-
1
-
-
57649122948
-
-
Geneva: World Health Organisation, 2008, 1
-
World Malaria Report 2008, Geneva: World Health Organisation, 2008, 1.
-
World Malaria Report 2008
-
-
-
4
-
-
0035521154
-
-
Coombs G.H., Goldberg D.E., Klemba M., Berry C., Kay J., and Mottram J.C. Trends Parasitol. 17 (2001) 532
-
(2001)
Trends Parasitol.
, vol.17
, pp. 532
-
-
Coombs, G.H.1
Goldberg, D.E.2
Klemba, M.3
Berry, C.4
Kay, J.5
Mottram, J.C.6
-
5
-
-
68149093503
-
-
Global burden of disease: 2004 update Geneva: World Health Organization, 2004.
-
Global burden of disease: 2004 update Geneva: World Health Organization, 2004.
-
-
-
-
6
-
-
0028287766
-
-
Dame J.B., Reddy G.R., Yowell C.A., Dunn B.M., Kay J., and Berry C. Mol. Biochem. Parasitol. 64 (1994) 177
-
(1994)
Mol. Biochem. Parasitol.
, vol.64
, pp. 177
-
-
Dame, J.B.1
Reddy, G.R.2
Yowell, C.A.3
Dunn, B.M.4
Kay, J.5
Berry, C.6
-
7
-
-
0037154180
-
-
Banerjee R., Liu J., Beatty W., Pelosof L., Klemba M., and Goldberg D.E. Proc. Natl. Acad. Sci. U.S.A. 99 (2002) 990
-
(2002)
Proc. Natl. Acad. Sci. U.S.A.
, vol.99
, pp. 990
-
-
Banerjee, R.1
Liu, J.2
Beatty, W.3
Pelosof, L.4
Klemba, M.5
Goldberg, D.E.6
-
9
-
-
54849435041
-
-
Luksch T., Chan N.S., Brass S., Sotriffer C.A., Klebe G., and Diederich W.E. Chemmedchem. 3 (2008) 1323
-
(2008)
Chemmedchem.
, vol.3
, pp. 1323
-
-
Luksch, T.1
Chan, N.S.2
Brass, S.3
Sotriffer, C.A.4
Klebe, G.5
Diederich, W.E.6
-
10
-
-
55749114914
-
-
Hidaka K., Kimura T., Ruben A.J., Uemura T., Kamiya M., Kiso A., Okamoto T., Tsuchiya Y., Hayashi Y., Freire E., and Kiso Y. Bioorg. Med. Chem. 16 (2008) 10049
-
(2008)
Bioorg. Med. Chem.
, vol.16
, pp. 10049
-
-
Hidaka, K.1
Kimura, T.2
Ruben, A.J.3
Uemura, T.4
Kamiya, M.5
Kiso, A.6
Okamoto, T.7
Tsuchiya, Y.8
Hayashi, Y.9
Freire, E.10
Kiso, Y.11
-
11
-
-
0141448822
-
-
Dame J.B., Yowell C.A., Omara-Opyene L., Carlton J.M., Cooper R.A., and Li T. Mol. Biochem. Parasitol. 130 (2003) 1
-
(2003)
Mol. Biochem. Parasitol.
, vol.130
, pp. 1
-
-
Dame, J.B.1
Yowell, C.A.2
Omara-Opyene, L.3
Carlton, J.M.4
Cooper, R.A.5
Li, T.6
-
12
-
-
1842662675
-
-
Li T., Yowell C.A., Beyer B.B., Hung S.-H., Westling J., Lam M.T., Dunn B.M., and Dame J.B. Mol. Biochem. Parasitol. 135 (2004) 101
-
(2004)
Mol. Biochem. Parasitol.
, vol.135
, pp. 101
-
-
Li, T.1
Yowell, C.A.2
Beyer, B.B.3
Hung, S.-H.4
Westling, J.5
Lam, M.T.6
Dunn, B.M.7
Dame, J.B.8
-
13
-
-
33646573016
-
-
Clemente J.C., Govindasamy L., Madabushi A., Fisher S.Z., Moose R.E., Yowell C.A., Hidaka K., Kimura T., Hayashi Y., Kiso Y., Agbandje-McKenna M., Dame J.B., Dunn B.M., and McKenna R. Acta Crystallogr., Sect. D 62 (2006) 246
-
(2006)
Acta Crystallogr., Sect. D
, vol.62
, pp. 246
-
-
Clemente, J.C.1
Govindasamy, L.2
Madabushi, A.3
Fisher, S.Z.4
Moose, R.E.5
Yowell, C.A.6
Hidaka, K.7
Kimura, T.8
Hayashi, Y.9
Kiso, Y.10
Agbandje-McKenna, M.11
Dame, J.B.12
Dunn, B.M.13
McKenna, R.14
-
14
-
-
11144237489
-
-
Omara-Opyene A.L., Moura P.A., Sulsona C.R., Bonilla J.A., Yowell C.A., Fujioka H., Fidock D.A., and Dame J.B. J. Biol. Chem. 279 (2004) 54088
-
(2004)
J. Biol. Chem.
, vol.279
, pp. 54088
-
-
Omara-Opyene, A.L.1
Moura, P.A.2
Sulsona, C.R.3
Bonilla, J.A.4
Yowell, C.A.5
Fujioka, H.6
Fidock, D.A.7
Dame, J.B.8
-
16
-
-
34250620398
-
-
Bonilla J.A., Bonilla T.D., Yowell C.A., Fujioka H., and Dame J.B. Mol. Microbiol. 65 (2007) 64
-
(2007)
Mol. Microbiol.
, vol.65
, pp. 64
-
-
Bonilla, J.A.1
Bonilla, T.D.2
Yowell, C.A.3
Fujioka, H.4
Dame, J.B.5
-
17
-
-
0037780064
-
-
Nezami A., Kimura T., Hidaka K., Kiso A., Liu J., Kiso Y., Goldberg D.E., and Freire E. Biochemistry 42 (2003) 8459
-
(2003)
Biochemistry
, vol.42
, pp. 8459
-
-
Nezami, A.1
Kimura, T.2
Hidaka, K.3
Kiso, A.4
Liu, J.5
Kiso, Y.6
Goldberg, D.E.7
Freire, E.8
-
18
-
-
8644243887
-
-
Kiso A., Hidaka K., Kimura T., Hayashi Y., Nezami A., Freire E., and Kiso Y. J. Pept. Sci. 10 (2004) 641
-
(2004)
J. Pept. Sci.
, vol.10
, pp. 641
-
-
Kiso, A.1
Hidaka, K.2
Kimura, T.3
Hayashi, Y.4
Nezami, A.5
Freire, E.6
Kiso, Y.7
-
19
-
-
29144501184
-
-
Ekegren J.K., Unge T., Safa M.Z., Wallberg H., Samuelsson B., and Hallberg A. J. Med. Chem. 48 (2005) 8098
-
(2005)
J. Med. Chem.
, vol.48
, pp. 8098
-
-
Ekegren, J.K.1
Unge, T.2
Safa, M.Z.3
Wallberg, H.4
Samuelsson, B.5
Hallberg, A.6
-
20
-
-
33746931600
-
-
Ekegren J.K., Gising J., Wallberg H., Larhed M., Samuelsson B., and Hallberg A. Org. Biomol. Chem. 4 (2006) 3040
-
(2006)
Org. Biomol. Chem.
, vol.4
, pp. 3040
-
-
Ekegren, J.K.1
Gising, J.2
Wallberg, H.3
Larhed, M.4
Samuelsson, B.5
Hallberg, A.6
-
21
-
-
39749165062
-
-
Wu X.Y., Öhrngren P., Ekegren J.K., Unge J., Unge T., Wallberg H., Samuelsson B., Hallberg A., and Larhed M. J. Med. Chem. 51 (2008) 1053
-
(2008)
J. Med. Chem.
, vol.51
, pp. 1053
-
-
Wu, X.Y.1
Öhrngren, P.2
Ekegren, J.K.3
Unge, J.4
Unge, T.5
Wallberg, H.6
Samuelsson, B.7
Hallberg, A.8
Larhed, M.9
-
22
-
-
13644263256
-
-
Beyer B.B., Johnson J.V., Chung A.Y., Li T., Madabushi A., Agbandje-McKenna M., McKenna R., Dame J.B., and Dunn B.M. Biochemistry 44 (2005) 1768
-
(2005)
Biochemistry
, vol.44
, pp. 1768
-
-
Beyer, B.B.1
Johnson, J.V.2
Chung, A.Y.3
Li, T.4
Madabushi, A.5
Agbandje-McKenna, M.6
McKenna, R.7
Dame, J.B.8
Dunn, B.M.9
-
23
-
-
84899807125
-
-
Howard-Lock H.E., Lock C.J.L., Martins M.L., Smalley P.S., and Bell R.A. Can. J. Chem. 64 (1986) 1215
-
(1986)
Can. J. Chem.
, vol.64
, pp. 1215
-
-
Howard-Lock, H.E.1
Lock, C.J.L.2
Martins, M.L.3
Smalley, P.S.4
Bell, R.A.5
-
24
-
-
0035534548
-
-
Yamansarova E.T., Kukovinets A.G., Kukovinets O.S., Zainullin R.A., Galin F.Z., Kunakova R.V., Zorin V.V., and Tolstikov G.A. Russ. J. Org. Chem. 37 (2001) 246
-
(2001)
Russ. J. Org. Chem.
, vol.37
, pp. 246
-
-
Yamansarova, E.T.1
Kukovinets, A.G.2
Kukovinets, O.S.3
Zainullin, R.A.4
Galin, F.Z.5
Kunakova, R.V.6
Zorin, V.V.7
Tolstikov, G.A.8
-
25
-
-
0031282557
-
-
Westling J., Yowell C.A., Majer P., Erickson J.W., Dame J.B., and Dunn B.M. Exp. Parasitol. 87 (1997) 185
-
(1997)
Exp. Parasitol.
, vol.87
, pp. 185
-
-
Westling, J.1
Yowell, C.A.2
Majer, P.3
Erickson, J.W.4
Dame, J.B.5
Dunn, B.M.6
-
26
-
-
34548348687
-
-
For a review, see:
-
For a review, see:. Bjelic S., Nervall M., Gutierrez-de-Terán H., Ersmark K., Hallberg A., and Åqvist J. Cell. Mol. Life Sci. 64 (2007) 2285
-
(2007)
Cell. Mol. Life Sci.
, vol.64
, pp. 2285
-
-
Bjelic, S.1
Nervall, M.2
Gutierrez-de-Terán, H.3
Ersmark, K.4
Hallberg, A.5
Åqvist, J.6
-
27
-
-
33748256153
-
-
Gutiérrez-de-Terán H., Nervall M., Ersmark K., Liu P., Janka L.K., Dunn B., Hallberg A., and Åqvist J. Biochemistry 45 (2006) 10529
-
(2006)
Biochemistry
, vol.45
, pp. 10529
-
-
Gutiérrez-de-Terán, H.1
Nervall, M.2
Ersmark, K.3
Liu, P.4
Janka, L.K.5
Dunn, B.6
Hallberg, A.7
Åqvist, J.8
-
28
-
-
34247849388
-
-
Hidaka K., Kimura T., Tsuchiya Y., Kamiya M., Ruben A.J., Freire E., Hayashi Y., and Kiso Y. Bioorg. Med. Chem. Lett. 17 (2007) 3048
-
(2007)
Bioorg. Med. Chem. Lett.
, vol.17
, pp. 3048
-
-
Hidaka, K.1
Kimura, T.2
Tsuchiya, Y.3
Kamiya, M.4
Ruben, A.J.5
Freire, E.6
Hayashi, Y.7
Kiso, Y.8
-
29
-
-
11144356514
-
-
Brynda J., Rezacova P., Fabry M., Horejsi M., Stouracova R., Sedlacek J., Soucek M., Hradilek M., Lepsik M., and Konvalinka J. J. Med. Chem. 47 (2004) 2030
-
(2004)
J. Med. Chem.
, vol.47
, pp. 2030
-
-
Brynda, J.1
Rezacova, P.2
Fabry, M.3
Horejsi, M.4
Stouracova, R.5
Sedlacek, J.6
Soucek, M.7
Hradilek, M.8
Lepsik, M.9
Konvalinka, J.10
-
30
-
-
52749095342
-
-
Janka L., Clemente J., Vaiana N., Sparatore A., Romeo S., and Dunn B.M. Protein Pept. Lett. 15 (2008) 868
-
(2008)
Protein Pept. Lett.
, vol.15
, pp. 868
-
-
Janka, L.1
Clemente, J.2
Vaiana, N.3
Sparatore, A.4
Romeo, S.5
Dunn, B.M.6
-
31
-
-
0036499447
-
-
Liu X.W., Hu X.E., Tian X.R., Mazur A., and Ebetino F.H. J. Organomet. Chem. 646 (2002) 212
-
(2002)
J. Organomet. Chem.
, vol.646
, pp. 212
-
-
Liu, X.W.1
Hu, X.E.2
Tian, X.R.3
Mazur, A.4
Ebetino, F.H.5
-
34
-
-
0033587124
-
-
Mimoto T., Kato R., Takaku H., Nojima S., Terashima K., Misawa S., Fukazawa T., Ueno T., Sato H., Shintani M., Kiso Y., and Hayashi H. J. Med. Chem. 42 (1999) 1789
-
(1999)
J. Med. Chem.
, vol.42
, pp. 1789
-
-
Mimoto, T.1
Kato, R.2
Takaku, H.3
Nojima, S.4
Terashima, K.5
Misawa, S.6
Fukazawa, T.7
Ueno, T.8
Sato, H.9
Shintani, M.10
Kiso, Y.11
Hayashi, H.12
-
36
-
-
0026627809
-
-
Thompson W.J., Fitzgerald P.M.D., Holloway M.K., Emini E.A., Darke P.L., Mckeever B.M., Schleif W.A., Quintero J.C., Zugay J.A., Tucker T.J., Schwering J.E., Homnick C.F., Nunberg J., Springer J.P., and Huff J.R. J. Med. Chem. 35 (1992) 1685
-
(1992)
J. Med. Chem.
, vol.35
, pp. 1685
-
-
Thompson, W.J.1
Fitzgerald, P.M.D.2
Holloway, M.K.3
Emini, E.A.4
Darke, P.L.5
Mckeever, B.M.6
Schleif, W.A.7
Quintero, J.C.8
Zugay, J.A.9
Tucker, T.J.10
Schwering, J.E.11
Homnick, C.F.12
Nunberg, J.13
Springer, J.P.14
Huff, J.R.15
-
37
-
-
0032880049
-
-
Westling J., Cipullo P., Hung S.H., Saft H., Dame J.B., and Dunn B.M. Protein Sci. 8 (1999) 2001
-
(1999)
Protein Sci.
, vol.8
, pp. 2001
-
-
Westling, J.1
Cipullo, P.2
Hung, S.H.3
Saft, H.4
Dame, J.B.5
Dunn, B.M.6
-
38
-
-
0033594354
-
-
Haque T.S., Skillman A.G., Lee C.E., Habashita H., Gluzman I.Y., Ewing T.J.A., Goldberg D.E., Kuntz I.D., and Ellman J.A. J. Med. Chem. 42 (1999) 1428
-
(1999)
J. Med. Chem.
, vol.42
, pp. 1428
-
-
Haque, T.S.1
Skillman, A.G.2
Lee, C.E.3
Habashita, H.4
Gluzman, I.Y.5
Ewing, T.J.A.6
Goldberg, D.E.7
Kuntz, I.D.8
Ellman, J.A.9
-
39
-
-
68149105204
-
-
Copeland R.A. (Ed), VCH, New York, NY
-
Copeland R.A. In: Copeland R.A. (Ed). Enzymes: A Practical Introduction to Structure, Mechanism, and Data Analysis (1996), VCH, New York, NY 300
-
(1996)
Enzymes: A Practical Introduction to Structure, Mechanism, and Data Analysis
, pp. 300
-
-
Copeland, R.A.1
-
42
-
-
0030664454
-
-
Nillroth U., Vrang L., Markgren P.-O., Hulten J., Hallberg A., and Danielson U.H. Antimicrob. Agents Chemother. 41 (1997) 2383
-
(1997)
Antimicrob. Agents Chemother.
, vol.41
, pp. 2383
-
-
Nillroth, U.1
Vrang, L.2
Markgren, P.-O.3
Hulten, J.4
Hallberg, A.5
Danielson, U.H.6
-
43
-
-
53749088436
-
-
Bäck M., Nyhlén J., Kvarnström I., Appelgren S., Borkakoti N., Jansson K., Lindberg J., Nyström S., Hallberg A., Rosenquist A., and Samuelsson B. Bioorg. Med. Chem. 16 (2008) 9471
-
(2008)
Bioorg. Med. Chem.
, vol.16
, pp. 9471
-
-
Bäck, M.1
Nyhlén, J.2
Kvarnström, I.3
Appelgren, S.4
Borkakoti, N.5
Jansson, K.6
Lindberg, J.7
Nyström, S.8
Hallberg, A.9
Rosenquist, A.10
Samuelsson, B.11
-
44
-
-
0031552362
-
-
Jones G., Willett P., Glen R.C., Leach A.R., and Taylor R. J. Mol. Biol. 267 (1997) 727
-
(1997)
J. Mol. Biol.
, vol.267
, pp. 727
-
-
Jones, G.1
Willett, P.2
Glen, R.C.3
Leach, A.R.4
Taylor, R.5
-
47
-
-
0004016501
-
-
Jorgensen W.L., Chandrasekhar J., Madura J.D., Impey R.W., and Klein M.L. J. Chem. Phys. 79 (1983) 926
-
(1983)
J. Chem. Phys.
, vol.79
, pp. 926
-
-
Jorgensen, W.L.1
Chandrasekhar, J.2
Madura, J.D.3
Impey, R.W.4
Klein, M.L.5
|