High-throughput X-ray crystallography for drug discovery

Current Opinion in Pharmacology

Volumn 4, Issue 5, 2004, Pages 490-496

  Blundell, Tom L ^a   Patel, S ^b  

^a UNIVERSITY OF CAMBRIDGE   (United Kingdom)

^b ASTEX PHARMACEUTICALS   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

AMPRENAVIR; NELFINAVIR; ZANAMIVIR; LIGAND; PROTEIN;

ARTICLE; BINDING SITE; DRUG DESIGN; DRUG TARGETING; HIGH THROUGHPUT SCREENING; LIGAND BINDING; MOLECULAR WEIGHT; NUCLEAR MAGNETIC RESONANCE; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN STRUCTURE; STRUCTURE ACTIVITY RELATION; X RAY CRYSTALLOGRAPHY; CHEMICAL STRUCTURE; CHEMISTRY; ISOLATION AND PURIFICATION; PHARMACEUTICS; REVIEW;

CRYSTALLOGRAPHY, X-RAY; DRUG DESIGN; LIGANDS; MODELS, MOLECULAR; PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP; TECHNOLOGY, PHARMACEUTICAL;

EID: 15944394229     PISSN: 14714892     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.coph.2004.04.007     Document Type: Review

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