Robust lanthanide-based assays for the detection of anti-apoptotic Bcl-2-family protein antagonists

Bioorganic Chemistry

Volumn 35, Issue 2, 2007, Pages 113-120

  Rega, Michele F ^a   Reed, John C ^a   Pellecchia, Maurizio ^a  

^a BURNHAM INSTITUTE   (United States)

Author keywords

Apoptosis; Bcl 2; Bcl xL; BH3; FRET

Indexed keywords

ANTINEOPLASTIC AGENT; BH3 PROTEIN; LANTHANIDE; PROTEIN BCL 2; PROTEIN INHIBITOR;

ARTICLE; DRUG DETERMINATION; HIGH THROUGHPUT SCREENING; PRIORITY JOURNAL; PROTEIN FAMILY; PROTEIN PROTEIN INTERACTION; REPRODUCIBILITY;

AMINO ACID SEQUENCE; ANTINEOPLASTIC AGENTS; APOPTOSIS; BH3 INTERACTING DOMAIN DEATH AGONIST PROTEIN; DOSE-RESPONSE RELATIONSHIP, DRUG; ENZYME-LINKED IMMUNOSORBENT ASSAY; FLUORESCENCE RESONANCE ENERGY TRANSFER; FLUOROIMMUNOASSAY; HUMANS; LANTHANOID SERIES ELEMENTS; MOLECULAR SEQUENCE DATA; PROTO-ONCOGENE PROTEINS C-BCL-2; REPRODUCIBILITY OF RESULTS;

EID: 33847631287     PISSN: 00452068     EISSN: 10902120     Source Type: Journal    
DOI: 10.1016/j.bioorg.2006.07.006     Document Type: Article

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