Rapid desensitization of the serotonin2c receptor system: Effector pathway and agonist dependence

Journal of Pharmacology and Experimental Therapeutics

Volumn 302, Issue 3, 2002, Pages 957-962

  Stout, Brian D ^a   Clarke, William P ^a,b   Berg, Kelly A ^a  

^a UNIVERSITY OF TEXAS HEALTH SCIENCE CENTER AT SAN ANTONIO   (United States)

^b Mays Cancer Center at UT Health San Antonio   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

(3 CHLOROPHENYL)PIPERAZINE; 1 (3 TRIFLUOROMETHYLPHENYL)PIPERAZINE; ARACHIDONIC ACID; BUFOTENINE; INOSITOL; INOSITOL PHOSPHATE; LYSERGIDE; PHOSPHOLIPASE A2; PHOSPHOLIPASE C; QUIPAZINE; SEROTONIN; SEROTONIN 2C AGONIST; SEROTONIN 2C RECEPTOR;

ANIMAL CELL; ARACHIDONIC ACID METABOLISM; ARTICLE; CELL KINETICS; CHO CELL; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG MECHANISM; DRUG RECEPTOR BINDING; EFFECTOR CELL; ENZYME METABOLISM; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BINDING; RECEPTOR DOWN REGULATION; RECEPTOR OCCUPANCY; REGULATORY MECHANISM; SENSITIVITY ANALYSIS; SEROTONIN RELEASE; SIGNAL TRANSDUCTION;

ALGORITHMS; ANIMALS; CHO CELLS; CRICETINAE; KINETICS; PHOSPHATIDYLINOSITOLS; PHOSPHOLIPASE C; PHOSPHOLIPASES A; RECEPTOR, SEROTONIN, 5-HT2C; RECEPTORS, SEROTONIN; SEROTONIN; SEROTONIN AGONISTS; SEROTONIN ANTAGONISTS; SIGNAL TRANSDUCTION;

EID: 0036720639     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: 10.1124/jpet.302.3.957     Document Type: Article

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