SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 16, 2002, Pages 2205-2208

N-aryl-prolyl-dipeptides as potent antagonists of VLA-4

(13) Kamenecka, Theodore M a Lanza, Jr , Thomas a De Laszlo, Stephen E a Li, Bing a McCauley, Ermengilda D a Van Riper, Gail a Egger, Linda A a Kidambi, Usha a Mumford, Richard A a Tong, Sharon a MacCoss, Malcolm a Schmidt, John A a Hagmann, William K a

a MERCK RESEARCH LABORATORIES (United States)

Author keywords

[No Author keywords available]

Indexed keywords

PEPTIDE DERIVATIVE; UNCLASSIFIED DRUG; VERY LATE ACTIVATION ANTIGEN 4 ANATGONIST; DIPEPTIDE; VERY LATE ACTIVATION ANTIGEN 4;

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DRUG BIOAVAILABILITY; DRUG BLOOD LEVEL; DRUG CLEARANCE; DRUG DESIGN; DRUG HALF LIFE; DRUG POTENCY; DRUG SYNTHESIS; NONHUMAN; RAT; ANIMAL; BLOOD; CHEMICAL STRUCTURE; DRUG ANTAGONISM; HALF LIFE TIME; METABOLIC CLEARANCE RATE; SPRAGUE DAWLEY RAT; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

ANIMALS; DIPEPTIDES; HALF-LIFE; INTEGRIN ALPHA4BETA1; METABOLIC CLEARANCE RATE; MOLECULAR STRUCTURE; RATS; RATS, SPRAGUE-DAWLEY; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 18444393997 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(02)00356-6 Document Type: Article

Times cited : (16)

References (27)

1
- 0025195762
- (1990) Immunol. Rev. , vol.114 , pp. 45
- Hemler, M.E.¹ Elices, M.J.² Parker, C.³ Takada, Y.⁴

2
- 0001434504
- (1999) Curr. Opin. Anti-inflam. Immunol. , vol.1 , pp. 15
- Elices, M.J.¹

3
- 77956790327
- (1999) Annu. Rep. Med. Chem. , vol.34 , pp. 179
- Adams, S.P.¹ Lobb, R.R.²

4
- 0001182073
- (2000) Idrugs , vol.3 , pp. 788
- Porter, J.R.¹

5
- 0001569451
- (2001) Prog. Respir. Res. , vol.31 , pp. 302
- Adams, S.P.¹ Lobb, R.R.²

6
- 0034678645
- (2000) Bioorg. Med. Chem. Lett. , vol.10 , pp. 725
- Chen, L.¹ Tilley, J.W.² Huang, T.N.³ Miklowski, D.⁴ Trilles, R.⁵ Guthrie, R.W.⁶ Luk, K.⁷ Hanglow, A.⁸ Rowan, K.⁹ Schwinge, V.¹⁰ Wolitzky, B.¹¹

7
- 0034678785
- (2000) Bioorg. Med. Chem. Lett. , vol.10 , pp. 729
- Chen, L.¹ Tilley, J.W.² Guthrie, R.W.³ Mennona, F.⁴ Huang, T.-N.⁵ Kaplan, G.⁶ Trilles, R.⁷ Miklowski, D.⁸ Huby, N.⁹ Schwinge, V.¹⁰ Wolitzky, B.¹¹ Rowen, K.¹²

8
- 0034608632
- (2000) Bioorg. Med. Chem. Lett. , vol.10 , pp. 1163
- Tilley, J.W.¹ Kaplan, G.² Fotouhi, N.³ Wolitzky, B.⁴ Rowan, K.⁵

9
- 0034608594
- (2000) Bioorg. Med. Chem. Lett. , vol.10 , pp. 1167
- Fotouhi, N.¹ Joshi, P.² Tilley, J.W.³ Rowan, K.⁴ Schwinge, V.⁵ Wolitzky, B.⁶

10
- 0034897707
- (2001) Bioorg. Med. Chem. Lett. , vol.9 , pp. 2195
- Astles, P.C.¹ Harris, N.V.² Morley, A.D.³

11
- 0003450707
- New Orleans, LA, American Chemical Society: Washington, DC, 1999, MEDI 61.
- Abstracts of Papers, Part 1, 218th National Meeting of the American Chemical Society
- Furth, P.S.¹ Chiang, S.L.² Sircar, I.³ Griffith, R.C.⁴ Nowlin, D.⁵ Gorscan, F.S.⁶ Mah, J.⁷ Lazarides, E.⁸

12
- 33846403293
- 220th National Meeting of the American Chemical Society, Washington, DC, American Chemical Society: Washington, DC, 2000, MEDI 133.
- Abstracts of Papers, Part 2
- Semko, C.M.¹ Dressen, D.B.² Grant, F.S.³ Konradi, A.W.⁴ Pleiss, M.A.⁵ Thorsett, E.D.⁶ Freedman, S.B.⁷ Holsztynska, E.J.⁸ Quinn, K.P.⁹ Yednock, T.¹⁰

14
- 0005827450
- Unpublished results
- De Laszlo, S.E.¹ Gutteridge, C.²

16
- 4243825627
- PCT Application WO98/53817A1, 1998
- (1998) Chem. Abstr. , vol.130
- Durette, P.L.¹ Hagmann, W.K.² MacCoss, M.³ Mills, S.⁴ Mumford, R.⁵

17
- 0005825206
- note

18
- 0030575791
- (1996) Tetrahedron: Asymmetry , vol.7 , pp. 3075
- Ma, D.¹ Yao, J.²

19
- 0032501446
- (1998) J. Am. Chem. Soc. , vol.120 , pp. 12459
- Ma, D.¹ Zhang, Y.² Yao, J.³ Wu, S.⁴ Tao, F.⁵

20
- 0028997484
- (1995) J. Org. Chem. , vol.60 , pp. 3561
- Carpino, L.A.¹ El-Faham, A.² Albericio, F.³

21
- 0001012518
- (1996) J. Org. Chem. , vol.61 , pp. 2460
- Carpino, L.A.¹ Ionescu, D.² El-Faham, A.³

22
- 33748621833
- (1995) Angew. Chem., Int. Ed. Engl. , vol.34 , pp. 1348
- Guram, S.¹ Rennels, R.A.² Buchwald, S.L.³

23
- 0034712156
- (2000) J. Org. Chem. , vol.65 , pp. 1158
- Wolfe, J.P.¹ Tomori, H.² Sadighi, J.P.³ Yin, J.⁴ Buchwald, S.L.⁵

24
- 0035917354
- (2001) J. Org. Chem. , vol.66 , pp. 2560
- Ali, M.H.¹ Buchwald, S.L.²

25
- 0005784752
- note

26
- 0005788941
- note

27
- 18244399393
- (2002) Bioorg. Med. Chem. Lett. , vol.12 , pp. 637
- Kopka, I.E.¹ Young, D.N.² Lin, L.S.³ Mumford, R.A.⁴ Magriotis, P.A.⁵ MacCross, M.⁶ Mills, S.G.⁷ Van Ripper, G.⁸ McCauley, E.⁹ Egger, L.E.¹⁰ Kidambi, U.¹¹ Schmidt, J.A.¹² Lyons, K.¹³ Stearns, R.¹⁴ Vincent, S.¹⁵ Colletti, A.¹⁶ Wang, Z.¹⁷ Tong, S.¹⁸ Wang, J.¹⁹ Owens, K.²⁰ Levorse, D.²¹ Hagmann, W.K.²² more..

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.