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Biochemistry

Volumn 40, Issue 24, 2001, Pages 7084-7091

Structural determinants for potent, selective dual site inhibition of human pp60c-src by 4-anilinoquinazolines

(4) Tian, G a,b Cory, M a Smith, A A a Blaine Knight, W a

a GLAXOSMITHKLINE (United States)

b ASTRAZENECA (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ADENOSINETRIPHOSPHATE; BINDING ENERGY; ENZYME KINETICS; PROTEINS; SUBSTRATES;

CARBOCYCLIC RING;

BIOCHEMISTRY;

4 ANILINOQUINAZOLINE; ADENOSINE TRIPHOSPHATE; PROTEIN KINASE INHIBITOR; PROTEIN KINASE P60; PROTEIN TYROSINE KINASE; QUINAZOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; BINDING SITE; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; ENZYME INHIBITION; ENZYME KINETICS; ENZYME MODIFICATION; ENZYME PURIFICATION; ENZYME STRUCTURE; HUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; STRUCTURE ANALYSIS;

EID: 0035912929 PISSN: 00062960 EISSN: None Source Type: Journal
DOI: 10.1021/bi0100586 Document Type: Article

Times cited : (37)

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