An inhibitor of TRPV1 channels isolated from funnel web spider venom

Biochemistry

Volumn 44, Issue 47, 2005, Pages 15544-15549

  Kitaguchi, Tetsuya ^a   Swartz, Kenton J ^a,b  

^a NATIONAL INSTITUTE OF NEUROLOGICAL DISORDERS AND STROKE   (United States)

^b NATIONAL INSTITUTES OF HEALTH   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CELL MEMBRANES; ENZYME INHIBITION; MUTAGENESIS; NEUROLOGY; POSITIVE IONS;

CATION CHANNELS; PORE-BLOCKING MECHANISM; WEB SPIDER VENOM;

TOXIC MATERIALS;

ACYLPOLYAMINE TOXIN; AG 489; AG 505; CATION CHANNEL; POLYAMINE; PROTEIN TRPV1 INHIBITOR; SPIDER VENOM; UNCLASSIFIED DRUG; VANILLOID RECEPTOR 1; VANILLOID RECEPTOR 1 INHIBITOR;

AGELENOPSIS APERTA; ANIMAL CELL; ARTICLE; BINDING AFFINITY; DRUG PURIFICATION; GENE MUTATION; INHIBITION KINETICS; MUTAGENESIS; NOCICEPTIVE STIMULATION; NONHUMAN; PRIORITY JOURNAL; PROTEIN ANALYSIS; PROTEIN PURIFICATION; RECEPTOR BLOCKING; REVERSED PHASE HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; SCANNING MUTAGENESIS; SENSORY NERVE; SPIDER; VOLTAGE CLAMP;

ANIMALS; CHEMICAL FRACTIONATION; ELECTROPHYSIOLOGY; MODELS, MOLECULAR; MUTAGENESIS; OOCYTES; POLYAMINES; RATS; SPIDER VENOMS; TRANSFECTION; TRPV CATION CHANNELS; XENOPUS;

AGELENOPSIS APERTA; ANIMALIA; ARANEAE; DIPLURIDAE;

EID: 28244475780     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi051494l     Document Type: Article

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