메뉴 건너뛰기




Volumn 39, Issue , 2017, Pages 531-541

Salt effect on solubilization of hydrophobic drugs in block copolymeric micelles and investigation of their in vitro and in vivo oral efficiency

Author keywords

Caco 2 permeability; Cytotoxicity; Drug release; Pharmacokinetics; Scattering; Tetronics

Indexed keywords

COPOLYMER; CURCUMIN; ETHYLENE OXIDE; PROPYLENE OXIDE; QUERCETIN; SODIUM CHLORIDE;

EID: 85019635254     PISSN: 17732247     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.jddst.2017.05.007     Document Type: Article
Times cited : (16)

References (82)
  • 1
    • 84864751544 scopus 로고    scopus 로고
    • Functional block copolymers: nanostructured materials with emerging applications
    • Schacher, F.H., Rupar, P.A., Manners, I., Functional block copolymers: nanostructured materials with emerging applications. Angew. Chem. Int. Ed. 51 (2012), 7898–7921.
    • (2012) Angew. Chem. Int. Ed. , vol.51 , pp. 7898-7921
    • Schacher, F.H.1    Rupar, P.A.2    Manners, I.3
  • 2
    • 84900797097 scopus 로고    scopus 로고
    • Directed self-assembly of block copolymers: a tutorial review of strategies for enabling nanotechnology with soft matter
    • Hu, H., Gopinadhan, M., Osuji, C.O., Directed self-assembly of block copolymers: a tutorial review of strategies for enabling nanotechnology with soft matter. Soft matter 10 (2014), 3867–3889.
    • (2014) Soft matter , vol.10 , pp. 3867-3889
    • Hu, H.1    Gopinadhan, M.2    Osuji, C.O.3
  • 3
    • 0142169280 scopus 로고    scopus 로고
    • Developments in Block Copolymer Science and Technology
    • Wiley Online Library
    • Hamley, I.W., Developments in Block Copolymer Science and Technology. 2004, Wiley Online Library.
    • (2004)
    • Hamley, I.W.1
  • 4
    • 84953449707 scopus 로고    scopus 로고
    • Recent advances in polymeric micelles for anti-cancer drug delivery
    • Biswas, S., Kumari, P., Lakhani, P.M., Ghosh, B., Recent advances in polymeric micelles for anti-cancer drug delivery. Eur. J. Pharm. Sci. 83 (2016), 184–202.
    • (2016) Eur. J. Pharm. Sci. , vol.83 , pp. 184-202
    • Biswas, S.1    Kumari, P.2    Lakhani, P.M.3    Ghosh, B.4
  • 6
    • 0029271147 scopus 로고
    • Poly (ethylene oxide) poly (propylene oxide) poly (ethylene oxide) block copolymer surfactants in aqueous solutions and at interfaces: thermodynamics, structure, dynamics, and modeling
    • Alexandridis, P., Hatton, T.A., Poly (ethylene oxide) poly (propylene oxide) poly (ethylene oxide) block copolymer surfactants in aqueous solutions and at interfaces: thermodynamics, structure, dynamics, and modeling. Colloids Surf. A Physicochem. Eng. Asp. 96 (1995), 1–46.
    • (1995) Colloids Surf. A Physicochem. Eng. Asp. , vol.96 , pp. 1-46
    • Alexandridis, P.1    Hatton, T.A.2
  • 8
    • 34248577169 scopus 로고    scopus 로고
    • Poly (ethylene oxide)–poly (propylene oxide) block copolymer micelles as drug delivery agents: improved hydrosolubility, stability and bioavailability of drugs
    • Chiappetta, D.A., Sosnik, A., Poly (ethylene oxide)–poly (propylene oxide) block copolymer micelles as drug delivery agents: improved hydrosolubility, stability and bioavailability of drugs. Eur. J. Pharm. Biopharm. 66 (2007), 303–317.
    • (2007) Eur. J. Pharm. Biopharm. , vol.66 , pp. 303-317
    • Chiappetta, D.A.1    Sosnik, A.2
  • 10
    • 54549103368 scopus 로고    scopus 로고
    • Self-associative behavior and drug-solubilizing ability of poloxamine (tetronic) block copolymers
    • Gonzalez-Lopez, J., Alvarez-Lorenzo, C., Taboada, P., Sosnik, A., Sandez-Macho, I., Concheiro, A., Self-associative behavior and drug-solubilizing ability of poloxamine (tetronic) block copolymers. Langmuir 24 (2008), 10688–10697.
    • (2008) Langmuir , vol.24 , pp. 10688-10697
    • Gonzalez-Lopez, J.1    Alvarez-Lorenzo, C.2    Taboada, P.3    Sosnik, A.4    Sandez-Macho, I.5    Concheiro, A.6
  • 13
    • 30744476534 scopus 로고    scopus 로고
    • Salt influence upon the structure of aqueous solutions of branched PEO–PPO–PEO copolymers
    • Perreur, C., Habas, J.-P., Lapp, A., Peyrelasse, J., Salt influence upon the structure of aqueous solutions of branched PEO–PPO–PEO copolymers. Polymer 47 (2006), 841–848.
    • (2006) Polymer , vol.47 , pp. 841-848
    • Perreur, C.1    Habas, J.-P.2    Lapp, A.3    Peyrelasse, J.4
  • 17
    • 84872311861 scopus 로고    scopus 로고
    • PEO–PPO based star-block copolymer T904 as pH responsive nanocarriers for quercetin: solubilization and release study
    • Parmar, A.V., Bahadur, A., Kuperkar, K., Bahadur, P., PEO–PPO based star-block copolymer T904 as pH responsive nanocarriers for quercetin: solubilization and release study. Eur. Polym. J. 49 (2013), 12–21.
    • (2013) Eur. Polym. J. , vol.49 , pp. 12-21
    • Parmar, A.V.1    Bahadur, A.2    Kuperkar, K.3    Bahadur, P.4
  • 18
    • 43049176634 scopus 로고    scopus 로고
    • Health effects of quercetin: from antioxidant to nutraceutical
    • Boots, A.W., Haenen, G.R., Bast, A., Health effects of quercetin: from antioxidant to nutraceutical. Eur. J. Pharmacol. 585 (2008), 325–337.
    • (2008) Eur. J. Pharmacol. , vol.585 , pp. 325-337
    • Boots, A.W.1    Haenen, G.R.2    Bast, A.3
  • 19
    • 84866045756 scopus 로고    scopus 로고
    • Life or death: neuroprotective and anticancer effects of quercetin
    • Dajas, F., Life or death: neuroprotective and anticancer effects of quercetin. J. Ethnopharmacol. 143 (2012), 383–396.
    • (2012) J. Ethnopharmacol. , vol.143 , pp. 383-396
    • Dajas, F.1
  • 20
    • 81855164783 scopus 로고    scopus 로고
    • The flavonoid quercetin in disease prevention and therapy: facts and fancies
    • Russo, M., Spagnuolo, C., Tedesco, I., Bilotto, S., Russo, G.L., The flavonoid quercetin in disease prevention and therapy: facts and fancies. Biochem. Pharmacol. 83 (2012), 6–15.
    • (2012) Biochem. Pharmacol. , vol.83 , pp. 6-15
    • Russo, M.1    Spagnuolo, C.2    Tedesco, I.3    Bilotto, S.4    Russo, G.L.5
  • 21
    • 55949117806 scopus 로고    scopus 로고
    • Potential therapeutic effects of curcumin, the anti-inflammatory agent, against neurodegenerative, cardiovascular, pulmonary, metabolic, autoimmune and neoplastic diseases
    • Aggarwal, B.B., Harikumar, K.B., Potential therapeutic effects of curcumin, the anti-inflammatory agent, against neurodegenerative, cardiovascular, pulmonary, metabolic, autoimmune and neoplastic diseases. Int. J. Biochem. Cell Biol. 41 (2009), 40–59.
    • (2009) Int. J. Biochem. Cell Biol. , vol.41 , pp. 40-59
    • Aggarwal, B.B.1    Harikumar, K.B.2
  • 22
    • 84867891335 scopus 로고    scopus 로고
    • A randomized, pilot study to assess the efficacy and safety of curcumin in patients with active rheumatoid arthritis
    • Chandran, B., Goel, A., A randomized, pilot study to assess the efficacy and safety of curcumin in patients with active rheumatoid arthritis. Phytother. Res. 26 (2012), 1719–1725.
    • (2012) Phytother. Res. , vol.26 , pp. 1719-1725
    • Chandran, B.1    Goel, A.2
  • 24
    • 0025311288 scopus 로고
    • Epithelial transport of drugs in cell culture. I: a model for studying the passive diffusion of drugs over intestinal absorbtive (Caco-2) cells
    • Artursson, P., Epithelial transport of drugs in cell culture. I: a model for studying the passive diffusion of drugs over intestinal absorbtive (Caco-2) cells. J. Pharm. Sci. 79 (1990), 476–482.
    • (1990) J. Pharm. Sci. , vol.79 , pp. 476-482
    • Artursson, P.1
  • 25
    • 0025804183 scopus 로고
    • Correlation between oral drug absorption in humans and apparent drug permeability coefficients in human intestinal epithelial (Caco-2) cells
    • Artursson, P., Karlsson, J., Correlation between oral drug absorption in humans and apparent drug permeability coefficients in human intestinal epithelial (Caco-2) cells. Biochem. Biophys. Res. Commun. 175 (1991), 880–885.
    • (1991) Biochem. Biophys. Res. Commun. , vol.175 , pp. 880-885
    • Artursson, P.1    Karlsson, J.2
  • 27
    • 0003851111 scopus 로고    scopus 로고
    • Dynamic Light Scattering: With Applications to Chemistry, Biology, and Physics
    • Courier Corporation
    • Berne, B.J., Pecora, R., Dynamic Light Scattering: With Applications to Chemistry, Biology, and Physics. 2000, Courier Corporation.
    • (2000)
    • Berne, B.J.1    Pecora, R.2
  • 28
    • 0006373986 scopus 로고    scopus 로고
    • Small-angle neutron scattering diffractometer at Dhruva reactor
    • Aswal, V., Goyal, P., Small-angle neutron scattering diffractometer at Dhruva reactor. Curr. Sci. 79 (2000), 947–953.
    • (2000) Curr. Sci. , vol.79 , pp. 947-953
    • Aswal, V.1    Goyal, P.2
  • 30
    • 0021061819 scopus 로고
    • Rapid colorimetric assay for cellular growth and survival: application to proliferation and cytotoxicity assays
    • Mosmann, T., Rapid colorimetric assay for cellular growth and survival: application to proliferation and cytotoxicity assays. J. Immunol. methods 65 (1983), 55–63.
    • (1983) J. Immunol. methods , vol.65 , pp. 55-63
    • Mosmann, T.1
  • 31
    • 0024595042 scopus 로고
    • Re-examination and further development of a precise and rapid dye method for measuring cell growth/cell kill
    • Hansen, M.B., Nielsen, S.E., Berg, K., Re-examination and further development of a precise and rapid dye method for measuring cell growth/cell kill. J. Immunol. methods 119 (1989), 203–210.
    • (1989) J. Immunol. methods , vol.119 , pp. 203-210
    • Hansen, M.B.1    Nielsen, S.E.2    Berg, K.3
  • 32
    • 38449084547 scopus 로고    scopus 로고
    • Determination of drug permeability and prediction of drug absorption in Caco-2 monolayers
    • Hubatsch, I., Ragnarsson, E.G., Artursson, P., Determination of drug permeability and prediction of drug absorption in Caco-2 monolayers. Nat. Protoc. 2 (2007), 2111–2119.
    • (2007) Nat. Protoc. , vol.2 , pp. 2111-2119
    • Hubatsch, I.1    Ragnarsson, E.G.2    Artursson, P.3
  • 33
    • 84868556401 scopus 로고    scopus 로고
    • HPLC method for determination of atenolol in human plasma and application to a pharmacokinetic study in Turkey
    • Yilmaz, B., Arslan, S., Asci, A., HPLC method for determination of atenolol in human plasma and application to a pharmacokinetic study in Turkey. J. Chromatogr. Sci. 50 (2012), 914–919.
    • (2012) J. Chromatogr. Sci. , vol.50 , pp. 914-919
    • Yilmaz, B.1    Arslan, S.2    Asci, A.3
  • 34
    • 84897929089 scopus 로고    scopus 로고
    • Development and validation of RP-HPLC method for simultaneous estimation of Clonazepam and propranolol hydrochloride in bulk and pharmaceutical dosage forms
    • Meghana, D., Lahari, K., Kumari, K.S., Prakash, K., Development and validation of RP-HPLC method for simultaneous estimation of Clonazepam and propranolol hydrochloride in bulk and pharmaceutical dosage forms. Invent. Rapid Pharm. Anal. Qual. Assur. 3 (2012), 12–16.
    • (2012) Invent. Rapid Pharm. Anal. Qual. Assur. , vol.3 , pp. 12-16
    • Meghana, D.1    Lahari, K.2    Kumari, K.S.3    Prakash, K.4
  • 35
    • 84882800944 scopus 로고    scopus 로고
    • Simultaneous estimation of curcumin and silibinin using validated RP-HPLC-PDA method and its application in pharmaceutical nanoformulation
    • Moorthi, C., Kathiresan, K., Simultaneous estimation of curcumin and silibinin using validated RP-HPLC-PDA method and its application in pharmaceutical nanoformulation. Int. J. Pharm. Pharm. Sci. 5 (2013), 475–478.
    • (2013) Int. J. Pharm. Pharm. Sci. , vol.5 , pp. 475-478
    • Moorthi, C.1    Kathiresan, K.2
  • 37
    • 84866859325 scopus 로고    scopus 로고
    • Development of a spectrofluorimetric method for the determination of curcumin
    • Gupta, N.K., Nahata, A., Dixit, V.K., Development of a spectrofluorimetric method for the determination of curcumin. Asian J. Trad. Med. 5 (2010), 12–18.
    • (2010) Asian J. Trad. Med. , vol.5 , pp. 12-18
    • Gupta, N.K.1    Nahata, A.2    Dixit, V.K.3
  • 38
    • 85019588729 scopus 로고    scopus 로고
    • Development of a spectrofluorimetric method for the determination of quercetin
    • 亚洲传统医药.
    • S. Srivastava, M. Singh, D. Singh. Development of a spectrofluorimetric method for the determination of quercetin. 亚洲传统医药. 9 136–142.
    • , vol.9 , pp. 136-142
    • Srivastava, S.1    Singh, M.2    Singh, D.3
  • 40
    • 4944245912 scopus 로고    scopus 로고
    • Solubilisation of polyaromatic hydrocarbons in aqueous solutions of poloxamine T803
    • Dong, J., Chowdhry, B.Z., Leharne, S.A., Solubilisation of polyaromatic hydrocarbons in aqueous solutions of poloxamine T803. Colloids Surf. A Physicochem. Eng. Asp. 246 (2004), 91–98.
    • (2004) Colloids Surf. A Physicochem. Eng. Asp. , vol.246 , pp. 91-98
    • Dong, J.1    Chowdhry, B.Z.2    Leharne, S.A.3
  • 41
    • 3543001629 scopus 로고    scopus 로고
    • Thermodynamic modelling of the effect of pH upon aggregation transitions in aqueous solutions of the poloxamine, T701
    • Dong, J., Armstrong, J., Chowdhry, B.Z., Leharne, S.A., Thermodynamic modelling of the effect of pH upon aggregation transitions in aqueous solutions of the poloxamine, T701. Thermochim. acta 417 (2004), 201–206.
    • (2004) Thermochim. acta , vol.417 , pp. 201-206
    • Dong, J.1    Armstrong, J.2    Chowdhry, B.Z.3    Leharne, S.A.4
  • 42
    • 84930674105 scopus 로고    scopus 로고
    • Selective tuning of the self-assembly and gelation of a hydrophilic poloxamine by cyclodextrins
    • González-Gaitano, G., da Silva, M.A., Radulescu, A., Dreiss, C.c.A., Selective tuning of the self-assembly and gelation of a hydrophilic poloxamine by cyclodextrins. Langmuir 31 (2015), 5645–5655.
    • (2015) Langmuir , vol.31 , pp. 5645-5655
    • González-Gaitano, G.1    da Silva, M.A.2    Radulescu, A.3    Dreiss, C.C.A.4
  • 43
    • 0032182194 scopus 로고    scopus 로고
    • Micellar structure of an ethylene oxide-propylene oxide block copolymer: a small-angle neutron scattering study
    • Jain, N.J., Aswal, V., Goyal, P., Bahadur, P., Micellar structure of an ethylene oxide-propylene oxide block copolymer: a small-angle neutron scattering study. J. Phys. Chem. B 102 (1998), 8452–8458.
    • (1998) J. Phys. Chem. B , vol.102 , pp. 8452-8458
    • Jain, N.J.1    Aswal, V.2    Goyal, P.3    Bahadur, P.4
  • 44
    • 0029634549 scopus 로고
    • Solubilization of aromatic solutes in block copolymers
    • Gadelle, F., Koros, W.J., Schechter, R.S., Solubilization of aromatic solutes in block copolymers. Macromolecules 28 (1995), 4883–4892.
    • (1995) Macromolecules , vol.28 , pp. 4883-4892
    • Gadelle, F.1    Koros, W.J.2    Schechter, R.S.3
  • 45
    • 0034652564 scopus 로고    scopus 로고
    • Effect of salts on the micellization, clouding, and solubilization behavior of Pluronic F127 solutions
    • Pandit, N., Trygstad, T., Croy, S., Bohorquez, M., Koch, C., Effect of salts on the micellization, clouding, and solubilization behavior of Pluronic F127 solutions. J. colloid interface Sci. 222 (2000), 213–220.
    • (2000) J. colloid interface Sci. , vol.222 , pp. 213-220
    • Pandit, N.1    Trygstad, T.2    Croy, S.3    Bohorquez, M.4    Koch, C.5
  • 46
    • 0031276732 scopus 로고    scopus 로고
    • Differential scanning calorimetry investigation of the effect of salts on aqueous solution properties of an amphiphilic block copolymer (Poloxamer)
    • Alexandridis, P., Holzwarth, J.F., Differential scanning calorimetry investigation of the effect of salts on aqueous solution properties of an amphiphilic block copolymer (Poloxamer). Langmuir 13 (1997), 6074–6082.
    • (1997) Langmuir , vol.13 , pp. 6074-6082
    • Alexandridis, P.1    Holzwarth, J.F.2
  • 47
    • 0036141804 scopus 로고    scopus 로고
    • The effect of salts on the micellization temperature of aqueous poly (ethylene oxide)-b-poly (propylene oxide)-b-poly (ethylene oxide) solutions and the dissolution rate and water diffusion coefficient in their corresponding gels
    • Anderson, B.C., Cox, S.M., Ambardekar, A.V., Mallapragada, S.K., The effect of salts on the micellization temperature of aqueous poly (ethylene oxide)-b-poly (propylene oxide)-b-poly (ethylene oxide) solutions and the dissolution rate and water diffusion coefficient in their corresponding gels. J. Pharm. Sci. 91 (2002), 180–188.
    • (2002) J. Pharm. Sci. , vol.91 , pp. 180-188
    • Anderson, B.C.1    Cox, S.M.2    Ambardekar, A.V.3    Mallapragada, S.K.4
  • 48
    • 61949094846 scopus 로고    scopus 로고
    • Effect of surfactant mixing on partitioning of model hydrophobic drug, naproxen, between aqueous and micellar phases
    • Bhat, P.A., Rather, G.M., Dar, A.A., Effect of surfactant mixing on partitioning of model hydrophobic drug, naproxen, between aqueous and micellar phases. J. Phys. Chem. B 113 (2009), 997–1006.
    • (2009) J. Phys. Chem. B , vol.113 , pp. 997-1006
    • Bhat, P.A.1    Rather, G.M.2    Dar, A.A.3
  • 49
    • 80051781019 scopus 로고    scopus 로고
    • Solubility of nonsteroidal anti-inflammatory drugs (NSAIDs) in aqueous solutions of non-ionic surfactants
    • Ullah, I., Baloch, M.K., Durrani, G.F., Solubility of nonsteroidal anti-inflammatory drugs (NSAIDs) in aqueous solutions of non-ionic surfactants. J. Solut. Chem. 40 (2011), 1341–1348.
    • (2011) J. Solut. Chem. , vol.40 , pp. 1341-1348
    • Ullah, I.1    Baloch, M.K.2    Durrani, G.F.3
  • 50
    • 0037249698 scopus 로고    scopus 로고
    • Microcalorimetric Evidence and Rheological Consequences of the Salt Effect on Carbopol-surfactant Interactions, Aqueous Polymer—Cosolute Systems
    • Springer
    • Barreiro-Iglesias, R., Alvarez-Lorenzo, C., Concheiro, A., Microcalorimetric Evidence and Rheological Consequences of the Salt Effect on Carbopol-surfactant Interactions, Aqueous Polymer—Cosolute Systems. 2003, Springer, 95–102.
    • (2003) , pp. 95-102
    • Barreiro-Iglesias, R.1    Alvarez-Lorenzo, C.2    Concheiro, A.3
  • 51
    • 0038433339 scopus 로고    scopus 로고
    • The mitochondrial uncoupler dicumarol disrupts the MTT assay
    • Collier, A.C., Pritsos, C.A., The mitochondrial uncoupler dicumarol disrupts the MTT assay. Biochem. Pharmacol. 66 (2003), 281–287.
    • (2003) Biochem. Pharmacol. , vol.66 , pp. 281-287
    • Collier, A.C.1    Pritsos, C.A.2
  • 52
    • 79960974092 scopus 로고    scopus 로고
    • Osteogenic efficiency of in situ gelling poloxamine systems with and without bone morphogenetic protein-2
    • Rey-Rico, A., Silva, M., Couceiro, J., Concheiro, A., Alvarez-Lorenzo, C., Osteogenic efficiency of in situ gelling poloxamine systems with and without bone morphogenetic protein-2. Eur. Cell Mater 21 (2011), 317–340.
    • (2011) Eur. Cell Mater , vol.21 , pp. 317-340
    • Rey-Rico, A.1    Silva, M.2    Couceiro, J.3    Concheiro, A.4    Alvarez-Lorenzo, C.5
  • 53
    • 23644440992 scopus 로고    scopus 로고
    • Semi-synthetic collagen/poloxamine matrices for tissue engineering
    • Sosnik, A., Sefton, M.V., Semi-synthetic collagen/poloxamine matrices for tissue engineering. Biomaterials 26 (2005), 7425–7435.
    • (2005) Biomaterials , vol.26 , pp. 7425-7435
    • Sosnik, A.1    Sefton, M.V.2
  • 54
    • 31044454002 scopus 로고    scopus 로고
    • Collagen/poloxamine hydrogels: cytocompatibility of embedded HepG2 cells and surface-attached endothelial cells
    • Sosnik, A., Leung, B., McGuigan, A.P., Sefton, M.V., Collagen/poloxamine hydrogels: cytocompatibility of embedded HepG2 cells and surface-attached endothelial cells. Tissue Eng. 11 (2005), 1807–1816.
    • (2005) Tissue Eng. , vol.11 , pp. 1807-1816
    • Sosnik, A.1    Leung, B.2    McGuigan, A.P.3    Sefton, M.V.4
  • 55
    • 47049102057 scopus 로고    scopus 로고
    • Lactoyl-poloxamine/collagen matrix for cell-containing tissue engineering modules
    • Sosnik, A., Leung, B.M., Sefton, M.V., Lactoyl-poloxamine/collagen matrix for cell-containing tissue engineering modules. J. Biomed. Mater. Res. Part A 86 (2008), 339–353.
    • (2008) J. Biomed. Mater. Res. Part A , vol.86 , pp. 339-353
    • Sosnik, A.1    Leung, B.M.2    Sefton, M.V.3
  • 56
    • 77955665042 scopus 로고    scopus 로고
    • N-alkylation of poloxamines modulates micellar assembly and encapsulation and release of the antiretroviral efavirenz
    • Chiappetta, D.A., Alvarez-Lorenzo, C., Rey-Rico, A., Taboada, P., Concheiro, A., Sosnik, A., N-alkylation of poloxamines modulates micellar assembly and encapsulation and release of the antiretroviral efavirenz. Eur. J. Pharm. Biopharm. 76 (2010), 24–37.
    • (2010) Eur. J. Pharm. Biopharm. , vol.76 , pp. 24-37
    • Chiappetta, D.A.1    Alvarez-Lorenzo, C.2    Rey-Rico, A.3    Taboada, P.4    Concheiro, A.5    Sosnik, A.6
  • 57
    • 85019558301 scopus 로고    scopus 로고
    • Polymeric Micelles for Formulation of Anti-cancer Drugs, Nanotechnology for Cancer Therapy
    • CRC Press
    • Amiji, M.M., Lim Soo, P., Liu, J., Allen, C., Lee, H., Butler, M., Polymeric Micelles for Formulation of Anti-cancer Drugs, Nanotechnology for Cancer Therapy. 2006, CRC Press, 317–355.
    • (2006) , pp. 317-355
    • Amiji, M.M.1    Lim Soo, P.2    Liu, J.3    Allen, C.4    Lee, H.5    Butler, M.6
  • 58
    • 0030787532 scopus 로고    scopus 로고
    • A human colonic cell line sharing similarities with enterocytes as a model to examine oral absorption: advantages and limitations of the Caco-2 model
    • Delie, F., Rubas, W., A human colonic cell line sharing similarities with enterocytes as a model to examine oral absorption: advantages and limitations of the Caco-2 model. Crit. Reviews™ Ther. Drug Carr. Syst., 14, 1997.
    • (1997) Crit. Reviews™ Ther. Drug Carr. Syst. , vol.14
    • Delie, F.1    Rubas, W.2
  • 59
    • 12244290744 scopus 로고    scopus 로고
    • Towards standardization of an in vitro method of drug absorption
    • Volpe, D., Faustino, P., Yu, L., Hussain, A., Towards standardization of an in vitro method of drug absorption. Pharmacopeial Forum, 2001, 2916–2922.
    • (2001) Pharmacopeial Forum , pp. 2916-2922
    • Volpe, D.1    Faustino, P.2    Yu, L.3    Hussain, A.4
  • 61
    • 0003455057 scopus 로고    scopus 로고
    • Guidance for Industry: Waiver of in Vivo Bioavailability and Bioequivalence Studies for Immediate-release Solid Oral Dosage Forms Based on a Biopharmaceutics Classification System
    • Food and Drug Administration Rockville, MD
    • Food, D. Administration, Guidance for Industry: Waiver of in Vivo Bioavailability and Bioequivalence Studies for Immediate-release Solid Oral Dosage Forms Based on a Biopharmaceutics Classification System. 2000, Food and Drug Administration Rockville, MD.
    • (2000)
    • Food, D. Administration,1
  • 62
    • 0034992583 scopus 로고    scopus 로고
    • Evaluation of human intestinal absorption data and subsequent derivation of a quantitative structure–activity relationship (QSAR) with the Abraham descriptors
    • Zhao, Y.H., Le, J., Abraham, M.H., Hersey, A., Eddershaw, P.J., Luscombe, C.N., Boutina, D., Beck, G., Sherborne, B., Cooper, I., Evaluation of human intestinal absorption data and subsequent derivation of a quantitative structure–activity relationship (QSAR) with the Abraham descriptors. J. Pharm. Sci. 90 (2001), 749–784.
    • (2001) J. Pharm. Sci. , vol.90 , pp. 749-784
    • Zhao, Y.H.1    Le, J.2    Abraham, M.H.3    Hersey, A.4    Eddershaw, P.J.5    Luscombe, C.N.6    Boutina, D.7    Beck, G.8    Sherborne, B.9    Cooper, I.10
  • 63
    • 0031781430 scopus 로고    scopus 로고
    • Correlating partitioning and Caco-2 cell permeability of structurally diverse small molecular weight compounds
    • Yazdanian, M., Glynn, S.L., Wright, J.L., Hawi, A., Correlating partitioning and Caco-2 cell permeability of structurally diverse small molecular weight compounds. Pharm. Res. 15 (1998), 1490–1494.
    • (1998) Pharm. Res. , vol.15 , pp. 1490-1494
    • Yazdanian, M.1    Glynn, S.L.2    Wright, J.L.3    Hawi, A.4
  • 64
    • 19944388360 scopus 로고    scopus 로고
    • Permeability classification of representative fluoroquinolones by a cell culture method
    • Volpe, D.A., Permeability classification of representative fluoroquinolones by a cell culture method. AAPS PharmSci. 6 (2004), 1–6.
    • (2004) AAPS PharmSci. , vol.6 , pp. 1-6
    • Volpe, D.A.1
  • 66
    • 0037467170 scopus 로고    scopus 로고
    • Microcrystals for dissolution rate enhancement of poorly water-soluble drugs
    • Rasenack, N., Hartenhauer, H., Müller, B.W., Microcrystals for dissolution rate enhancement of poorly water-soluble drugs. Int. J. Pharm. 254 (2003), 137–145.
    • (2003) Int. J. Pharm. , vol.254 , pp. 137-145
    • Rasenack, N.1    Hartenhauer, H.2    Müller, B.W.3
  • 67
    • 33846234714 scopus 로고    scopus 로고
    • Curcumin–phospholipid complex: preparation, therapeutic evaluation and pharmacokinetic study in rats
    • Maiti, K., Mukherjee, K., Gantait, A., Saha, B.P., Mukherjee, P.K., Curcumin–phospholipid complex: preparation, therapeutic evaluation and pharmacokinetic study in rats. Int. J. Pharm. 330 (2007), 155–163.
    • (2007) Int. J. Pharm. , vol.330 , pp. 155-163
    • Maiti, K.1    Mukherjee, K.2    Gantait, A.3    Saha, B.P.4    Mukherjee, P.K.5
  • 68
    • 84925501129 scopus 로고    scopus 로고
    • Pharmacokinetic Study of Nanoparticulate Curcumin: Oral Formulation for Enhanced Bioavailability
    • Ravichandran, R., Pharmacokinetic Study of Nanoparticulate Curcumin: Oral Formulation for Enhanced Bioavailability. 2013.
    • (2013)
    • Ravichandran, R.1
  • 69
    • 0035940059 scopus 로고    scopus 로고
    • Recent advances in the understanding of uptake of microparticulates across the gastrointestinal lymphatics
    • Hussain, N., Jaitley, V., Florence, A.T., Recent advances in the understanding of uptake of microparticulates across the gastrointestinal lymphatics. Adv. drug Deliv. Rev. 50 (2001), 107–142.
    • (2001) Adv. drug Deliv. Rev. , vol.50 , pp. 107-142
    • Hussain, N.1    Jaitley, V.2    Florence, A.T.3
  • 70
    • 0033977066 scopus 로고    scopus 로고
    • A new liposomal formulation for antisense oligodeoxynucleotides with small size, high incorporation efficiency and good stability
    • Stuart, D., Allen, T., A new liposomal formulation for antisense oligodeoxynucleotides with small size, high incorporation efficiency and good stability. Biochim. Biophys. Acta (BBA)-Biomembr. 1463 (2000), 219–229.
    • (2000) Biochim. Biophys. Acta (BBA)-Biomembr. , vol.1463 , pp. 219-229
    • Stuart, D.1    Allen, T.2
  • 71
    • 1842684453 scopus 로고    scopus 로고
    • Self-emulsifying drug delivery systems (SEDDS) for improved oral delivery of lipophilic drugs
    • Gursoy, R.N., Benita, S., Self-emulsifying drug delivery systems (SEDDS) for improved oral delivery of lipophilic drugs. Biomed. Pharmacother. 58 (2004), 173–182.
    • (2004) Biomed. Pharmacother. , vol.58 , pp. 173-182
    • Gursoy, R.N.1    Benita, S.2
  • 72
    • 7444255422 scopus 로고    scopus 로고
    • Altered chemical and biological activities of all-trans retinoic acid incorporated in solid lipid nanoparticle powders
    • Lim, S.-J., Lee, M.-K., Kim, C.-K., Altered chemical and biological activities of all-trans retinoic acid incorporated in solid lipid nanoparticle powders. J. Control. release 100 (2004), 53–61.
    • (2004) J. Control. release , vol.100 , pp. 53-61
    • Lim, S.-J.1    Lee, M.-K.2    Kim, C.-K.3
  • 74
    • 67349107075 scopus 로고    scopus 로고
    • Nanoparticle encapsulation improves oral bioavailability of curcumin by at least 9-fold when compared to curcumin administered with piperine as absorption enhancer
    • Shaikh, J., Ankola, D., Beniwal, V., Singh, D., Kumar, M.R., Nanoparticle encapsulation improves oral bioavailability of curcumin by at least 9-fold when compared to curcumin administered with piperine as absorption enhancer. Eur. J. Pharm. Sci. 37 (2009), 223–230.
    • (2009) Eur. J. Pharm. Sci. , vol.37 , pp. 223-230
    • Shaikh, J.1    Ankola, D.2    Beniwal, V.3    Singh, D.4    Kumar, M.R.5
  • 75
    • 34248549039 scopus 로고    scopus 로고
    • Formulation and characterization of curcuminoids loaded solid lipid nanoparticles
    • Tiyaboonchai, W., Tungpradit, W., Plianbangchang, P., Formulation and characterization of curcuminoids loaded solid lipid nanoparticles. Int. J. Pharm. 337 (2007), 299–306.
    • (2007) Int. J. Pharm. , vol.337 , pp. 299-306
    • Tiyaboonchai, W.1    Tungpradit, W.2    Plianbangchang, P.3
  • 77
    • 84862992759 scopus 로고    scopus 로고
    • Comparative oral bioavailability advantage from curcumin formulations
    • Munjal, B., Pawar, Y.B., Patel, S.B., Bansal, A.K., Comparative oral bioavailability advantage from curcumin formulations. Drug Deliv. Transl. Res. 1 (2011), 322–331.
    • (2011) Drug Deliv. Transl. Res. , vol.1 , pp. 322-331
    • Munjal, B.1    Pawar, Y.B.2    Patel, S.B.3    Bansal, A.K.4
  • 78
    • 76649085489 scopus 로고    scopus 로고
    • Significance of protein binding in pharmacokinetics and pharmacodynamics
    • Schmidt, S., Gonzalez, D., Derendorf, H., Significance of protein binding in pharmacokinetics and pharmacodynamics. J. Pharm. Sci. 99 (2010), 1107–1122.
    • (2010) J. Pharm. Sci. , vol.99 , pp. 1107-1122
    • Schmidt, S.1    Gonzalez, D.2    Derendorf, H.3
  • 79
    • 84992393684 scopus 로고    scopus 로고
    • Pharmacokinetic comparison between quercetin and quercetin 3-O-β-glucuronide in rats by UHPLC-MS/MS
    • Yang, L.-L., Xiao, N., Li, X.-W., Fan, Y., Alolga, R.N., Sun, X.-Y., Wang, S.-L., Li, P., Qi, L.-W., Pharmacokinetic comparison between quercetin and quercetin 3-O-β-glucuronide in rats by UHPLC-MS/MS. Sci. Rep., 6, 2016, 35460.
    • (2016) Sci. Rep. , vol.6 , pp. 35460
    • Yang, L.-L.1    Xiao, N.2    Li, X.-W.3    Fan, Y.4    Alolga, R.N.5    Sun, X.-Y.6    Wang, S.-L.7    Li, P.8    Qi, L.-W.9
  • 80
    • 84933525096 scopus 로고    scopus 로고
    • Poly (n-butylcyanoacrylate) nanoparticles for oral delivery of quercetin: preparation, characterization, and pharmacokinetics and biodistribution studies in Wistar rats
    • Bagad, M., Khan, Z.A., Poly (n-butylcyanoacrylate) nanoparticles for oral delivery of quercetin: preparation, characterization, and pharmacokinetics and biodistribution studies in Wistar rats. Int. J. Nanomed., 10, 2015, 3921.
    • (2015) Int. J. Nanomed. , vol.10 , pp. 3921
    • Bagad, M.1    Khan, Z.A.2
  • 81
    • 84867102456 scopus 로고    scopus 로고
    • Influence of the preparation method on the physicochemical properties of econazole-loaded poly (butyl cyanoacrylate) colloidal nanoparticles
    • Yordanov, G., Influence of the preparation method on the physicochemical properties of econazole-loaded poly (butyl cyanoacrylate) colloidal nanoparticles. Colloids Surf. A Physicochem. Eng. Asp. 413 (2012), 260–265.
    • (2012) Colloids Surf. A Physicochem. Eng. Asp. , vol.413 , pp. 260-265
    • Yordanov, G.1
  • 82
    • 79960297652 scopus 로고    scopus 로고
    • Enhanced brain targeting of temozolomide in polysorbate-80 coated polybutylcyanoacrylate nanoparticles
    • Tian, X.-h., Lin, X.-N., Wei, F., Feng, W., Huang, Z.-C., Wang, P., Ren, L., Diao, Y., Enhanced brain targeting of temozolomide in polysorbate-80 coated polybutylcyanoacrylate nanoparticles. Int. J. Nanomed. 6 (2011), 445–452.
    • (2011) Int. J. Nanomed. , vol.6 , pp. 445-452
    • Tian, X.-H.1    Lin, X.-N.2    Wei, F.3    Feng, W.4    Huang, Z.-C.5    Wang, P.6    Ren, L.7    Diao, Y.8


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.