Voltage-dependent block of native AMPA receptor channels by dicationic compounds

British Journal of Pharmacology

Volumn 129, Issue 2, 2000, Pages 265-274

  Tikhonov, D B ^a   Samoilova, M V ^a   Buldakova, S L ^a   Gmiro, V E ^b   Magazanik, L G ^a  

^a SECHENOV INSTITUTE OF EVOLUTIONARY PHYSIOLOGY AND BIOCHEMISTRY   (Russian Federation)

^b INSTITUTE OF BIOMEDICAL CHEMISTRY   (Russian Federation)

Author keywords

AMPA receptor; Channel block; Kinetics; Permeation; Structure activity relationships; Voltage dependence

Indexed keywords

1 (1 ADAMANTYLMETHYLAMMONIO) 5 TRIMETHYLAMMONIOPENTANE DIBROMIDE; 1 ADAMANTYLMETHYLAMMONIO 5 AMMONIOPENTANE DIBROMIDE; 1 TRIMETHYLAMMONIO 5 (1 ADAMANTANEMETHYLAMMONIOPENTANE) DIBROMIDE; 5 AMINOPENTYL 1 PHENYLCYCLOHEXYLAMINE DIBROMIDE; AMPA RECEPTOR; DIVALENT CATION; N (5 AMMONIOPENTYL) 1 PHENYLCYCLOHEXYLAMMONIUM DIBROMIDE; RECEPTOR SUBUNIT; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CELL MEMBRANE POTENTIAL; CONTROLLED STUDY; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; HIPPOCAMPUS; HYPERPOLARIZATION; NERVE CELL; NEWBORN; NONHUMAN; PATCH CLAMP; PRIORITY JOURNAL; RAT; RECEPTOR BLOCKING;

EID: 0033978845     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0703043     Document Type: Article

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