Compounds exhibiting selective efficacy for different β subunits of human recombinant γ-aminobutyric acidA receptors

Journal of Pharmacology and Experimental Therapeutics

Volumn 311, Issue 2, 2004, Pages 601-609

  Smith, Alison J ^a   Oxley, Beth ^a   Malpas, Sallie ^a   Pillai, Gopalan V ^a   Simpson, Peter B ^a  

^a NEUROSCIENCE RESEARCH CENTRE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

3ALPHA HYDROXY 5ALPHA PREGNAN 20 ONE; 4 AMINOBUTYRIC ACID A RECEPTOR; 4 ETHYL 6,7 DIMETHOXY BETA CARBOLINE 3 CARBOXYLIC ACID METHYL ESTER; 4 PIPERIDINESULFONIC ACID; ANTIINFLAMMATORY AGENT; BIS(1,3 DIETHYL 2 THIOBARBITURATE)TRIMETHINEOXONOL; CHLOROCOUMARIN 2 DIMYRISTOYLPHOSPHATIDYLETHANOLAMINE; DIFLUNISAL; ETOMIDATE; FLUFENAMIC ACID; GABOXADOL; LORECLEZOLE; MECLOFENAMIC ACID; MEFENAMIC ACID; NIFLUMIC ACID; PENTOBARBITAL; PHOSPHATIDYLETHANOLAMINE; PROPOFOL; RECEPTOR SUBUNIT; RECOMBINANT PROTEIN; RENANOLONE; STEROID; THIOBARBITURIC ACID DERIVATIVE; TOLFENAMIC ACID; UNCLASSIFIED DRUG;

ALLOSTERISM; AMPLITUDE MODULATION; ANIMAL CELL; ARTICLE; CENTRAL NERVOUS SYSTEM DISEASE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG EFFICACY; DRUG POTENCY; DRUG RECEPTOR BINDING; FLUORESCENCE RESONANCE ENERGY TRANSFER; GABAERGIC SYSTEM; HUMAN; HUMAN CELL; MEMBRANE DEPOLARIZATION; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION;

ANESTHETICS; ANIMALS; ANTI-INFLAMMATORY AGENTS; GABA ANTAGONISTS; GAMMA-AMINOBUTYRIC ACID; HUMANS; MICE; PROTEIN SUBUNITS; RECEPTORS, GABA-A; TRANSFECTION;

EID: 6344256342     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: 10.1124/jpet.104.070342     Document Type: Article

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