Design, synthesis, and evaluation of peptides with estrogen-like activity

Biopolymers - Peptide Science Section

Volumn 76, Issue 5, 2004, Pages 404-420

  Kasher, Roni ^a   Gayer, Batya ^a   Kulik, Tikva ^a   Somjen, Dalia ^b   Venkatesh, Natarajan ^a   Fridkin, Mati ^a   Katchalski Katzir, Ephraim ^a   Kohen, Fortune ^a  

^a WEIZMANN INSTITUTE OF SCIENCE   (Israel)

^b TEL AVIV UNIVERSITY   (Israel)

Author keywords

Estrogen receptor alpha; Estrogen receptor beta; Estrogen mimetic peptides; Monoclonal antiestradiol antibody

Indexed keywords

DISEASE CONTROL; DRUG PRODUCTS; MONOCLONAL ANTIBODIES; SYNTHESIS (CHEMICAL); TISSUE; TUMORS;

BREAST CANCER; ESTROGENIC DRUGS; ESTROGENS; PEPTIDES;

PROTEINS;

ESTRADIOL; ESTROGEN MIMETIC PEPTIDE 1; ESTROGEN MIMETIC PEPTIDE 2; ESTROGEN RECEPTOR; HEPTAPEPTIDE; LIGAND; MONOCLONAL ANTIBODY; PEPTIDE LIBRARY; SELECTIVE ESTROGEN RECEPTOR MODULATOR; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ANTIGEN BINDING; ARTICLE; BINDING AFFINITY; BREAST CANCER; CONTROLLED STUDY; DNA SYNTHESIS; DRUG BINDING; DRUG DESIGN; DRUG INHIBITION; DRUG SCREENING; DRUG SELECTIVITY; DRUG SYNTHESIS; ESTROGEN ACTIVITY; FEMALE; HORMONE DEPENDENCE; IC 50; LIGAND BINDING; MOUSE; NONHUMAN; OSTEOPOROSIS; PEPTIDE SYNTHESIS; PHAGE DISPLAY; RAT; RECEPTOR BINDING; RISK FACTOR;

ALANINE; AMINO ACID SEQUENCE; ANTIBODIES, MONOCLONAL; DNA REPLICATION; DRUG DESIGN; ESTROGENS; MOLECULAR SEQUENCE DATA; PEPTIDES; PROTEIN ENGINEERING; RECEPTORS, ESTROGEN;

EID: 9144232273     PISSN: 00063525     EISSN: None     Source Type: Journal    
DOI: 10.1002/bip.20133     Document Type: Article

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