Allosteric modulation of [3H]EBOB binding to GABAA receptors by diflunisal analogues

Neurochemistry International

Volumn 49, Issue 7, 2006, Pages 676-682

  Uusi Oukari, Mikko ^a,b   Maksay, Gábor ^a  

^a CHEMICAL RESEARCH CENTER   (Hungary)

^b UNIVERSITY OF TURKU   (Finland)

Author keywords

Allosteric modulation; Diflunisal; GABA; GABA receptor; Meclofenamate

Indexed keywords

4 AMINOBUTYRIC ACID A RECEPTOR; 4' ETHYNYLBICYCLOORTHOBENZOATE H 3; BLOCKING AGENT; CONVULSANT AGENT; DIFLUNISAL; EFENAMIC ACID; MECLOFENAMIC ACID; UNCLASSIFIED DRUG; 1 (4 ETHYNYLPHENYL) 4 PROPYL 2,6,7 TRIOXABICYCLO(2.2.2)OCTANE; 1-(4-ETHYNYLPHENYL)-4-PROPYL-2,6,7-TRIOXABICYCLO(2.2.2)OCTANE; 4 AMINOBUTYRIC ACID; BIPHENYL DERIVATIVE; DRUG DERIVATIVE; FUSED HETEROCYCLIC RINGS; HYDROXYL RADICAL; NONSTEROID ANTIINFLAMMATORY AGENT;

ALLOSTERISM; ANIMAL TISSUE; ANTIINFLAMMATORY ACTIVITY; ARTICLE; BINDING AFFINITY; DRUG EFFECT; DRUG POTENCY; DRUG RECEPTOR BINDING; ELECTRON; ELECTRON TRANSPORT; FOREBRAIN; GABAERGIC TRANSMISSION; MALE; NEUROCHEMISTRY; NEUROMODULATION; NEUROPHARMACOLOGY; NONHUMAN; PHARMACODYNAMICS; PRIORITY JOURNAL; RAT; STRUCTURE ACTIVITY RELATION; SYNAPTIC MEMBRANE; AFFINITY LABELING; ANIMAL; BINDING COMPETITION; BINDING SITE; CHEMICAL STRUCTURE; CHEMISTRY; CONFORMATION; METABOLISM; PHYSIOLOGY; RADIOASSAY; SPRAGUE DAWLEY RAT; SYNAPTIC TRANSMISSION;

AFFINITY LABELS; ALLOSTERIC REGULATION; ANIMALS; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; BICYCLO COMPOUNDS, HETEROCYCLIC; BINDING SITES; BINDING, COMPETITIVE; BIPHENYL COMPOUNDS; DIFLUNISAL; GAMMA-AMINOBUTYRIC ACID; HYDROXYL RADICAL; MALE; MECLOFENAMIC ACID; MOLECULAR CONFORMATION; MOLECULAR STRUCTURE; PROSENCEPHALON; RADIOLIGAND ASSAY; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, GABA-A; SYNAPTIC TRANSMISSION;

EID: 33750020869     PISSN: 01970186     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.neuint.2006.06.001     Document Type: Article

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