Mutant 5-hydroxytryptamine1A receptor D116A is a receptor activated solely by synthetic ligands with a rich pharmacology

Journal of Pharmacology and Experimental Therapeutics

Volumn 331, Issue 1, 2009, Pages 222-233

  Cussac, Didier ^a   Palmier, Christiane ^a   Finana, Frédéric ^a   De Vries, Luc ^a   Tardif, Stéphanie ^a   Léger, Céline ^a   Bernois, Sophie ^a   Heusler, Peter ^a  

^a INSTITUT DE RECHERCHE PIERRE FABRE   (France)

Author keywords

[No Author keywords available]

Indexed keywords

1 [2 (4 FLUOROBENZAMIDO)ETHYL] 4 (7 METHOXY 1 NAPHTHYL)PIPERAZINE; 2 DIPROPYLAMINO 8 HYDROXYTETRALIN; 4 DIPROPYLAMINO 1,3,4,5 TETRAHYDROBENZ[CD]INDOLE 6 CARBOXAMIDE; 5 CARBAMOYLTRYPTAMINE; ASPARTIC ACID; BUSPIRONE; ETHYLAMINE; FLESINOXAN; GUANOSINE; N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDYL)CYCLOHEXANECARBOXAMIDE; PINDOLOL; POTASSIUM CHANNEL; SEROTONIN 1A RECEPTOR; SEROTONIN 1A RECEPTOR D116A; SPIPERONE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BIOENGINEERING; CALCIUM MOBILIZATION; CHO CELL; CONTROLLED STUDY; NONHUMAN; NUCLEOTIDE SEQUENCE; OOCYTE; PRIORITY JOURNAL; SIGNAL TRANSDUCTION; XENOPUS LAEVIS;

8-HYDROXY-2-(DI-N-PROPYLAMINO)TETRALIN; ALANINE; AMINO ACID SUBSTITUTION; ANIMALS; ASPARTIC ACID; BINDING, COMPETITIVE; CHO CELLS; CRICETINAE; CRICETULUS; FEMALE; HUMANS; LIGANDS; MUTAGENESIS, SITE-DIRECTED; PIPERAZINES; PROTEIN BINDING; PYRIDINES; RECEPTOR, SEROTONIN, 5-HT1A; SEROTONIN RECEPTOR AGONISTS; XENOPUS LAEVIS;

EID: 70349308398     PISSN: 00223565     EISSN: 15210103     Source Type: Journal    
DOI: 10.1124/jpet.109.156307     Document Type: Article

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