Modulation of 5-HT1A receptor-mediated Ca2+ responses by co-expression with various recombinant Gα proteins in CH0-K1 cells

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 368, Issue 2, 2003, Pages 99-105

  Wurch, Thierry ^a   Pauwels, Petrus J ^a  

^a INSTITUT DE RECHERCHE PIERRE FABRE   (France)

Author keywords

5 HT1A receptor; Ca 2+ response; Efficacious and partial agonists; Recombinant G protein

Indexed keywords

2 DIPROPYLAMINO 8 HYDROXYTETRALIN; BUSPIRONE; CALCIUM ION; FLESINOXAN; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANINE NUCLEOTIDE BINDING PROTEIN ALPHA; IPSAPIRONE; METITEPINE; N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDYL)CYCLOHEXANECARBOXAMIDE; N [4 [5 [3 (2 AMINOETHYL) 1H INDOL 5 YL] 1,2,4 OXADIAZOL 3 YL]BENZYL]METHANESULFONAMIDE; PERTUSSIS TOXIN; SEROTONIN 1A RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CALCIUM TRANSPORT; CHIMERA; CHO CELL; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG EFFECT; DRUG POTENCY; KINETICS; NONHUMAN; NUCLEOTIDE SEQUENCE; PROTEIN EXPRESSION; PROTEIN PROTEIN INTERACTION;

ANIMALS; CALCIUM; CHO CELLS; CRICETINAE; CRICETULUS; ENZYME ACTIVATION; GTP-BINDING PROTEIN ALPHA SUBUNITS; HUMANS; KINETICS; LIGANDS; PHOSPHOLIPASE C; RECEPTOR, SEROTONIN, 5-HT1A; RECOMBINANT PROTEINS; SEROTONIN AGONISTS; SEROTONIN ANTAGONISTS; TIME FACTORS; TRANSFECTION;

EID: 0042878687     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/s00210-003-0769-5     Document Type: Article

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