메뉴 건너뛰기




Volumn 2, Issue 4, 2000, Pages 318-329

Solid-phase synthesis of tetrasubstituted pyrazoles, novel ligands for the estrogen receptor

Author keywords

[No Author keywords available]

Indexed keywords

ESTROGEN RECEPTOR; LIGAND; PYRAZOLE DERIVATIVE;

EID: 0034219844     PISSN: 15204766     EISSN: None     Source Type: Journal    
DOI: 10.1021/cc0000040     Document Type: Article
Times cited : (88)

References (20)
  • 1
    • 0033156688 scopus 로고    scopus 로고
    • Comprehensive survey of combinatorial library synthesis
    • Dolle, R. E.; Nelson, K. H. J. Comprehensive Survey of Combinatorial Library Synthesis. J. Comb. Chem. 1999, 1, 235-282.
    • (1999) J. Comb. Chem. , vol.1 , pp. 235-282
    • Dolle, R.E.1    Nelson, K.H.J.2
  • 2
    • 0031888317 scopus 로고    scopus 로고
    • Selective estrogen receptor modulators (SERMS)
    • Grese, T. A.; Dodge, J. A. Selective Estrogen Receptor Modulators (SERMS) [Review]. Curr. Pharm. Des. 1998, 4, 71-92.
    • (1998) Curr. Pharm. Des. , vol.4 , pp. 71-92
    • Grese, T.A.1    Dodge, J.A.2
  • 5
    • 0030062225 scopus 로고    scopus 로고
    • Synthesis of tetrasubstituted ethylenes on solid support via resin capture
    • Brown, D. S.; Armstrong, R. W. Synthesis of tetrasubstituted ethylenes on solid support via resin capture. J. Am. Chem. Soc. 1996, 118, 6331-6332.
    • (1996) J. Am. Chem. Soc. , vol.118 , pp. 6331-6332
    • Brown, D.S.1    Armstrong, R.W.2
  • 6
    • 0033117680 scopus 로고    scopus 로고
    • Novel structural templates for estrogenreceptor ligands and prospects for combinatorial synthesis of estrogens
    • Fink, B. E.; Mortensen, D. S.; Stauffer, S. R.; Aron, Z. D.; Katzenellenbogen, J. A. Novel structural templates for estrogenreceptor ligands and prospects for combinatorial synthesis of estrogens. Chem. Biol. 1999, 6, 205-219.
    • (1999) Chem. Biol. , vol.6 , pp. 205-219
    • Fink, B.E.1    Mortensen, D.S.2    Stauffer, S.R.3    Aron, Z.D.4    Katzenellenbogen, J.A.5
  • 7
    • 0004752110 scopus 로고    scopus 로고
    • Novel ligands that function as selective estrogens or antiestrogens for estrogen receptor-α or estrogen receptor-β
    • Sun, J.; Meyers, M. J.; Fink, B. E.; Rajendran, R.; Katzenellenbogen, J. A.; Katzenellenbogen, B. S. Novel ligands that function as selective estrogens or antiestrogens for estrogen receptor-α or estrogen receptor-β. Endocrinology 1999, 140, 800-804.
    • (1999) Endocrinology , vol.140 , pp. 800-804
    • Sun, J.1    Meyers, M.J.2    Fink, B.E.3    Rajendran, R.4    Katzenellenbogen, J.A.5    Katzenellenbogen, B.S.6
  • 8
    • 0032403545 scopus 로고    scopus 로고
    • ER beta: A novel estrogen receptor offers the potential for new drug development
    • Nilsson, S.; Kuiper, G.; Gustafsson, J. A. ER beta: a novel estrogen receptor offers the potential for new drug development [Review]. Trends Endocrinol. Metab. 1998, 9, 387-395.
    • (1998) Trends Endocrinol. Metab. , vol.9 , pp. 387-395
    • Nilsson, S.1    Kuiper, G.2    Gustafsson, J.A.3
  • 9
    • 0030061466 scopus 로고    scopus 로고
    • Solid support synthesis of highly functionalized pyrazoles and isoxazoles; scaffolds for molecular diversity
    • Marzinik, A. L.; Felder, E. R. Solid support synthesis of highly functionalized pyrazoles and isoxazoles; scaffolds for molecular diversity. Tetrahedron Lett. 1996, 37, 1003-1006.
    • (1996) Tetrahedron Lett. , vol.37 , pp. 1003-1006
    • Marzinik, A.L.1    Felder, E.R.2
  • 10
    • 0001266786 scopus 로고    scopus 로고
    • Key intermediates in combinatorial chemistry: Access to various heterocycles from α,β-unsaturated ketones on the solid phase
    • Marzinzik, A. L.; Felder, E. R. Key intermediates in combinatorial chemistry: access to various heterocycles from α,β-unsaturated ketones on the solid phase. J. Org. Chem. 1998, 63, 723-727.
    • (1998) J. Org. Chem. , vol.63 , pp. 723-727
    • Marzinzik, A.L.1    Felder, E.R.2
  • 11
  • 12
    • 0032580403 scopus 로고    scopus 로고
    • Solid-phase synthesis of 5-aminopyrazoles and derivatives
    • Wilson, R. D.; Watson, S. P.; Richards, S. A. Solid-phase synthesis of 5-aminopyrazoles and derivatives. Tetrahedron Lett. 1998, 39, 2827-2830.
    • (1998) Tetrahedron Lett. , vol.39 , pp. 2827-2830
    • Wilson, R.D.1    Watson, S.P.2    Richards, S.A.3
  • 13
    • 0029060771 scopus 로고
    • Solid-phase synthesis of lavendustin analogues
    • Green, J. Solid-Phase synthesis of lavendustin analogues. J. Org. Chem. 1995, 60, 4287-4290.
    • (1995) J. Org. Chem. , vol.60 , pp. 4287-4290
    • Green, J.1
  • 14
    • 0029128552 scopus 로고
    • An expedient and high-yielding method for the solid-phase synthesis of diverse 1,4-benzodiazepine-2,5-diones
    • Boojamra, C. G.; Burow, K. M.; Ellman, J. A. An Expedient and High-Yielding Method for the Solid-Phase Synthesis of Diverse 1,4-Benzodiazepine-2,5-Diones. J. Org. Chem. 1995, 60, 5742-5743.
    • (1995) J. Org. Chem. , vol.60 , pp. 5742-5743
    • Boojamra, C.G.1    Burow, K.M.2    Ellman, J.A.3
  • 15
    • 84982386784 scopus 로고
    • Carbonate ion on a polymeric support: Hydrolysis of alkyl halides and cyclic iodocarbonates
    • Cardillo, G.; Orena, M.; Porzi, G.; Sandri, S. Carbonate ion on a polymeric support: hydrolysis of alkyl halides and cyclic iodocarbonates. Synthesis 1981, 793-794.
    • (1981) Synthesis , pp. 793-794
    • Cardillo, G.1    Orena, M.2    Porzi, G.3    Sandri, S.4
  • 16
    • 0002714675 scopus 로고
    • Rapid chromatographic technique for preparative separations with moderate resolution
    • Still, W. C.; Kahn, M.; Mitra, A. Rapid Chromatographic technique for preparative separations with moderate resolution. J. Org. Chem. 1978, 43, 2923-2926.
    • (1978) J. Org. Chem. , vol.43 , pp. 2923-2926
    • Still, W.C.1    Kahn, M.2    Mitra, A.3
  • 17
    • 0015902629 scopus 로고
    • Photoaffinity labels for estrogen binding proteins of rat uterus
    • Katzenellenbogen, J. A.; Johnson, H. J., Jr.; Myers, H. N. Photoaffinity labels for estrogen binding proteins of rat uterus. Biochemistry 1973, 12, 4085-4092.
    • (1973) Biochemistry , vol.12 , pp. 4085-4092
    • Katzenellenbogen, J.A.1    Johnson H.J., Jr.2    Myers, H.N.3
  • 18
  • 19
    • 0030593681 scopus 로고    scopus 로고
    • ERβ: Identification and characterization of a novel human estrogen receptor
    • Mosselman, S.; Polman, J.; Dijkema, R. ERβ: identification and characterization of a novel human estrogen receptor. FEBS 1996, 392, 49-53.
    • (1996) FEBS , vol.392 , pp. 49-53
    • Mosselman, S.1    Polman, J.2    Dijkema, R.3
  • 20
    • 84970546247 scopus 로고
    • The reactivity of p-nitrophenyl esters with surfactants in apolar solvents. VII* substituent effects on the reactivity of 4′-nitrophenyl 4-substituted benzoates in benzene solutions of dodecylammonium propionate and butane-1,4-diamine bis(dodecanoate)
    • O'Connor, C. J.; Lomax, T. D. The reactivity of p-nitrophenyl esters with surfactants in apolar solvents. VII* substituent effects on the reactivity of 4′-nitrophenyl 4-substituted benzoates in benzene solutions of dodecylammonium propionate and butane-1,4-diamine bis(dodecanoate). Aust. J. Chem. 1983, 36, 917-925.
    • (1983) Aust. J. Chem. , vol.36 , pp. 917-925
    • O'Connor, C.J.1    Lomax, T.D.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.