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Volumn 9, Issue 9, 2003, Pages 1959-1962

Potential inhibition of cytochrome P450 3A4 by propofol in human primary hepatocytes

Author keywords

[No Author keywords available]

Indexed keywords

ANESTHETIC AGENT; CYTOCHROME P450; CYTOCHROME P450 3A4; CYTOCHROME P450 3A4 INHIBITOR; CYTOCHROME P450 INHIBITOR; DOPAMINE; EPHEDRINE; FENTANYL; HEMOPROTEIN; ISOENZYME; LIDOCAINE; LIVER ENZYME; PHENOBARBITAL; PROPOFOL; PROTEIN; RANITIDINE; ROCURONIUM; UNCLASSIFIED DRUG; VASOPRESSIN; VECURONIUM; XENOBIOTIC AGENT;

EID: 0141829778     PISSN: 10079327     EISSN: None     Source Type: Journal    
DOI: 10.3748/wjg.v9.i9.1959     Document Type: Article
Times cited : (22)

References (36)
  • 2
    • 0032924934 scopus 로고    scopus 로고
    • Cytochrome P-450 3A4: Regulation and role in drug metabolism
    • Guengerich FP. Cytochrome P-450 3A4: Regulation and role in drug metabolism. Annu Rev Pharmacol Toxicol 1999; 39: 1-17
    • (1999) Annu Rev Pharmacol Toxicol , vol.39 , pp. 1-17
    • Guengerich, F.P.1
  • 3
    • 0036881096 scopus 로고    scopus 로고
    • Cytochrome P450 3A4 and P-glycoprotein mediate the interaction between an oral erythromycin breath test and rifampin
    • Paine MF, Wagner DA, Hoffmaster KA, Watkins PB. Cytochrome P450 3A4 and P-glycoprotein mediate the interaction between an oral erythromycin breath test and rifampin. Clin Pharmacol Ther 2002; 72: 524-535
    • (2002) Clin Pharmacol Ther , vol.72 , pp. 524-535
    • Paine, M.F.1    Wagner, D.A.2    Hoffmaster, K.A.3    Watkins, P.B.4
  • 5
    • 0033836179 scopus 로고    scopus 로고
    • Propofol inhibits renal cytochrome P450 activity and enflurane defluorinatiion in vitro in hamsters
    • Chen TL, Chen TG, Tai YT, Chang HC, Chen RM, Lin CJ, Ueng TH. Propofol inhibits renal cytochrome P450 activity and enflurane defluorinatiion in vitro in hamsters. Can J Anaesth 2000; 47: 680-686
    • (2000) Can J Anaesth , vol.47 , pp. 680-686
    • Chen, T.L.1    Chen, T.G.2    Tai, Y.T.3    Chang, H.C.4    Chen, R.M.5    Lin, C.J.6    Ueng, T.H.7
  • 7
    • 0034964158 scopus 로고    scopus 로고
    • Human hepatocyte culture systems for the in vitro evaluation of cytochrome P450 expression and regulation
    • LeCluyse EL. Human hepatocyte culture systems for the in vitro evaluation of cytochrome P450 expression and regulation. Eur J Pharm Sci 2001; 13: 343-368
    • (2001) Eur J Pharm Sci , vol.13 , pp. 343-368
    • LeCluyse, E.L.1
  • 8
    • 0030824718 scopus 로고    scopus 로고
    • The use of primary hepatocyte cultures for the evaluation of chemoprotective agents
    • Morel F, Langouet S, Maheo K, Guillouzo A. The use of primary hepatocyte cultures for the evaluation of chemoprotective agents. Cell Biol Toxicol 1997; 13: 323-329
    • (1997) Cell Biol Toxicol , vol.13 , pp. 323-329
    • Morel, F.1    Langouet, S.2    Maheo, K.3    Guillouzo, A.4
  • 9
    • 0031877778 scopus 로고    scopus 로고
    • Culture and transfection of mammalian primary hepatocytes and hepatocyte-derived cell lines
    • Liddle C, Goodwin BJ, Tapner M. Culture and transfection of mammalian primary hepatocytes and hepatocyte-derived cell lines. J Gastroenterol Hepatol 1998; 13: 855-858
    • (1998) J Gastroenterol Hepatol , vol.13 , pp. 855-858
    • Liddle, C.1    Goodwin, B.J.2    Tapner, M.3
  • 10
    • 0015162365 scopus 로고
    • Some recent refinements of quantitative histochemical analysis
    • Lowry OH, Passonneau JV. Some recent refinements of quantitative histochemical analysis. Curr Probl Clin Biochem 1971; 3: 63-84
    • (1971) Curr Probl Clin Biochem , vol.3 , pp. 63-84
    • Lowry, O.H.1    Passonneau, J.V.2
  • 11
    • 0033956881 scopus 로고    scopus 로고
    • Lipoxygenase-mediated hydrogen peroxide-dependent N-demethylation of N,N-dimethylaniline and related compounds
    • Hover CG, Kulkarni AP. Lipoxygenase-mediated hydrogen peroxide-dependent N-demethylation of N,N-dimethylaniline and related compounds. Chem Biol Interact 2000; 124: 191-203
    • (2000) Chem Biol Interact , vol.124 , pp. 191-203
    • Hover, C.G.1    Kulkarni, A.P.2
  • 13
    • 0030726508 scopus 로고    scopus 로고
    • Preclinical evaluation of drug-drug interaction potential: Present status of the application of primary human hepatocytes in the evaluation of cytochrome P450 induction
    • Li AP, Maurel P, Gomez-Lechon MJ, Cheng LC, Jurima-Romet M. Preclinical evaluation of drug-drug interaction potential: Present status of the application of primary human hepatocytes in the evaluation of cytochrome P450 induction. Chem Biol Interact 1997; 107: 5-16
    • (1997) Chem Biol Interact , vol.107 , pp. 5-16
    • Li, A.P.1    Maurel, P.2    Gomez-Lechon, M.J.3    Cheng, L.C.4    Jurima-Romet, M.5
  • 14
    • 0035684268 scopus 로고    scopus 로고
    • Chiral metabolism of propafenone in rat hepatic microsomes treated with two inducers
    • Zhou Q, Yao TW, Zeng S. Chiral metabolism of propafenone in rat hepatic microsomes treated with two inducers. World J Gastroenterol 2001; 7: 830-835
    • (2001) World J Gastroenterol , vol.7 , pp. 830-835
    • Zhou, Q.1    Yao, T.W.2    Zeng, S.3
  • 15
    • 0027489375 scopus 로고
    • Use of human hepatocyte cultures for drug metabolism studies
    • Guillouzo A, Morel F, Fardel O, Meunier B. Use of human hepatocyte cultures for drug metabolism studies. Toxicology 1993; 82: 209-219
    • (1993) Toxicology , vol.82 , pp. 209-219
    • Guillouzo, A.1    Morel, F.2    Fardel, O.3    Meunier, B.4
  • 16
    • 0027349191 scopus 로고
    • Sexually differentiated expression of genes encoding the P4502C cytochromes in rat liver - A model system for studying the action of growth hormone
    • Mode A. Sexually differentiated expression of genes encoding the P4502C cytochromes in rat liver - A model system for studying the action of growth hormone. Reprod Fertil Suppl 1993; 46: 77-86
    • (1993) Reprod Fertil Suppl , vol.46 , pp. 77-86
    • Mode, A.1
  • 17
    • 0036694258 scopus 로고    scopus 로고
    • Pharmacokinetics and electrocardiographic effects of a new controlled-release form of flecainide acetate: Comparison with the standard form and influence of the CYP2D6 polymorphism
    • Tenneze L, TarralE, Ducloux N, Funck-Brentano C. Pharmacokinetics and electrocardiographic effects of a new controlled-release form of flecainide acetate: Comparison with the standard form and influence of the CYP2D6 polymorphism. Clin Pharmacol Ther 2002; 72: 112-122
    • (2002) Clin Pharmacol Ther , vol.72 , pp. 112-122
    • Tenneze, L.1    Tarral, E.2    Ducloux, N.3    Funck-Brentano, C.4
  • 20
    • 0036073564 scopus 로고    scopus 로고
    • Cytochrome P450 phenotyping/genotyping in patients receiving antipsychotics: Useful aid to prescribing?
    • Dahl ML. Cytochrome P450 phenotyping/genotyping in patients receiving antipsychotics: Useful aid to prescribing? Clin Pharmacokinet 2002; 41: 453-470
    • (2002) Clin Pharmacokinet , vol.41 , pp. 453-470
    • Dahl, M.L.1
  • 21
    • 0029028932 scopus 로고
    • Geographical/interracial differences in polymorphic drug oxidation. Current state of knowledge of cytochromes P450 (CYP) 2D6 and 2C19
    • Bertilsson L. Geographical/interracial differences in polymorphic drug oxidation. Current state of knowledge of cytochromes P450 (CYP) 2D6 and 2C19. Clin Pharmacokinet 1995; 29: 192-209
    • (1995) Clin Pharmacokinet , vol.29 , pp. 192-209
    • Bertilsson, L.1
  • 22
    • 0035675195 scopus 로고    scopus 로고
    • Clinical interpretation of pharmacokinetic and pharmacodynamic propofol-opioid interactions
    • Vuyk J. Clinical interpretation of pharmacokinetic and pharmacodynamic propofol-opioid interactions. Acta Anaesthesiol Belg 2001; 52: 445-451
    • (2001) Acta Anaesthesiol Belg , vol.52 , pp. 445-451
    • Vuyk, J.1
  • 23
    • 0035906912 scopus 로고    scopus 로고
    • Propofol-induced cytochrome P450 inhibition: An in vitro and in vivo study in rats
    • Gemayel J, Geloen A, Mion F. Propofol-induced cytochrome P450 inhibition: An in vitro and in vivo study in rats. Life Sci 2001; 68: 2957-2965
    • (2001) Life Sci , vol.68 , pp. 2957-2965
    • Gemayel, J.1    Geloen, A.2    Mion, F.3
  • 24
    • 0032942249 scopus 로고    scopus 로고
    • The effect of oxygen on propofol-induced inhibition of microsomal cytochrome P450 3A4
    • Miller E, Park GR. The effect of oxygen on propofol-induced inhibition of microsomal cytochrome P450 3A4. Anaesthesia 1999; 54: 320-322
    • (1999) Anaesthesia , vol.54 , pp. 320-322
    • Miller, E.1    Park, G.R.2
  • 25
    • 0031669251 scopus 로고    scopus 로고
    • Effects of propofol on human hepatic microsomal cytochrome P450 activities
    • McKillop D, Wild MJ, Butters CJ, Simcock C. Effects of propofol on human hepatic microsomal cytochrome P450 activities. Xenobiotica 1998; 28: 845-853
    • (1998) Xenobiotica , vol.28 , pp. 845-853
    • McKillop, D.1    Wild, M.J.2    Butters, C.J.3    Simcock, C.4
  • 26
    • 0028874616 scopus 로고
    • Difference between in vivo and in vitro effects of propofol on defluorination and metabolic activities of hamster hepatic cytochrome P450-dependent mono-oxygenases
    • Chen TL, Wang MJ, Huang CH, Liu CC, Ueng TH. Difference between in vivo and in vitro effects of propofol on defluorination and metabolic activities of hamster hepatic cytochrome P450-dependent mono-oxygenases. Br J Anaesth 1995; 75: 462-466
    • (1995) Br J Anaesth , vol.75 , pp. 462-466
    • Chen, T.L.1    Wang, M.J.2    Huang, C.H.3    Liu, C.C.4    Ueng, T.H.5
  • 27
    • 0032417493 scopus 로고    scopus 로고
    • Molecular basis of P450 inhibition and activation: Implications for drug development and drug therapy
    • Szklarz GD, Halpert JR. Molecular basis of P450 inhibition and activation: Implications for drug development and drug therapy. Drug Metab Dispos 1998; 26: 1179-1184
    • (1998) Drug Metab Dispos , vol.26 , pp. 1179-1184
    • Szklarz, G.D.1    Halpert, J.R.2
  • 28
    • 0036713019 scopus 로고    scopus 로고
    • Bispectral index in patients with target-controlled or manually-controlled infusion of propofol
    • Lehmann A, Boldt J, Thaler E, Piper S, Weisse U. Bispectral index in patients with target-controlled or manually-controlled infusion of propofol. Anesth Analg 2002; 95: 639-644
    • (2002) Anesth Analg , vol.95 , pp. 639-644
    • Lehmann, A.1    Boldt, J.2    Thaler, E.3    Piper, S.4    Weisse, U.5
  • 29
    • 0036724080 scopus 로고    scopus 로고
    • Target-controlled infusion of propofol induction with or without plasma concentration constraint in high-risk adult patients under-going cardiac surgery
    • Macquaire V, Cantraine F, Schmartz D, Coussaert E, Barvais L. Target-controlled infusion of propofol induction with or without plasma concentration constraint in high-risk adult patients under-going cardiac surgery. Acta Anaesthesiol Scand 2002; 46: 1010-1016
    • (2002) Acta Anaesthesiol Scand , vol.46 , pp. 1010-1016
    • Macquaire, V.1    Cantraine, F.2    Schmartz, D.3    Coussaert, E.4    Barvais, L.5
  • 30
    • 0036192257 scopus 로고    scopus 로고
    • Propofol effective concentration 50 and its relationship to bispectral index
    • Irwin MG, Hui TW, Milne SE, Kenny GN. Propofol effective concentration 50 and its relationship to bispectral index. Anaesthesia 2002; 57: 242-248
    • (2002) Anaesthesia , vol.57 , pp. 242-248
    • Irwin, M.G.1    Hui, T.W.2    Milne, S.E.3    Kenny, G.N.4
  • 31
    • 0030444880 scopus 로고    scopus 로고
    • Effect of diltiazem on midazolam and alfentanil disposition in patients undergoing coronary artery bypass grafting
    • Ahonen J, Olkkola KT, Salmenpera M, Hynynen M, Neuvonen PJ. Effect of diltiazem on midazolam and alfentanil disposition in patients undergoing coronary artery bypass grafting. Anesthesiology 1996; 85: 1246-1252
    • (1996) Anesthesiology , vol.85 , pp. 1246-1252
    • Ahonen, J.1    Olkkola, K.T.2    Salmenpera, M.3    Hynynen, M.4    Neuvonen, P.J.5
  • 32
    • 0033062463 scopus 로고    scopus 로고
    • Fentanyl inhibits metabolism of midazolam: Competitive inhibition of CYP3A4 in vitro
    • Oda Y, Mizutani K, Hase I, Nakamoto T, Hamaoka N, Asada A. Fentanyl inhibits metabolism of midazolam: Competitive inhibition of CYP3A4 in vitro. Br J Anaesth 1999; 82: 900-903
    • (1999) Br J Anaesth , vol.82 , pp. 900-903
    • Oda, Y.1    Mizutani, K.2    Hase, I.3    Nakamoto, T.4    Hamaoka, T.5    Asada, A.6
  • 33
    • 0030925252 scopus 로고    scopus 로고
    • In vivo induction and in vitro inhibition of hepatic cytochrome P450 activity by the benzodiazepine anticonvulsants clonazepam and diazepam
    • Nims RW, Prough RA, Jones CR, Stockus DL, Dragnev KH, Thomas PE, Lubet RA. In vivo induction and in vitro inhibition of hepatic cytochrome P450 activity by the benzodiazepine anticonvulsants clonazepam and diazepam. Drug Metab Dispos 1997; 25: 750-756
    • (1997) Drug Metab Dispos , vol.25 , pp. 750-756
    • Nims, R.W.1    Prough, R.A.2    Jones, C.R.3    Stockus, D.L.4    Dragnev, K.H.5    Thomas, P.E.6    Lubet, R.A.7
  • 34
    • 0031566987 scopus 로고    scopus 로고
    • Interaction of methadone with substrates of human hepatic cytochrome P450 3A4
    • Iribarne C, Dreano Y, Bardou LG, Menez JF, Berthou F. Interaction of methadone with substrates of human hepatic cytochrome P450 3A4. Toxicology 1997; 117: 13-23
    • (1997) Toxicology , vol.117 , pp. 13-23
    • Iribarne, C.1    Dreano, Y.2    Bardou, L.G.3    Menez, J.F.4    Berthou, F.5
  • 36
    • 0034782509 scopus 로고    scopus 로고
    • Coordinate regulation of xenobiotic and bile acid homeostasis by pregnane X receptor
    • Staudinger J, Liu Y, Madan A, Habaeebu S, Klaassen CD. Coordinate regulation of xenobiotic and bile acid homeostasis by pregnane X receptor. Drug Metab Dispos 2001; 29: 1467-1472
    • (2001) Drug Metab Dispos , vol.29 , pp. 1467-1472
    • Staudinger, J.1    Liu, Y.2    Madan, A.3    Habaeebu, S.4    Klaassen, C.D.5


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