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A very comprehensive review that deals with all aspects of the chemistry of different classes of CCK1R and CCK2R antagonists.
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Herranz R. Cholecystokinin antagonists: pharmacological and therapeutic potential. Med Res Rev 23 (2003) 559-605. A very comprehensive review that deals with all aspects of the chemistry of different classes of CCK1R and CCK2R antagonists.
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Herranz, R.1
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Role of CCK/gastrin receptors in gastrointestinal/metabolic diseases and results of human studies using gastrin/CCK receptor agonists/antagonists in these diseases
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A comprehensive paper that reviews both studies of CCK ligands in gastrointestinal diseases as well as the data supporting potential uses in other disorders.
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Berna M.J., and Jensen R.T. Role of CCK/gastrin receptors in gastrointestinal/metabolic diseases and results of human studies using gastrin/CCK receptor agonists/antagonists in these diseases. Curr Top Med Chem 7 (2007) 1211-1231. A comprehensive paper that reviews both studies of CCK ligands in gastrointestinal diseases as well as the data supporting potential uses in other disorders.
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Curr Top Med Chem
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Berna, M.J.1
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Strategies for the design of non-peptide CCK2 receptor agonist and antagonist ligand
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An up-to-date report that reviews the development and characterization of the different classes of nonpeptide CCK2R agonists/antagonists.
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Kalindjian S.B., and McDonald I.M. Strategies for the design of non-peptide CCK2 receptor agonist and antagonist ligand. Curr Top Med Chem 7 (2007) 1195-1204. An up-to-date report that reviews the development and characterization of the different classes of nonpeptide CCK2R agonists/antagonists.
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Kalindjian, S.B.1
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Strategies for design of non peptide CCK1R agonist/antagonist ligands
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An up-to-date report that reviews the development and characterization of the different classes of nonpeptide CCK1R agonists/antagonists.
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Garcia-Lopez M.T., Gonzalez-Muniz R., Martin-Martinez M., and Herranz R. Strategies for design of non peptide CCK1R agonist/antagonist ligands. Curr Top Med Chem 7 (2007) 1180-1194. An up-to-date report that reviews the development and characterization of the different classes of nonpeptide CCK1R agonists/antagonists.
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Curr Top Med Chem
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A comprehensive review of the chemistry and pharmacology of recently developed nonpeptide CCK1R agonists.
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A up-to-date comprehensive review of the cell biology, pharmacology and physiology of both CCK and gastrin and their receptors.
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A concise review of the results of clinical studies of CCK1R antagonists as well as a review of the evidence suggesting other diseases they may be useful in.
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An extensive review of the investigated and possible gastrointestinal disorders that CCK or gastrin receptors may be involved in and in which either CCKR agonists or antagonists might be useful therapeutically.
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