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Bioorganic and Medicinal Chemistry

Volumn 9, Issue 8, 2001, Pages 2195-2202

Diamine containing VLA-4 antagonists

(3) Astles, Peter C a Harris, Neil V a Morley, Andrew D a,b

a Aventis Pharmaceuticals (United Kingdom)

b ASTRAZENECA (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

2 BENZYLOXYCARBONYLAMINO 3 [4 [[2 [3 METHOXY 4 [3 (2 TOLYL)UREIDO]PHENYL]ACETYLAMINO]METHYL]PIPERIDIN 1 YL]PROPIONIC ACID; 3 [4 [[2 [3 METHOXY 4 [3 (2 TOLYL)UREIDO]PHENYL]ACETYLAMINO]METHYL]PIPERIDIN 1 YL]BUTYRIC ACID; BETA1 INTEGRIN; BLOCKING AGENT; DIAMINE; FIBRONECTIN; UNCLASSIFIED DRUG; VASCULAR CELL ADHESION MOLECULE 1;

ARTICLE; CELL STRAIN; CONTROLLED STUDY; DERIVATIZATION; DRUG DESIGN; DRUG POTENCY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IC 50; PHARMACOPHORE; STRUCTURE ACTIVITY RELATION;

CELL ADHESION; DIAMINES; DRUG DESIGN; HUMANS; INTEGRIN ALPHA4BETA1; INTEGRINS; RECEPTORS, LYMPHOCYTE HOMING; STRUCTURE-ACTIVITY RELATIONSHIP; TUMOR CELLS, CULTURED;

EID: 0034897707 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/S0968-0896(01)00132-8 Document Type: Article

Times cited : (13)

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