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Bioorganic and Medicinal Chemistry

Volumn 14, Issue 9, 2006, Pages 2978-2984

Design, synthesis, and anti-integrase activity of catechol-DKA hybrids

(5) Maurin, Cédric a Bailly, Fabrice a Mbemba, Gladys b Mouscadet, Jean François b Cotelle, Philippe a

a UNIV LILLE (France)

b UNIVERSITÉ PARIS SACLAY (France)

Author keywords

Antiviral; Catechols; DKA; HIV 1 integrase inhibitors

Indexed keywords

2 HYDROXY 4 OXO 4 (2 HYDROXYPHENYL)BUTENOIC ACID; 2 HYDROXY 4 OXO 4 (3,4 DIHYDROXYPHENYL)BUTENOIC ACID; 2 HYDROXY 4 OXO 4 (3,4 DIMETHOXYPHENYL)BUTENOIC ACID; 2 HYDROXY 4 OXO 4 (6,7 DIHYDROXYNAPHTHYL)BUTENOIC ACID; CATECHOL; DIKETOACID DERIVATIVE; INTEGRASE INHIBITOR; L 708906; METAL ION; METHYL 2 HYDROXY 4 OXO 4 (3,4 DIHYDROXYPHENYL)BUTENOATE; METHYL 2 HYDROXY 4 OXO 4 (6,7 DIHYDROXYNAPHTHYL)BUTENOATE; OXOACID; UNCLASSIFIED DRUG;

ANTIVIRAL ACTIVITY; ARTICLE; DRUG DESIGN; DRUG INHIBITION; DRUG SYNTHESIS; IC 50;

ACIDS; CATALYSIS; CATECHOLS; DIMERIZATION; DRUG DESIGN; HIV INTEGRASE; HIV INTEGRASE INHIBITORS; HIV-1; MOLECULAR STRUCTURE; STRUCTURE-ACTIVITY RELATIONSHIP;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 33644970103 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/j.bmc.2005.12.039 Document Type: Article

Times cited : (22)

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