Molecular basis of p450 inhibition and activation. Implications for drug development and drug therapy

Drug Metabolism and Disposition

Volumn 26, Issue 12, 1998, Pages 1179-1184

  Szklarz, Grazyna D ^b   Halpert, James R ^a  

^a University of Texas Medical Branch School of Medicine   (United States)

^b WEST VIRGINIA UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CYTOCHROME P450 2B1; CYTOCHROME P450 3A4; CYTOCHROME P450 ISOENZYME; UNCLASSIFIED DRUG;

DRUG METABOLISM; ENZYME INHIBITION; ENZYME SPECIFICITY; ENZYME SUBSTRATE COMPLEX; MICHAELIS MENTEN KINETICS; PRIORITY JOURNAL; REVIEW; SITE DIRECTED MUTAGENESIS;

ANIMALS; CYTOCHROME P-450 ENZYME SYSTEM; DRUG DESIGN; DRUG THERAPY; ENZYME ACTIVATION; ENZYME INHIBITORS; HUMANS;

BACTERIA (MICROORGANISMS);

EID: 0032417493     PISSN: 00909556     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review

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