Additional interaction of allophenylnorstatine-containing tripeptidomimetics with malarial aspartic protease plasmepsin II

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 11, 2007, Pages 3048-3052

  Hidaka, Koushi ^a   Kimura, Tooru ^a   Tsuchiya, Yumi ^a   Kamiya, Mami ^a   Ruben, Adam J ^b   Freire, Ernesto ^b   Hayashi, Yoshio ^a   Kiso, Yoshiaki ^a  

^a Center for Frontier Research in Medicinal Science   (Japan)

^b JOHNS HOPKINS UNIVERSITY   (United States)

Author keywords

Allophenylnorstatine; Aspartic protease; Malaria; Peptidomimetic; Plasmepsin inhibitor

Indexed keywords

ALLOPHENYLNORSTATINE; ANTIPARASITIC AGENT; ASPARTIC PROTEINASE; KNI 10033; KNI 10061; KNI 10062; KNI 10232; KNI 10233; KNI 10313; KNI 10315; KNI 10316; KNI 10332; KNI 10333; KNI 10341; KNI 10343; KNI 10368; KNI 10372; KNI 10395; PLASMEPSIN II; STATINE DERIVATIVE; TRIPEPTIDE DERIVATIVE; TRIPEPTIDOMIMETIC DERIVATIVE; UNCLASSIFIED DRUG;

AMINO TERMINAL SEQUENCE; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG STRUCTURE; ENZYME INHIBITION; HYDROPHOBICITY; NONHUMAN; PLASMODIUM FALCIPARUM;

ANIMALS; ANTIMALARIALS; ASPARTIC ENDOPEPTIDASES; BIOMIMETIC MATERIALS; OLIGOPEPTIDES; PHENYLBUTYRATES; PLASMODIUM FALCIPARUM; PROTEASE INHIBITORS; PROTEIN CONFORMATION; STRUCTURE-ACTIVITY RELATIONSHIP;

PLASMODIUM FALCIPARUM;

EID: 34247849388     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2007.03.052     Document Type: Article

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