-
2
-
-
0037355137
-
-
Marminon C., Pierre A., Pfeiffer B., Pérez V., Léonce S., Renard P., and Prudhomme M. Bioorg. Med. Chem. 11 (2003) 679-687
-
(2003)
Bioorg. Med. Chem.
, vol.11
, pp. 679-687
-
-
Marminon, C.1
Pierre, A.2
Pfeiffer, B.3
Pérez, V.4
Léonce, S.5
Renard, P.6
Prudhomme, M.7
-
3
-
-
0035924236
-
-
Mahboobi S., Pongratz H., Hufsky H., Hockemeyer J., Frieser M., Lyssenko A., Paper D., Burgermeister J., Bohmer F., Fiebig H., Burger A., Baasner S., and Beckers T. J. Med. Chem. 44 (2001) 4535-4553
-
(2001)
J. Med. Chem.
, vol.44
, pp. 4535-4553
-
-
Mahboobi, S.1
Pongratz, H.2
Hufsky, H.3
Hockemeyer, J.4
Frieser, M.5
Lyssenko, A.6
Paper, D.7
Burgermeister, J.8
Bohmer, F.9
Fiebig, H.10
Burger, A.11
Baasner, S.12
Beckers, T.13
-
4
-
-
2442687670
-
-
Messaoudi S., Anizon F., Pfeiffer B., Golsteyn R., and Prudhomme M. Tetrahedron Lett. 45 (2004) 4643-4647
-
(2004)
Tetrahedron Lett.
, vol.45
, pp. 4643-4647
-
-
Messaoudi, S.1
Anizon, F.2
Pfeiffer, B.3
Golsteyn, R.4
Prudhomme, M.5
-
8
-
-
2542434120
-
-
O'Neil D.J., Shen L., Prouty C., Conway B.R., Westover L., Xu J.Z., Zhang H.-C., Maryanoff B.E., Murray W.V., Demarest K.T., and Kuo G.-H. Bioorg. Med. Chem. 12 (2004) 3167-3185
-
(2004)
Bioorg. Med. Chem.
, vol.12
, pp. 3167-3185
-
-
O'Neil, D.J.1
Shen, L.2
Prouty, C.3
Conway, B.R.4
Westover, L.5
Xu, J.Z.6
Zhang, H.-C.7
Maryanoff, B.E.8
Murray, W.V.9
Demarest, K.T.10
Kuo, G.-H.11
-
12
-
-
33750089733
-
-
Gluszok S., Goossens L., Depreux P., Barbry D., and Hénichart J.-P. Synth. Commun. 36 (2006) 2797-2805
-
(2006)
Synth. Commun.
, vol.36
, pp. 2797-2805
-
-
Gluszok, S.1
Goossens, L.2
Depreux, P.3
Barbry, D.4
Hénichart, J.-P.5
-
13
-
-
33646497023
-
-
Wang X., Zhi B., Baum J., Chen Y., Crockett R., Huang L., Eisenberg S., Ng J., Larsen R., Martinelli M., and Reider P. J. Org. Chem. 71 (2006) 4021-4023
-
(2006)
J. Org. Chem.
, vol.71
, pp. 4021-4023
-
-
Wang, X.1
Zhi, B.2
Baum, J.3
Chen, Y.4
Crockett, R.5
Huang, L.6
Eisenberg, S.7
Ng, J.8
Larsen, R.9
Martinelli, M.10
Reider, P.11
-
14
-
-
33847782088
-
-
Guillard J., Decrop M., Gallay N., Espanel C., Boissier E., Herault O., and Viaud-Massuard M.C. Bioorg. Med. Chem. Lett. 17 (2007) 1934-1937
-
(2007)
Bioorg. Med. Chem. Lett.
, vol.17
, pp. 1934-1937
-
-
Guillard, J.1
Decrop, M.2
Gallay, N.3
Espanel, C.4
Boissier, E.5
Herault, O.6
Viaud-Massuard, M.C.7
-
15
-
-
33746655450
-
-
Bignan G.C., Battista K., Connolly P.J., Orsini J.J., Liu J., Middleton S.A., and Reitz A.B. Bioorg. Med. Chem. Lett. 16 (2006) 3524-3528
-
(2006)
Bioorg. Med. Chem. Lett.
, vol.16
, pp. 3524-3528
-
-
Bignan, G.C.1
Battista, K.2
Connolly, P.J.3
Orsini, J.J.4
Liu, J.5
Middleton, S.A.6
Reitz, A.B.7
-
16
-
-
34447645673
-
-
Elokdah H., Li D., McFarlane G., Bernotas R.C., Robichaud A.J., Magolda R.L., Zhang G.M., Smith D., and Schechter L.E. Bioorg. Med. Chem. 15 (2007) 6208-6226
-
(2007)
Bioorg. Med. Chem.
, vol.15
, pp. 6208-6226
-
-
Elokdah, H.1
Li, D.2
McFarlane, G.3
Bernotas, R.C.4
Robichaud, A.J.5
Magolda, R.L.6
Zhang, G.M.7
Smith, D.8
Schechter, L.E.9
-
17
-
-
34447283531
-
-
Hugon B., Anizon F., Bailly C., Golsteyn R.M., Pierré A., Léonce S., Hickman J., Pfeiffer B., and Prudhomme M. Bioorg. Med. Chem. 15 (2007) 5965-5980
-
(2007)
Bioorg. Med. Chem.
, vol.15
, pp. 5965-5980
-
-
Hugon, B.1
Anizon, F.2
Bailly, C.3
Golsteyn, R.M.4
Pierré, A.5
Léonce, S.6
Hickman, J.7
Pfeiffer, B.8
Prudhomme, M.9
-
18
-
-
33746805407
-
-
Huang S., Li R., Connolly P.J., Emanuel S., and Middleton S.A. Bioorg. Med. Chem. Lett. 16 (2006) 4818-4821
-
(2006)
Bioorg. Med. Chem. Lett.
, vol.16
, pp. 4818-4821
-
-
Huang, S.1
Li, R.2
Connolly, P.J.3
Emanuel, S.4
Middleton, S.A.5
-
20
-
-
34548475073
-
-
Potashman M.H., Bready J., Coxon A., DeMelfi T.M., DiPrietro L., Doerr N., Elbaum D., Estrada J., Gallant P., Germain J., Gu Y., Harmange J.-C., Kaufman S.A., Kendall R., Kim J.L., Kumar G.N., Long A.M., Neervannan S., Patel V.F., Polverino A., Rose P., van der Plas S., Whittington D., Zanon R., and Zhao H. J. Med. Chem. 50 (2007) 4351-4373
-
(2007)
J. Med. Chem.
, vol.50
, pp. 4351-4373
-
-
Potashman, M.H.1
Bready, J.2
Coxon, A.3
DeMelfi, T.M.4
DiPrietro, L.5
Doerr, N.6
Elbaum, D.7
Estrada, J.8
Gallant, P.9
Germain, J.10
Gu, Y.11
Harmange, J.-C.12
Kaufman, S.A.13
Kendall, R.14
Kim, J.L.15
Kumar, G.N.16
Long, A.M.17
Neervannan, S.18
Patel, V.F.19
Polverino, A.20
Rose, P.21
van der Plas, S.22
Whittington, D.23
Zanon, R.24
Zhao, H.25
more..
-
21
-
-
4544224760
-
-
Nazaré M., Scheneider C., Lindenschmidt A., and Will D.W. Angew. Chem., Int. Ed. 43 (2004) 4526-4528
-
(2004)
Angew. Chem., Int. Ed.
, vol.43
, pp. 4526-4528
-
-
Nazaré, M.1
Scheneider, C.2
Lindenschmidt, A.3
Will, D.W.4
-
27
-
-
0037023480
-
-
Zhang Z., Yang Z., Meanwell N.A., Kadow J.F., and Wang T. J. Org. Chem. 67 (2002) 2345-2347
-
(2002)
J. Org. Chem.
, vol.67
, pp. 2345-2347
-
-
Zhang, Z.1
Yang, Z.2
Meanwell, N.A.3
Kadow, J.F.4
Wang, T.5
-
30
-
-
33748598708
-
-
and references cited therein
-
Zheng X., and Kerr M.A. Org. Lett. 8 (2006) 3777-3779 and references cited therein
-
(2006)
Org. Lett.
, vol.8
, pp. 3777-3779
-
-
Zheng, X.1
Kerr, M.A.2
-
32
-
-
0033593964
-
-
Curtis N., Kulagowski J., Leeson P., Ridgill M., Emms F., Freedman S.B., Patel S., and Patel S. Bioorg. Med. Chem. Lett. 9 (1999) 585-588
-
(1999)
Bioorg. Med. Chem. Lett.
, vol.9
, pp. 585-588
-
-
Curtis, N.1
Kulagowski, J.2
Leeson, P.3
Ridgill, M.4
Emms, F.5
Freedman, S.B.6
Patel, S.7
Patel, S.8
-
38
-
-
0029929186
-
-
Hands D., Bishop B., Cameron M., Edwards J., Cottrell I., and Wright S. Synthesis (1996) 877-882
-
(1996)
Synthesis
, pp. 877-882
-
-
Hands, D.1
Bishop, B.2
Cameron, M.3
Edwards, J.4
Cottrell, I.5
Wright, S.6
-
42
-
-
12644258541
-
-
Dillard R.D., Bach N.J., Draheim S.E., Berry D.R., Carlson D.G., Chirgadze N.Y., Clawson D.K., Hartley L.W., Johnson L.M., Jones N.D., McKinney E.R., Mihelich E.D., Olkowski J.L., Schevits R.W., Smith A.C., Snyder D.W., Sommers C.D., and Wery J.-P. J. Med. Chem. 39 (1996) 5119-5136
-
(1996)
J. Med. Chem.
, vol.39
, pp. 5119-5136
-
-
Dillard, R.D.1
Bach, N.J.2
Draheim, S.E.3
Berry, D.R.4
Carlson, D.G.5
Chirgadze, N.Y.6
Clawson, D.K.7
Hartley, L.W.8
Johnson, L.M.9
Jones, N.D.10
McKinney, E.R.11
Mihelich, E.D.12
Olkowski, J.L.13
Schevits, R.W.14
Smith, A.C.15
Snyder, D.W.16
Sommers, C.D.17
Wery, J.-P.18
-
43
-
-
23944514825
-
-
Mattsson C., Sonesson C., Sandahl A., Greiner H.E., Gassen M., Plashke J., Leibrock J., and Böttcher H. Bioorg. Med. Chem. Lett. 15 (2005) 4230-4234
-
(2005)
Bioorg. Med. Chem. Lett.
, vol.15
, pp. 4230-4234
-
-
Mattsson, C.1
Sonesson, C.2
Sandahl, A.3
Greiner, H.E.4
Gassen, M.5
Plashke, J.6
Leibrock, J.7
Böttcher, H.8
-
44
-
-
36749060868
-
-
note
-
For the preparation of 3-methyl-2-(N-tert-butoxy carbonyl)aminopyridine see experimental procedures in Section 4.
-
-
-
-
47
-
-
0025787448
-
-
Clark R., Muchowski J., Fisher L., Flippin F., Repke D., and Souchet M. Synthesis (1991) 871-878
-
(1991)
Synthesis
, pp. 871-878
-
-
Clark, R.1
Muchowski, J.2
Fisher, L.3
Flippin, F.4
Repke, D.5
Souchet, M.6
|