Molecular determinants of cocaine block of human Ether-á-go-go-related gene potassium channels

Journal of Pharmacology and Experimental Therapeutics

Volumn 317, Issue 2, 2006, Pages 865-874

  Guo, Jun ^a   Gang, Hongying ^a   Zhang, Shetuan ^a  

^a UNIVERSITY OF MANITOBA   (Canada)

Author keywords

[No Author keywords available]

Indexed keywords

COCAINE; MUTANT PROTEIN; PHENYLALANINE; POTASSIUM CHANNEL HERG; THREONINE; TYROSINE;

ARTICLE; CELL STRAIN HEK293; CONTROLLED STUDY; CORRELATION ANALYSIS; EMBRYO; GENE MUTATION; GENE TARGETING; HUMAN; HUMAN CELL; HYDROPHOBICITY; MOLECULAR GENETICS; PATCH CLAMP; PRIORITY JOURNAL; SITE DIRECTED MUTAGENESIS; WILD TYPE;

BINDING, COMPETITIVE; CELL LINE; CISAPRIDE; COCAINE; DOSE-RESPONSE RELATIONSHIP, DRUG; ETHER-A-GO-GO POTASSIUM CHANNELS; HUMANS; ION CHANNEL GATING; MUTAGENESIS, SITE-DIRECTED; PATCH-CLAMP TECHNIQUES; POTASSIUM; POTASSIUM CHANNEL BLOCKERS;

EID: 33645880127     PISSN: 00223565     EISSN: 15210103     Source Type: Journal    
DOI: 10.1124/jpet.105.098103     Document Type: Article

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