Organic blockers escape from trapping in the AMPA receptor channels by leaking into the cytoplasm

Neuropharmacology

Volumn 54, Issue 4, 2008, Pages 653-664

  Tikhonova, T B ^a   Barygin, O I ^a   Gmiro, V E ^b   Tikhonov, D B ^a   Magazanik, L G ^a  

^a SECHENOV INSTITUTE OF EVOLUTIONARY PHYSIOLOGY AND BIOCHEMISTRY   (Russian Federation)

^b INSTITUTE OF EXPERIMENTAL MEDICINE   (Russian Federation)

Author keywords

AMPA receptor; Channel block; Channel gating; Permeation

Indexed keywords

ADAMANTANE DERIVATIVE; AMPA RECEPTOR; AMPA RECEPTOR ANTAGONIST; BENZENE DERIVATIVE; SPERMINE;

ANIMAL EXPERIMENT; ARTICLE; CHANNEL GATING; CONTROLLED STUDY; CYTOPLASM; DATA ANALYSIS; INTERNEURON; KINETICS; NONHUMAN; PRIORITY JOURNAL; QUANTITATIVE ANALYSIS; RAT; RECEPTOR BLOCKING; SYNAPTIC TRANSMISSION;

ANIMALS; ANIMALS, NEWBORN; BRAIN; CYTOPLASM; DOSE-RESPONSE RELATIONSHIP, RADIATION; ELECTRIC STIMULATION; EXCITATORY AMINO ACID AGONISTS; ION CHANNEL GATING; KAINIC ACID; KINETICS; MEMBRANE POTENTIALS; NEURONS; PATCH-CLAMP TECHNIQUES; QUATERNARY AMMONIUM COMPOUNDS; RATS; RATS, WISTAR; RECEPTORS, AMPA; TIME FACTORS;

EID: 38749105436     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.neuropharm.2007.11.014     Document Type: Article

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