Allosteric modulation of 5-HT3 serotonin receptors

European Journal of Pharmacology

Volumn 514, Issue 1, 2005, Pages 17-24

  Maksay, Gábor ^a   Bíró, Tímea ^a   Bugovics, Gyula ^b  

^a INSTITUTE OF EXPERIMENTAL MEDICINE   (Hungary)

^b GEDEON RICHTER LTD   (Hungary)

Author keywords

5 HT3 serotonin receptor binding; Allosteric modulation; Ifenprodil; NG 108 15 cell; Slope of displacement; Verapamil

Indexed keywords

4 (4 FLUOROPHENYL) 6 PROPIONYLOYL 1 AZABICYCLO[3.3.1]NON 3 ENE; GRANISETRON; GYKI 46903; IFENPRODIL; SEROTONIN 3 AGONIST; SEROTONIN 3 RECEPTOR; TRICHLOROETHANOL; UNCLASSIFIED DRUG; VERAPAMIL;

ALLOSTERISM; ANIMAL CELL; ARTICLE; CELL STRAIN; CONTROLLED STUDY; DRUG BINDING; FOREBRAIN; IN VITRO STUDY; MEDICAL LITERATURE; NONHUMAN; PRIORITY JOURNAL; QUANTITATIVE ANALYSIS; RAT; RECEPTOR BINDING;

ADRENERGIC ALPHA-ANTAGONISTS; ALGORITHMS; ALLOSTERIC REGULATION; ANIMALS; BINDING, COMPETITIVE; CELL LINE, TUMOR; DOSE-RESPONSE RELATIONSHIP, DRUG; GRANISETRON; HYBRID CELLS; KINETICS; MALE; MICE; MODELS, BIOLOGICAL; PIPERIDINES; RATS; RATS, WISTAR; RECEPTORS, SEROTONIN, 5-HT3; SEROTONIN; SEROTONIN AGENTS; TRITIUM; VERAPAMIL;

EID: 18844377448     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejphar.2005.03.019     Document Type: Article

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