High affinity, heterogeneous displacement of [3H]EBOB binding to cerebellar GABAA receptors by neurosteroids and GABA agonists

Neuropharmacology

Volumn 49, Issue 4, 2005, Pages 431-438

  Maksay, Gábor ^a   Bíró, Tímea ^a  

^a CHEMICAL RESEARCH CENTER   (Hungary)

Author keywords

6 GABAA receptors; 3H EBOB binding; Allopregnanolone; Furosemide; Taurine; THDOC epimers

Indexed keywords

3ALPHA HYDROXY 5ALPHA PREGNAN 20 ONE; 4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID A RECEPTOR; 4 AMINOBUTYRIC ACID RECEPTOR STIMULATING AGENT; 5ALPHA TETRAHYDRODEOXYCORTICOSTERONE; CONVULSANT AGENT; ETHYNYLBICYCLOORTHOBENZOATE H3; FUROSEMIDE; NEUROSTEROID; RADIOLIGAND; TAURINE; TETRAHYDRODEOXYCORTICOSTERONE; TRITIUM; UNCLASSIFIED DRUG;

ALLOSTERISM; ANIMAL TISSUE; ARTICLE; CEREBELLUM; CONCENTRATION RESPONSE; DRUG POTENCY; DRUG RECEPTOR BINDING; HIPPOCAMPUS; MOLECULAR INTERACTION; NEUROTRANSMISSION; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY;

ANIMALS; ANTI-ANXIETY AGENTS; BICYCLO COMPOUNDS, HETEROCYCLIC; BINDING, COMPETITIVE; CEREBELLUM; DESOXYCORTICOSTERONE; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG INTERACTIONS; GABA AGONISTS; GAMMA-AMINOBUTYRIC ACID; HIPPOCAMPUS; MALE; PREGNANOLONE; PROTEIN BINDING; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; RECEPTORS, GABA-A;

EID: 23844445260     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.neuropharm.2005.04.003     Document Type: Article

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