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ChemBioChem

Volumn 7, Issue 10, 2006, Pages 1478-1490

Highly potent vitamin D receptor antagonists: Design, synthesis, and biological evaluation

(2) Saito, Nozomi a Kittaka, Atsushi a

a TEIKYO UNIVERSITY (Japan)

Author keywords

Antagonists; Lactones; Receptors; Structure activity relationships; Vitamins

Indexed keywords

ETHYLENE; LACTONE DERIVATIVE; RECEPTOR BLOCKING AGENT; RUTHENIUM; TEI 9647; TEI 9648; UNCLASSIFIED DRUG; VITAMIN D; VITAMIN D RECEPTOR; VITAMIN D RECEPTOR ANTAGONIST; CALCITRIOL; CALCITRIOL RECEPTOR; DRUG DERIVATIVE; LACTONE;

BONE MALFORMATION; BONE REMODELING; CATALYSIS; CELL DIFFERENTIATION; CYCLOPROPANATION; DRUG ACTIVITY; DRUG DESIGN; DRUG IDENTIFICATION; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; IC 50; OSTEOCLAST; OSTEOPOROSIS; PAGET BONE DISEASE; PRIORITY JOURNAL; REVIEW; RING CLOSING METATHESIS; STRUCTURE ACTIVITY RELATION; ARTICLE; BINDING SITE; CELL STRAIN HL 60; CHEMICAL STRUCTURE; CHEMISTRY; DRUG POTENTIATION; METABOLISM; PROTEIN CONFORMATION; SYNTHESIS;

BINDING SITES; CALCITRIOL; HL-60 CELLS; HUMANS; LACTONES; MOLECULAR STRUCTURE; PROTEIN CONFORMATION; RECEPTORS, CALCITRIOL; VITAMIN D;

EID: 33749672595 PISSN: 14394227 EISSN: 14397633 Source Type: Journal
DOI: 10.1002/cbic.200600054 Document Type: Review

Times cited : (33)

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