Modulation of native and recombinant GABAA receptors by endogenous and synthetic neuroactive steroids

Brain Research Reviews

Volumn 37, Issue 1-3, 2001, Pages 68-80

  Lambert, Jeremy J ^a   Belelli, Delia ^a   Harney, Sarah C ^a   Peters, John A ^a   Frenguelli, Bruno G ^a  

^a UNIVERSITY OF DUNDEE   (United Kingdom)

Author keywords

GABA; GABAA receptor; Neuroactive steroids; Transmitter gated ion channel

Indexed keywords

21 CHLORO 3ALPHA HYDROXY 2BETA MORPHOLINO 5ALPHA PREGNAN 20 ONE METHANESULFONATE; 21 CHLORO 3ALPHA HYDROXY 2BETA(4 MORPHOLINYL) 5ALPHA PREGNAN 20 ONE; 2BETA (2,2 DIMETHYLMORPHOLINO) 3ALPHA HYDROXY 5ALPHA PREGNANE 11,20 DIONE; 3ALPHA HYDROXY 2BETA(2,2 DIMETHYLMORPHOLIN 4 YL) 5ALPHA PREGNANE 11,20 DIONE; 3ALPHA HYDROXY 5ALPHA PREGNAN 20 ONE; 3ALPHA,5ALPHA TETRAHYDRODEOXYCORTICOSTERONE; 4 AMINOBUTYRIC ACID A RECEPTOR; ALFAXALONE; ALTHESIN; AMPA RECEPTOR; ANDROSTERONE; BENZODIAZEPINE; BETAXALONE; ELTANOLONE; ESTRADIOL; ESTRONE; GANAXOLONE; GLYCINE RECEPTOR; KAINIC ACID RECEPTOR; METHYLTESTOSTERONE; MINAXOLONE; N METHYL DEXTRO ASPARTIC ACID RECEPTOR; NANDROLONE; NEUROSTEROID; NICOTINIC RECEPTOR; OXYTOCIN; PREGNANEDIOL; RECEPTOR SUBUNIT; RECOMBINANT RECEPTOR; SEROTONIN 3 RECEPTOR; STANOZOLOL; UNCLASSIFIED DRUG; UNINDEXED DRUG;

ALLOSTERISM; ANALGESIA; ANESTHESIA; ANTICONVULSANT ACTIVITY; BRAIN REGION; CLINICAL TRIAL; CONFERENCE PAPER; DRUG EFFECT; DRUG POTENCY; DRUG SELECTIVITY; ENDOCRINE GLAND; EPILEPSY; GABAERGIC SYSTEM; GLIA CELL; HUMAN; NERVE CELL; NEUROMODULATION; NONHUMAN; PARACRINE SIGNALING; PHOSPHORYLATION; PRIORITY JOURNAL; PROTEIN LIPID INTERACTION; PROTEIN TARGETING; SEDATION; STEROIDOGENESIS; SYNAPTIC INHIBITION; TRANQUILIZING ACTIVITY;

ANIMALS; CENTRAL NERVOUS SYSTEM; HUMANS; ION CHANNEL GATING; MODELS, MOLECULAR; NEURAL INHIBITION; RECEPTORS, GABA-A; RECOMBINANT PROTEINS; STEROIDS; SYNAPTIC TRANSMISSION;

EID: 0035660135     PISSN: 01650173     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0165-0173(01)00124-2     Document Type: Review

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