005, 7, 3649-3651.
- (2005) Org. Lett. , vol.7 , pp. 3649-3651
- Azizi, N.¹ Saidi, M.R.²

32
- 0020448543
- P. W. Erhardt, C. M. Woo, R. J. Gorczynski, W. G. Anderson, J. Med. Chem. 1982, 25, 1402-1407.
- (1982) J. Med. Chem. , vol.25 , pp. 1402-1407
- Erhardt, P.W.¹ Woo, C.M.² Gorczynski, R.J.³ Anderson, W.G.⁴

33
- 0020371621
- P. W Erhardt, C. M. Woo, W. G. Anderson, R. J. Gorczynski, J. Med. Chem. 1982, 25, 1408-1412.
- (1982) J. Med. Chem. , vol.25 , pp. 1408-1412
- Erhardt, P.W.¹ Woo, C.M.² Anderson, W.G.³ Gorczynski, R.J.⁴

34
- 0036171131
- S. Higashibayashi, T. Mori, K. Shinko, K. Hashimoto, M. Nakata, Heterocyeles 2002, 57, 111-122.
- (2002) Heterocyeles , vol.57 , pp. 111-122
- Higashibayashi, S.¹ Mori, T.² Shinko, K.³ Hashimoto, K.⁴ Nakata, M.⁵

35
- 0001915652
- H. Kotsuki, T. Shimanouchi, M. Teraguchi, M. Kataoka, A. Tatsukawa, H. Nishizawa, Chem. Lett. 1994, 2159-2162.
- (1994) Chem. Lett. , pp. 2159-2162
- Kotsuki, H.¹ Shimanouchi, T.² Teraguchi, M.³ Kataoka, M.⁴ Tatsukawa, A.⁵ Nishizawa, H.⁶

36
- 24944476232
- S. Rodriguez-Escrich, D. Popa, C Jimeno, A. Vidal-Ferran, M. A. Pericas, Org. Lett. 2005, 7, 3829-3832.
- (2005) Org. Lett. , vol.7 , pp. 3829-3832
- Rodriguez-Escrich, S.¹ Popa, D.² Jimeno, C.³ Vidal-Ferran, A.⁴ Pericas, M.A.⁵

37
- 4944267509
- K. C. Nicolaou, M. Zak, B. S. Safina, S. H. Lee, A. A. Estrada, Angew. Chem. Int. Ed. 2004, 43, 5092-5097.
- (2004) Angew. Chem. Int. Ed. , vol.43 , pp. 5092-5097
- Nicolaou, K.C.¹ Zak, M.² Safina, B.S.³ Lee, S.H.⁴ Estrada, A.A.⁵

38
- 0001651112
- C. Coudures, R. Pastor, S. Szonyi, A. Cambon, J. Fluorine Chem. 1984, 24, 105-115.
- (1984) J. Fluorine Chem. , vol.24 , pp. 105-115
- Coudures, C.¹ Pastor, R.² Szonyi, S.³ Cambon, A.⁴

39
- 34250156659
- N. Vaiana, L. Rizzi, S. Romeo, Chem. Lett. 2007, 36, 648-649.
- (2007) Chem. Lett. , vol.36 , pp. 648-649
- Vaiana, N.¹ Rizzi, L.² Romeo, S.³

40
- 33750732286
- F. Saitoh, T Mukaihira, H. Nishida, T. Satoh, A. Okano, Y. Yumiya, M. Ohkouchi, R. Johka, T. Matsusue, I. Shiromizu, Y. Hosaka, M. Matsumoto, S. Ohnishi, Chem. Pharm. Bull. 2006, 54, 1535-1544.
- (2006) Chem. Pharm. Bull. , vol.54 , pp. 1535-1544
- Saitoh, F.¹ Mukaihira, T.² Nishida, H.³ Satoh, T.⁴ Okano, A.⁵ Yumiya, Y.⁶ Ohkouchi, M.⁷ Johka, R.⁸ Matsusue, T.⁹ Shiromizu, I.¹⁰ Hosaka, Y.¹¹ Matsumoto, M.¹² Ohnishi, S.¹³

41
- 0029657210
- S. Kiyohara, M. Sasaki, K. Saito, K. Sugita, T. Sugo, J. Membr. Sci. 1996, 109, 87-92.
- (1996) J. Membr. Sci. , vol.109 , pp. 87-92
- Kiyohara, S.¹ Sasaki, M.² Saito, K.³ Sugita, K.⁴ Sugo, T.⁵

42
- 0031055496
- J. W Janetka, P. Raman, K. Satyshur, G. R. Flentke, D. H. Rich, J. Am. Chem. Soc. 1997, 119, 441-442.
- (1997) J. Am. Chem. Soc. , vol.119 , pp. 441-442
- Janetka, J.W.¹ Raman, P.² Satyshur, K.³ Flentke, G.R.⁴ Rich, D.H.⁵

43
- 34547960784
- L. Kolaczkowski, D. M. Barnes, Org. Lett. 2007, 9, 3029-3032.
- (2007) Org. Lett. , vol.9 , pp. 3029-3032
- Kolaczkowski, L.¹ Barnes, D.M.²

44
- 0034873368
- C. Gravier-Pelletier, M. Milla, Y. Le Merrer, J. C. Depezay, Eur. J. Org. Chem. 2001, 3089-3096.
- (2001) Eur. J. Org. Chem. , pp. 3089-3096
- Gravier-Pelletier, C.¹ Milla, M.² Le Merrer, Y.³ Depezay, J.C.⁴

45
- 0023918228
- T. Tashiro, S. Fushiya, S. Nozoe, Chem. Pharm. Bull. 1988, 36, 893-901.
- (1988) Chem. Pharm. Bull. , vol.36 , pp. 893-901
- Tashiro, T.¹ Fushiya, S.² Nozoe, S.³

46
- 34250177709
- M. Sova, A. Babic, S. Pecar, S. Gobec, Tetrahedron 2007, 63, 141-1.47.
- (2007) Tetrahedron , vol.63 , pp. 141-147
- Sova, M.¹ Babic, A.² Pecar, S.³ Gobec, S.⁴

47
- 32244443005
- A. Babic, M. Sova, S. Gobec, S. Pecar, Tetrahedron Lett. 2006, 47, 1733-1735.
- (2006) Tetrahedron Lett. , vol.47 , pp. 1733-1735
- Babic, A.¹ Sova, M.² Gobec, S.³ Pecar, S.⁴

48
- 67449101067
- C. Philippe, T. Milcent, B. Crousse, D. Bonnet-Delpon, Org. Biomol. Chem. 2009, 7, 2026-2028.
- (2009) Org. Biomol. Chem. , vol.7 , pp. 2026-2028
- Philippe, C.¹ Milcent, T.² Crousse, B.³ Bonnet-Delpon, D.⁴

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